Discovery of a Selective and Potent Inhibitor of Cyclin-Dependent Kinase 12/13 Employing a Noncovalent Mechanism
利用非共价机制发现一种选择性强、高效的细胞周期蛋白依赖性激酶12/13抑制剂
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.5c00743
Swyka, Robert A; Styduhar, Evan D; Wang, Anlai; Li, Xin; Zhang, Ke; Witten, Michael R; Zhao, Peng; Liang, Michael Z; Atasoylu, Onur; He, Peng; Soderquist, Ryan; Hansbury, Mike; Huo, Lu; Chen, Haiying; Zimmer, Derek; Zhang, Wenliang; Wang, Kathy; Volgina, Alla; Epling, Leslie B; Crowgey, Erin; Kumari, Ekta; Abdollahi, Angela; Zhang, Guofeng; Rupar, Mark; Schaffer, Michael; Mayes, Patrick A; Kim, Sunkyu; Vechorkin, Oleg; Wang, Xiaozhao