日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Developmental Selective GSK3α Inhibition Rescues Working Memory Deficits in a Mouse Model of Schizophrenia Predisposition

发育选择性 GSK3α 抑制可挽救精神分裂症易感小鼠模型的工作记忆缺陷

Passecker, Johannes; Aloimonos, Chloe M; Dagunts, Aleksandra; Wagner, Florence F; Kupferschmidt, David A; Gogos, Joseph; Gordon, Joshua A

A Fast-Binding, Functionally Reversible, COX-2 Radiotracer for CNS PET Imaging

一种用于中枢神经系统PET成像的快速结合、功能可逆的COX-2放射性示踪剂

Placzek, Michael S; Wilton, Daniel K; Weïwer, Michel; Manter, Mariah A; Reid, Sarah E; Meyer, Christopher J; Campbell, Arthur J; Bajrami, Besnik; Bigot, Antoine; Bricault, Sarah; Fayet, Agathe; Frouin, Arnaud; Gergits, Frederick; Gupta, Mehak; Jiang, Wei; Melanson, Michelle; Romano, Chiara D; Riley, Misha M; Wang, Jessica M; Wey, Hsiao-Ying; Wagner, Florence F; Stevens, Beth; Hooker, Jacob M

HDAC2 targeting stabilizes the CoREST complex in renal tubular cells and protects against renal ischemia/reperfusion injury

靶向 HDAC2 可稳定肾小管细胞中的 CoREST 复合物,并保护肾脏免受缺血/再灌注损伤。

Aufhauser, David D Jr; Hernandez, Paul; Concors, Seth J; O'Brien, Ciaran; Wang, Zhonglin; Murken, Douglas R; Samanta, Arabinda; Beier, Ulf H; Krumeich, Lauren; Bhatti, Tricia R; Wang, Yanfeng; Ge, Guanghui; Wang, Liqing; Cheraghlou, Shayan; Wagner, Florence F; Holson, Edward B; Kalin, Jay H; Cole, Philip A; Hancock, Wayne W; Levine, Matthew H

MISCAST: MIssense variant to protein StruCture Analysis web SuiTe

错配:蛋白质结构分析网络套件的错义变体

Iqbal, Sumaiya; Hoksza, David; Pérez-Palma, Eduardo; May, Patrick; Jespersen, Jakob B; Ahmed, Shehab S; Rifat, Zaara T; Heyne, Henrike O; Rahman, M Sohel; Cottrell, Jeffrey R; Wagner, Florence F; Daly, Mark J; Campbell, Arthur J; Lal, Dennis

Comprehensive characterization of amino acid positions in protein structures reveals molecular effect of missense variants

对蛋白质结构中氨基酸位置的全面表征揭示了错义变异的分子效应

Iqbal, Sumaiya; Pérez-Palma, Eduardo; Jespersen, Jakob B; May, Patrick; Hoksza, David; Heyne, Henrike O; Ahmed, Shehab S; Rifat, Zaara T; Rahman, M Sohel; Lage, Kasper; Palotie, Aarno; Cottrell, Jeffrey R; Wagner, Florence F; Daly, Mark J; Campbell, Arthur J; Lal, Dennis

Translation of HDAC6 PET Imaging Using [(18)F]EKZ-001-cGMP Production and Measurement of HDAC6 Target Occupancy in Nonhuman Primates

利用[(18)F]EKZ-001-cGMP生产进行HDAC6 PET成像,并测量非人灵长类动物中HDAC6靶点占有率

Celen, Sofie; Rokka, Johanna; Gilbert, Tonya M; Koole, Michel; Vermeulen, Isabeau; Serdons, Kim; Schroeder, Frederick A; Wagner, Florence F; Bleeser, Tom; Hightower, Baileigh G; Hu, Jiyun; Rahal, Dania; Beyzavi, Hudson; Vanduffel, Wim; Van Laere, Koen; Kranz, Janice E; Hooker, Jacob M; Bormans, Guy; Cawthorne, Christopher J

Progress in Understanding and Treating SCN2A-Mediated Disorders

对SCN2A介导疾病的理解和治疗进展

Sanders, Stephan J; Campbell, Arthur J; Cottrell, Jeffrey R; Moller, Rikke S; Wagner, Florence F; Auldridge, Angie L; Bernier, Raphael A; Catterall, William A; Chung, Wendy K; Empfield, James R; George, Alfred L Jr; Hipp, Joerg F; Khwaja, Omar; Kiskinis, Evangelos; Lal, Dennis; Malhotra, Dheeraj; Millichap, John J; Otis, Thomas S; Petrou, Steven; Pitt, Geoffrey; Schust, Leah F; Taylor, Cora M; Tjernagel, Jennifer; Spiro, John E; Bender, Kevin J

Entropy as a Driver of Selectivity for Inhibitor Binding to Histone Deacetylase 6

熵作为抑制剂与组蛋白去乙酰化酶6结合选择性的驱动因素

Porter, Nicholas J; Wagner, Florence F; Christianson, David W

HDAC6 Brain Mapping with [(18)F]Bavarostat Enabled by a Ru-Mediated Deoxyfluorination

利用钌介导的脱氧氟化反应,通过[(18)F]Bavarostat进行HDAC6脑图谱绘制

Strebl, Martin G; Campbell, Arthur J; Zhao, Wen-Ning; Schroeder, Frederick A; Riley, Misha M; Chindavong, Peter S; Morin, Thomas M; Haggarty, Stephen J; Wagner, Florence F; Ritter, Tobias; Hooker, Jacob M

Isoform-selective inhibitor of histone deacetylase 3 (HDAC3) limits pancreatic islet infiltration and protects female nonobese diabetic mice from diabetes.

组蛋白去乙酰化酶 3 (HDAC3) 的亚型选择性抑制剂可限制胰岛浸润,并保护雌性非肥胖糖尿病小鼠免受糖尿病的侵害

Dirice Ercument, Ng Raymond W S, Martinez Rachael, Hu Jiang, Wagner Florence F, Holson Edward B, Wagner Bridget K, Kulkarni Rohit N