日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification of small molecule inhibitors of PPM1D using an integrated drug discovery platform.

利用综合药物发现平台鉴定PPM1D小分子抑制剂

Shaw Subrata, Jiang Wei, Rush Jason, Dumont Nancy, Kim John, Singh Ritu, Skepner Adam, Khodier Carol, Raffier Cerise, Murphy Zachary, Yan Ni, Schluter Cameron, Yu Xiao, Szuchnicki Mateusz, Sathappa Murugappan, Kahn Josephine, Sperling Adam S, Wagner Florence, McKinney David C, Gould Alexandra E, Garvie Colin W, Miller Peter G

Developmental Selective GSK3α Inhibition Rescues Working Memory Deficits in a Mouse Model of Schizophrenia Predisposition

发育选择性 GSK3α 抑制可挽救精神分裂症易感小鼠模型的工作记忆缺陷

Passecker, Johannes; Aloimonos, Chloe M; Dagunts, Aleksandra; Wagner, Florence F; Kupferschmidt, David A; Gogos, Joseph; Gordon, Joshua A

A Fast-Binding, Functionally Reversible, COX-2 Radiotracer for CNS PET Imaging

一种用于中枢神经系统PET成像的快速结合、功能可逆的COX-2放射性示踪剂

Placzek, Michael S; Wilton, Daniel K; Weïwer, Michel; Manter, Mariah A; Reid, Sarah E; Meyer, Christopher J; Campbell, Arthur J; Bajrami, Besnik; Bigot, Antoine; Bricault, Sarah; Fayet, Agathe; Frouin, Arnaud; Gergits, Frederick; Gupta, Mehak; Jiang, Wei; Melanson, Michelle; Romano, Chiara D; Riley, Misha M; Wang, Jessica M; Wey, Hsiao-Ying; Wagner, Florence F; Stevens, Beth; Hooker, Jacob M

HDAC2 targeting stabilizes the CoREST complex in renal tubular cells and protects against renal ischemia/reperfusion injury

靶向 HDAC2 可稳定肾小管细胞中的 CoREST 复合物,并保护肾脏免受缺血/再灌注损伤。

Aufhauser, David D Jr; Hernandez, Paul; Concors, Seth J; O'Brien, Ciaran; Wang, Zhonglin; Murken, Douglas R; Samanta, Arabinda; Beier, Ulf H; Krumeich, Lauren; Bhatti, Tricia R; Wang, Yanfeng; Ge, Guanghui; Wang, Liqing; Cheraghlou, Shayan; Wagner, Florence F; Holson, Edward B; Kalin, Jay H; Cole, Philip A; Hancock, Wayne W; Levine, Matthew H

MISCAST: MIssense variant to protein StruCture Analysis web SuiTe

错配:蛋白质结构分析网络套件的错义变体

Iqbal, Sumaiya; Hoksza, David; Pérez-Palma, Eduardo; May, Patrick; Jespersen, Jakob B; Ahmed, Shehab S; Rifat, Zaara T; Heyne, Henrike O; Rahman, M Sohel; Cottrell, Jeffrey R; Wagner, Florence F; Daly, Mark J; Campbell, Arthur J; Lal, Dennis

Comprehensive characterization of amino acid positions in protein structures reveals molecular effect of missense variants

对蛋白质结构中氨基酸位置的全面表征揭示了错义变异的分子效应

Iqbal, Sumaiya; Pérez-Palma, Eduardo; Jespersen, Jakob B; May, Patrick; Hoksza, David; Heyne, Henrike O; Ahmed, Shehab S; Rifat, Zaara T; Rahman, M Sohel; Lage, Kasper; Palotie, Aarno; Cottrell, Jeffrey R; Wagner, Florence F; Daly, Mark J; Campbell, Arthur J; Lal, Dennis

Translation of HDAC6 PET Imaging Using [(18)F]EKZ-001-cGMP Production and Measurement of HDAC6 Target Occupancy in Nonhuman Primates

利用[(18)F]EKZ-001-cGMP生产进行HDAC6 PET成像,并测量非人灵长类动物中HDAC6靶点占有率

Celen, Sofie; Rokka, Johanna; Gilbert, Tonya M; Koole, Michel; Vermeulen, Isabeau; Serdons, Kim; Schroeder, Frederick A; Wagner, Florence F; Bleeser, Tom; Hightower, Baileigh G; Hu, Jiyun; Rahal, Dania; Beyzavi, Hudson; Vanduffel, Wim; Van Laere, Koen; Kranz, Janice E; Hooker, Jacob M; Bormans, Guy; Cawthorne, Christopher J

Dynamic architecture of the Escherichia coli structural maintenance of chromosomes (SMC) complex, MukBEF

大肠杆菌染色体结构维持(SMC)复合物的动态结构,MukBEF

Rajasekar, Karthik V; Baker, Rachel; Fisher, Gemma L M; Bolla, Jani R; Mäkelä, Jarno; Tang, Minzhe; Zawadzka, Katarzyna; Koczy, Oliwia; Wagner, Florence; Robinson, Carol V; Arciszewska, Lidia K; Sherratt, David J

Progress in Understanding and Treating SCN2A-Mediated Disorders

对SCN2A介导疾病的理解和治疗进展

Sanders, Stephan J; Campbell, Arthur J; Cottrell, Jeffrey R; Moller, Rikke S; Wagner, Florence F; Auldridge, Angie L; Bernier, Raphael A; Catterall, William A; Chung, Wendy K; Empfield, James R; George, Alfred L Jr; Hipp, Joerg F; Khwaja, Omar; Kiskinis, Evangelos; Lal, Dennis; Malhotra, Dheeraj; Millichap, John J; Otis, Thomas S; Petrou, Steven; Pitt, Geoffrey; Schust, Leah F; Taylor, Cora M; Tjernagel, Jennifer; Spiro, John E; Bender, Kevin J

Entropy as a Driver of Selectivity for Inhibitor Binding to Histone Deacetylase 6

熵作为抑制剂与组蛋白去乙酰化酶6结合选择性的驱动因素

Porter, Nicholas J; Wagner, Florence F; Christianson, David W