日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Dual inhibitors of Pseudomonas aeruginosa virulence factors LecA and LasB

铜绿假单胞菌毒力因子LecA和LasB的双重抑制剂

Metelkina, Olga; Konstantinović, Jelena; Klein, Andreas; Shafiei, Roya; Fares, Mario; Alhayek, Alaa; Yahiaoui, Samir; Elgaher, Walid A M; Haupenthal, Jörg; Titz, Alexander; Hirsch, Anna K H

Expression and characterization of pantothenate energy-coupling factor transporters as an anti-infective drug target

泛酸能量偶联因子转运蛋白的表达和表征及其作为抗感染药物靶点的研究

Shams, Atanaz; Bousis, Spyridon; Diamanti, Eleonora; Elgaher, Walid A M; Zeimetz, Lucie; Haupenthal, Jörg; Slotboom, Dirk J; Hirsch, Anna K H

NRF2 activators inhibit influenza A virus replication by interfering with nucleo-cytoplasmic export of viral RNPs in an NRF2-independent manner

NRF2激活剂通过干扰病毒核糖核蛋白(RNP)的核质输出,以不依赖于NRF2的方式抑制甲型流感病毒的复制。

Fakhar H Waqas,Mahmoud Shehata,Walid A M Elgaher,Antoine Lacour,Naziia Kurmasheva,Fabio Begnini,Anders E Kiib,Julia Dahlmann  ,Chutao Chen,Andreas Pavlou,Thomas B Poulsen,Sylvia Merkert  ,Ulrich Martin  ,Ruth Olmer  ,David Olagnier,Anna K H Hirsch  ,Stephan Pleschka  ,Frank Pessler

Hit-optimization using target-directed dynamic combinatorial chemistry: development of inhibitors of the anti-infective target 1-deoxy-d-xylulose-5-phosphate synthase

利用靶向动态组合化学进行先导化合物优化:开发抗感染靶标1-脱氧-D-木酮糖-5-磷酸合酶的抑制剂

Jumde, Ravindra P; Guardigni, Melissa; Gierse, Robin M; Alhayek, Alaa; Zhu, Di; Hamid, Zhoor; Johannsen, Sandra; Elgaher, Walid A M; Neusens, Philipp J; Nehls, Christian; Haupenthal, Jörg; Reiling, Norbert; Hirsch, Anna K H

Potential Dental Biofilm Inhibitors: Dynamic Combinatorial Chemistry Affords Sugar-Based Molecules that Target Bacterial Glucosyltransferase

潜在的牙菌斑抑制剂:动态组合化学方法制备靶向细菌葡萄糖基转移酶的糖基分子

Hartman, Alwin M; Jumde, Varsha R; Elgaher, Walid A M; Te Poele, Evelien M; Dijkhuizen, Lubbert; Hirsch, Anna K H

A hydrogel-based in vitro assay for the fast prediction of antibiotic accumulation in Gram-negative bacteria

基于水凝胶的体外检测方法快速预测革兰氏阴性细菌中抗生素的积累

Robert Richter, Mohamed A M Kamal, Mariel A García-Rivera, Jerome Kaspar, Maximilian Junk, Walid A M Elgaher, Sanjay Kumar Srikakulam, Alexander Gress, Anja Beckmann, Alexander Grißmer, Carola Meier, Michael Vielhaber, Olga Kalinina, Anna K H Hirsch, Rolf W Hartmann, Mark Brönstrup, Nicole Schneider

Discovery of Small-Molecule Stabilizers of 14-3-3 Protein-Protein Interactions via Dynamic Combinatorial Chemistry

利用动态组合化学发现14-3-3蛋白-蛋白相互作用的小分子稳定剂

Hartman, Alwin M; Elgaher, Walid A M; Hertrich, Nathalie; Andrei, Sebastian A; Ottmann, Christian; Hirsch, Anna K H