日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Fragment-based discovery enables direct targeting of the melanoma oncogene MITF

基于片段的发现能够直接靶向黑色素瘤癌基因MITF。

Castelletti, Deborah; Hinrichs, Jürgen; Malojčić, Goran; Ji, Fei; Desplat, Aurore; Reimer, Bryn; Henry, Christelle; Porter, Kathryn A; Mermet-Meillon, Fanny; Wartmann, Markus; Wirth, Emmanuelle; Delmas, Cécile; Fernández, César; Mayer, Philipp H O; Schmiedeberg, Niko; Plattner, Simone; Brun, Jvan; Kläusler, Stephan; Kurmann, Jessica; Yan, Kelly; Fuller, John; Schaeffer, Fanny; Maddalo, Danilo; Altorfer, Marc; Piperidou, Nikoletta; Pautrieux, Nicolas; Baysang, Frederic; Kaufmann, Markus; Cobos-Correa, Amanda; Wilcken, Rainer; Renatus, Martin; Vulpetti, Anna; Jahnke, Wolfgang

Combined Surgically Induced Macular Detachment and Autologous Internal Limiting Membrane Transplantation for Refractory Full Thickness Macular Hole

手术诱导黄斑脱离联合自体内界膜移植治疗难治性全层黄斑裂孔

Frisina, Rino; Di Leo, Laura; Gallo Afflitto, Ilenia; Vulpetti, Andrea; Motta, Lorenzo; De Salvo, Gabriella

Author Correction: DCAF1-based PROTACs with activity against clinically validated targets overcoming intrinsic- and acquired-degrader resistance

作者更正:基于 DCAF1 的 PROTAC 具有针对临床验证靶点的活性,可克服内在和获得性降解剂耐药性。

Schröder, Martin; Renatus, Martin; Liang, Xiaoyou; Meili, Fabian; Zoller, Thomas; Ferrand, Sandrine; Gauter, Francois; Li, Xiaoyan; Sigoillot, Frederic; Gleim, Scott; Stachyra, Therese-Marie; Thomas, Jason R; Begue, Damien; Khoshouei, Maryam; Lefeuvre, Peggy; Andraos-Rey, Rita; Chung, BoYee; Ma, Renate; Pinch, Benika; Hofmann, Andreas; Schirle, Markus; Schmiedeberg, Niko; Imbach, Patricia; Gorses, Delphine; Calkins, Keith; Bauer-Probst, Beatrice; Maschlej, Magdalena; Niederst, Matt; Maher, Rob; Henault, Martin; Alford, John; Ahrne, Erik; Tordella, Luca; Hollingworth, Greg; Thomä, Nicolas H; Vulpetti, Anna; Radimerski, Thomas; Holzer, Philipp; Carbonneau, Seth; Thoma, Claudio R

Flexor Tendon Continuity and Negative X-ray: The "Combo" Negative Features in Finger Subamputation

屈肌腱连续性和X光片阴性:手指部分截肢中的“组合”阴性特征

Pugliese, Pierfrancesco; Vulpetti, Mariangela; Tondini, Greta; Toia, Francesca

Discovery of a selective and biologically active low-molecular weight antagonist of human interleukin-1β

发现一种具有选择性和生物活性的低分子量人类白细胞介素-1β 拮抗剂

Ulrich Hommel, Konstanze Hurth, Jean-Michel Rondeau, Anna Vulpetti, Daniela Ostermeier, Andreas Boettcher, Jacob Peter Brady, Michael Hediger, Sylvie Lehmann, Elke Koch, Anke Blechschmidt, Rina Yamamoto, Valentina Tundo Dottorello, Sandra Haenni-Holzinger, Christian Kaiser, Philipp Lehr, Andreas Lin

Discovery of Ligands for TRIM58, a Novel Tissue-Selective E3 Ligase

发现新型组织选择性E3连接酶TRIM58的配体

Hoegenauer, Klemens; An, Shaojian; Axford, Jake; Benander, Christina; Bergsdorf, Christian; Botsch, Josephine; Chau, Suzanne; Fernández, César; Gleim, Scott; Hassiepen, Ulrich; Hunziker, Juerg; Joly, Emilie; Keller, Aramis; Lopez Romero, Sandra; Maher, Robert; Mangold, Anne-Sophie; Mickanin, Craig; Mihalic, Manuel; Neuner, Philippe; Patterson, Andrew W; Perruccio, Francesca; Roggo, Silvio; Scesa, Julien; Schröder, Martin; Shkoza, Dojna; Thai, Binh; Vulpetti, Anna; Renatus, Martin; Reece-Hoyes, John S

Discovery of New Binders for DCAF1, an Emerging Ligase Target in the Targeted Protein Degradation Field

在靶向蛋白降解领域,发现了一种新兴的连接酶靶点——DCAF1 的新型结合剂。

Vulpetti, Anna; Holzer, Philipp; Schmiedeberg, Niko; Imbach-Weese, Patricia; Pissot-Soldermann, Carole; Hollingworth, Gregory J; Radimerski, Thomas; Thoma, Claudio R; Stachyra, Therese-Marie; Wojtynek, Matthias; Maschlej, Magdalena; Chau, Suzanne; Schuffenhauer, Ansgar; Fernández, César; Schröder, Martin; Renatus, Martin

Design of Potent and Selective Covalent Inhibitors of Bruton's Tyrosine Kinase Targeting an Inactive Conformation

针对布鲁顿酪氨酸激酶非活性构象设计高效选择性共价抑制剂

Pulz, Robert; Angst, Daniela; Dawson, Janet; Gessier, Francois; Gutmann, Sascha; Hersperger, Rene; Hinniger, Alexandra; Janser, Philipp; Koch, Guido; Revesz, Laszlo; Vulpetti, Anna; Waelchli, Rudolf; Zimmerlin, Alfred; Cenni, Bruno

Discovery and Design of First Benzylamine-Based Ligands Binding to an Unlocked Conformation of the Complement Factor D

发现并设计了首批与补体因子D的未锁定构象结合的苄胺基配体

Vulpetti, Anna; Ostermann, Nils; Randl, Stefan; Yoon, Taeyoung; Mac Sweeney, Aengus; Cumin, Frederic; Lorthiois, Edwige; Rüdisser, Simon; Erbel, Paul; Maibaum, Jürgen