日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

SAG1.3-derived Frizzled-targeting small-molecule compounds.

源自 SAG1.3 的 Frizzled 靶向小分子化合物。

Grätz Lukas, Turku Ainoleena, Kozielewicz Pawel, Bowin Carl-Fredrik, Scharf Magdalena M, Voss Jan H, Kinsolving Julia, Shekhani Rawan, Oliva-Vilarnau Nuria, Koolmeister Tobias, Körber Marlies, Lauschke Volker M, Löber Stefan, Gmeiner Peter, Schulte Gunnar

Crystal structure of adenosine A(2A) receptor in complex with clinical candidate Etrumadenant reveals unprecedented antagonist interaction.

腺苷 A(2A) 受体与临床候选药物 Etrumadenant 复合物的晶体结构揭示了前所未有的拮抗剂相互作用

Claff Tobias, Schlegel Jonathan G, Voss Jan H, Vaaßen Victoria J, Weiße Renato H, Cheng Robert K Y, Markovic-Mueller Sandra, Bucher Denis, Sträter Norbert, Müller Christa E

Structure-affinity and structure-residence time relationships of macrocyclic Gα(q) protein inhibitors

大环Gα(q)蛋白抑制剂的结构亲和力和结构停留时间关系

Voss, Jan H; Crüsemann, Max; Bartling, Christian R O; Kehraus, Stefan; Inoue, Asuka; König, Gabriele M; Strømgaard, Kristian; Müller, Christa E

Imaging of Gα(q) Proteins in Mouse and Human Organs and Tissues

小鼠和人类器官及组织中Gα(q)蛋白的成像

Voss, Jan H; Al-Hroub, Haneen; Gedschold, Robin; Dietrich, Jennifer M; Gaffal, Evelyn; Toma, Marieta; Kehraus, Stefan; König, Gabriele M; Brust, Peter; Fleischmann, Bernd K; Wenzel, Daniela; Deuther-Conrad, Winnie; Müller, Christa E

Macrocyclic Gq Protein Inhibitors FR900359 and/or YM-254890-Fit for Translation?

大环Gq蛋白抑制剂FR900359和/或YM-254890——适合翻译吗?

Schlegel, Jonathan G; Tahoun, Mariam; Seidinger, Alexander; Voss, Jan H; Kuschak, Markus; Kehraus, Stefan; Schneider, Marion; Matthey, Michaela; Fleischmann, Bernd K; König, Gabriele M; Wenzel, Daniela; Müller, Christa E

Sensitive LC-MS/MS Method for the Quantification of Macrocyclic Gα(q) Protein Inhibitors in Biological Samples

用于定量分析生物样品中大环Gα(q)蛋白抑制剂的灵敏LC-MS/MS方法

Kuschak, Markus; Schlegel, Jonathan G; Schneider, Marion; Kehraus, Stefan; Voss, Jan H; Seidinger, Alexander; Matthey, Michaela; Wenzel, Daniela; Fleischmann, Bernd K; König, Gabriele M; Müller, Christa E