日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Optimization of Prodiginines as Single-Dose Curative Antimalarials

优化灵菌红素类药物作为单剂量治愈性抗疟药

Kumar, Amrendra; Li, Yuexin; Zhang, Xiaowei; Gaddam, Mahesh; Caridha, Diana; Madejczyk, Michael S; Jin, Xiannu; Dennis, William E; Chetree, Ravi; Blount, Cameron; DeLuca, Jesse; Vuong, Chau; Kudyba, Karl; Roncal, Norma; Ashraf, Kutub; Lee, Patricia J; Pannone, Kristina; Leed, Susan; Dinh, Hieu T; Mdaki, Kennedy; Navarrete, Kimberly; Charlton, Jordan; Binauhan, Angely J; Qahash, Tarrick; Kibe, Kevin Mugambi; Shoue, Douglas A; Checkley, Lisa; Ferdig, Michael T; Chim-Ong, Anongruk; Cui, Liwang; Orena, Stephen; Byaruhanga, Oswald; Assimwe, Jackson; Tibagambirwa, Innocent; Chithanna, Sivanna; Dodean, Rozalia A; Legac, Jennifer; Kreutzfeld, Oriana; Rosenthal, Philip J; Cooper, Roland A; Reynolds, Kevin A; Roth, Alison; Kelly, Jane X; Kancharla, Papireddy

Acridone Prodrugs with Enhanced Dual-Stage Antimalarial Efficacy

具有增强双阶段抗疟功效的吖啶酮前药

Dodean, Rozalia A; Li, Yuexin; Zhang, Xiaowei; Kumar, Amrendra; Pou, Sovitj; W Winter, Rolf; Liebman, Katherine M; Zakharov, Lev N; Caridha, Diana; Madejczyk, Michael S; Vuong, Chau; DeLuca, Jesse; Chin, Geoffrey; Kudyba, Karl; McEnearney, Sharon; Jin, Xiannu; Dennis, William E; Chetree, Ravi; Blount, Cameron; Pannone, Kristina; Dinh, Hieu T; Mdaki, Kennedy; Leed, Susan; Lee, Patricia J; Roth, Alison; Kancharla, Papireddy; Kelly, Jane X

DDDR-05. SPATIALLY RESOLVED DRUG SENSITIVITY PROFILING IN GLIOBLASTOMA

DDDR-05. 胶质母细胞瘤的空间分辨药物敏感性分析

Kumar, Amrendra; Li, Yuexin; Dodean, Rozalia A; Roth, Alison; Caridha, Diana; Madejczyk, Michael S; Jin, Xiannu; Dennis, William E; Lee, Patricia J; Pybus, Brandon S; Martin, Monica; Pannone, Kristina; Dinh, Hieu T; Blount, Cameron; Chetree, Ravi; DeLuca, Jesse; Evans, Martin; Nadeau, Robert; Vuong, Chau; Leed, Susan; Black, Chad; Sousa, Jason; Nolan, Christina; Ceja, Frida G; Rasmussen, Stephanie A; Tumwebaze, Patrick K; Rosenthal, Philip J; Cooper, Roland A; Rottmann, Matthias; Orjuela-Sanchez, Pamela; Meister, Stephan; Winzeler, Elizabeth A; Delves, Michael J; Matthews, Holly; Baum, Jake; Kirby, Robert W; Burrows, Jeremy N; Duffy, James; Peyton, David H; Reynolds, Kevin A; Kelly, Jane X; Kancharla, Papireddy; Buck, Alicia; Lee, Sohyon; Wegmann, Rebekka; Mena, Julien; Vasella, Flavio; Friesen, Julia; Regli, Luca; Le Rhun, Emilie; Zeitlberger, Anna Maria; Neidert, Marian Christoph; Tatari, Nazanin; Hutter, Gregor; Weller, Michael; Snijder, Berend; Weiss, Tobias

Author Correction: Homologous Pairs of Low and High Temperature Originating Proteins Spanning the Known Prokaryotic Universe

作者更正:已知原核生物宇宙中起源于低温和高温的同源蛋白对

Komp, Evan; Alanzi, Humood N; Francis, Ryan; Vuong, Chau; Roberts, Logan; Mosallanejad, Amin; Beck, David A C

Plasma Blood Levels of Tafenoquine following a Single Oral Dosage in BALBc Mice with Acute Babesia microti Infection That Resulted in Rapid Clearance of Microscopically Detectable Parasitemia

单次口服他非诺喹后,BALBc 小鼠急性巴贝虫感染后血浆中他非诺喹的浓度迅速降低,显微镜下可检测到的寄生虫血症也迅速消失。

Mordue, Dana G; Hale, Synthia J; Dennis, William E; Vuong, Chau V; Li, Xiu-Min; Yang, Nan; Wormser, Gary P

An Iterative Approach Guides Discovery of the FabI Inhibitor Fabimycin, a Late-Stage Antibiotic Candidate with In Vivo Efficacy against Drug-Resistant Gram-Negative Infections

迭代方法指导FabI抑制剂法比霉素的发现,法比霉素是一种后期抗生素候选药物,对耐药革兰氏阴性菌感染具有体内疗效。

Parker, Erica N; Cain, Brett N; Hajian, Behnoush; Ulrich, Rebecca J; Geddes, Emily J; Barkho, Sulyman; Lee, Hyang Yeon; Williams, John D; Raynor, Malik; Caridha, Diana; Zaino, Angela; Shekhar, Mrinal; Muñoz, Kristen A; Rzasa, Kara M; Temple, Emily R; Hunt, Diana; Jin, Xiannu; Vuong, Chau; Pannone, Kristina; Kelly, Aya M; Mulligan, Michael P; Lee, Katie K; Lau, Gee W; Hung, Deborah T; Hergenrother, Paul J

Correction to "An Iterative Approach Guides Discovery of the FabI Inhibitor Fabimycin, a Late-Stage Antibiotic Candidate with In Vivo Efficacy against Drug-Resistant Gram-Negative Infections"

对“迭代方法指导发现FabI抑制剂法比霉素,一种对耐药革兰氏阴性菌感染具有体内疗效的后期抗生素候选药物”一文的更正

Parker, Erica N; Cain, Brett N; Hajian, Behnoush; Ulrich, Rebecca J; Geddes, Emily J; Barkho, Sulyman; Lee, Hyang Yeon; Williams, John D; Raynor, Malik; Caridha, Diana; Zaino, Angela; Rohde, Jason M; Zak, Mark; Shekhar, Mrinal; Muñoz, Kristen A; Rzasa, Kara M; Temple, Emily R; Hunt, Diana; Jin, Xiannu; Vuong, Chau; Pannone, Kristina; Kelly, Aya M; Mulligan, Michael P; Lee, Katie K; Lau, Gee W; Hung, Deborah T; Hergenrother, Paul J

An open label study of the safety and efficacy of a single dose of weekly chloroquine and azithromycin administered for malaria prophylaxis in healthy adults challenged with 7G8 chloroquine-resistant Plasmodium falciparum in a controlled human malaria infection model

一项开放标签研究,旨在评估每周一次单剂量氯喹和阿奇霉素用于预防疟疾的安全性和有效性,研究对象为在受控的人类疟疾感染模型中感染7G8氯喹耐药恶性疟原虫的健康成年人。

Livezey, Jeffrey; Twomey, Patrick; Morrison, Meshell; Cicatelli, Susan; Duncan, Elizabeth H; Hamer, Melinda; Lee, Christine; Hutter, Jack; Mills, Kristin; DeLuca, Jesse; Poon, Lucas; Selig, Daniel; Vuong, Chau; Sousa, Jason; Oliver, Thomas; Bennett, Jason; Moon, James E; Sikaffy, April; Sedegah, Martha; Tosh, Donna; Kreishman-Deitrick, Mara; Waterman, Paige

Single-Dose Primaquine in a Preclinical Model of Glucose-6-Phosphate Dehydrogenase Deficiency: Implications for Use in Malaria Transmission-Blocking Programs

单剂量伯氨喹在葡萄糖-6-磷酸脱氢酶缺乏症临床前模型中的应用:对疟疾传播阻断计划的意义

Wickham, Kristina S; Baresel, Paul C; Marcsisin, Sean R; Sousa, Jason; Vuong, Chau T; Reichard, Gregory A; Campo, Brice; Tekwani, Babu L; Walker, Larry A; Rochford, Rosemary

Differential CYP 2D6 metabolism alters primaquine pharmacokinetics

CYP 2D6 代谢差异会改变伯氨喹的药代动力学

Potter, Brittney M J; Xie, Lisa H; Vuong, Chau; Zhang, Jing; Zhang, Ping; Duan, Dehui; Luong, Thu-Lan T; Bandara Herath, H M T; Dhammika Nanayakkara, N P; Tekwani, Babu L; Walker, Larry A; Nolan, Christina K; Sciotti, Richard J; Zottig, Victor E; Smith, Philip L; Paris, Robert M; Read, Lisa T; Li, Qigui; Pybus, Brandon S; Sousa, Jason C; Reichard, Gregory A; Marcsisin, Sean R