日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Synthesis of Biotinylated PAMAM G3 Dendrimers Substituted with R-Glycidol and Celecoxib/Simvastatin as Repurposed Drugs and Evaluation of Their Increased Additive Cytotoxicity for Cancer Cell Lines

合成生物素化 PAMAM G3 树枝状聚合物(用 R-缩水甘油和塞来昔布/辛伐他汀取代)作为再利用药物,并评估其对癌细胞系增加的附加细胞毒性

Konrad Wróbel, Stanisław Wołowiec, Joanna Markowicz, Elżbieta Wałajtys-Rode, Łukasz Uram

The Effect of Biotinylated PAMAM G3 Dendrimers Conjugated with COX-2 Inhibitor (celecoxib) and PPARγ Agonist (Fmoc-L-Leucine) on Human Normal Fibroblasts, Immortalized Keratinocytes and Glioma Cells in Vitro

生物素化的 PAMAM G3 树枝状聚合物与 COX-2 抑制剂 (塞来昔布) 和 PPARγ 激动剂 (Fmoc-L-亮氨酸) 结合对人正常成纤维细胞、永生化角质形成细胞和胶质瘤细胞体外的影响

Łukasz Uram, Maria Misiorek, Monika Pichla, Aleksandra Filipowicz-Rachwał, Joanna Markowicz, Stanisław Wołowiec, Elżbieta Wałajtys-Rode

Different patterns of nuclear and mitochondrial penetration by the G3 PAMAM dendrimer and its biotin-pyridoxal bioconjugate BC-PAMAM in normal and cancer cells in vitro

体外实验表明,G3 PAMAM 树状聚合物及其生物素-吡哆醛生物缀合物 BC-PAMAM 在正常细胞和癌细胞中具有不同的核和线粒体穿透模式。

Uram, Łukasz; Szuster, Magdalena; Filipowicz, Aleksandra; Gargasz, Krzysztof; Wołowiec, Stanisław; Wałajtys-Rode, Elżbieta

In vitro cytotoxicity of the ternary PAMAM G3-pyridoxal-biotin bioconjugate

PAMAM G3-吡哆醛-生物素三元生物缀合物的体外细胞毒性

Uram, Łukasz; Szuster, Magdalena; Gargasz, Krzysztof; Filipowicz, Aleksandra; Wałajtys-Rode, Elżbieta; Wołowiec, Stanisław