日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Accelerating drug target inhibitor discovery with a deep generative foundation model.

利用深度生成式基础模型加速药物靶点抑制剂的发现

Chenthamarakshan Vijil, Hoffman Samuel C, Owen C David, Lukacik Petra, Strain-Damerell Claire, Fearon Daren, Malla Tika R, Tumber Anthony, Schofield Christopher J, Duyvesteyn Helen M E, Dejnirattisai Wanwisa, Carrique Loic, Walter Thomas S, Screaton Gavin R, Matviiuk Tetiana, Mojsilovic Aleksandra, Crain Jason, Walsh Martin A, Stuart David I, Das Payel

Overall Survival Differences in Young Black Colorectal Cancer Patients: a Report from the National Cancer Database

年轻黑人结直肠癌患者的总体生存差异:来自国家癌症数据库的报告

Batten, Macelyn; Mukherjee, Rupak; Walter, Thomas S; Lancaster, William P

Bacteriophage PRD1 as a nanoscaffold for drug loading

噬菌体PRD1作为药物负载的纳米支架

Duyvesteyn, Helen M E; Santos-Pérez, Isaac; Peccati, Francesca; Martinez-Castillo, Ane; Walter, Thomas S; Reguera, David; Goñi, Felix M; Jiménez-Osés, Gonzalo; Oksanen, Hanna M; Stuart, David I; Abrescia, Nicola G A

Glutathione facilitates enterovirus assembly by binding at a druggable pocket

谷胱甘肽通过与一个可成药口袋结合,促进肠道病毒的组装。

Duyvesteyn, Helen M E; Ren, Jingshan; Walter, Thomas S; Fry, Elizabeth E; Stuart, David I

Assembly of complex viruses exemplified by a halophilic euryarchaeal virus

以嗜盐广古菌病毒为例,探讨复杂病毒的组装。

De Colibus, Luigi; Roine, Elina; Walter, Thomas S; Ilca, Serban L; Wang, Xiangxi; Wang, Nan; Roseman, Alan M; Bamford, Dennis; Huiskonen, Juha T; Stuart, David I

The structure of a prokaryotic viral envelope protein expands the landscape of membrane fusion proteins.

原核病毒包膜蛋白的结构拓展了膜融合蛋白的研究领域

El Omari Kamel, Li Sai, Kotecha Abhay, Walter Thomas S, Bignon Eduardo A, Harlos Karl, Somerharju Pentti, De Haas Felix, Clare Daniel K, Molin Mika, Hurtado Felipe, Li Mengqiu, Grimes Jonathan M, Bamford Dennis H, Tischler Nicole D, Huiskonen Juha T, Stuart David I, Roine Elina

A structural basis for antibody-mediated neutralization of Nipah virus reveals a site of vulnerability at the fusion glycoprotein apex

抗体介导的尼帕病毒中和作用的结构基础揭示了融合糖蛋白顶端的脆弱位点

Avanzato, Victoria A; Oguntuyo, Kasopefoluwa Y; Escalera-Zamudio, Marina; Gutierrez, Bernardo; Golden, Michael; Kosakovsky Pond, Sergei L; Pryce, Rhys; Walter, Thomas S; Seow, Jeffrey; Doores, Katie J; Pybus, Oliver G; Munster, Vincent J; Lee, Benhur; Bowden, Thomas A

High-speed fixed-target serial virus crystallography

高速固定靶串行病毒晶体学

Roedig, Philip; Ginn, Helen M; Pakendorf, Tim; Sutton, Geoff; Harlos, Karl; Walter, Thomas S; Meyer, Jan; Fischer, Pontus; Duman, Ramona; Vartiainen, Ismo; Reime, Bernd; Warmer, Martin; Brewster, Aaron S; Young, Iris D; Michels-Clark, Tara; Sauter, Nicholas K; Kotecha, Abhay; Kelly, James; Rowlands, David J; Sikorsky, Marcin; Nelson, Silke; Damiani, Daniel S; Alonso-Mori, Roberto; Ren, Jingshan; Fry, Elizabeth E; David, Christian; Stuart, David I; Wagner, Armin; Meents, Alke

Near-atomic structure of Japanese encephalitis virus reveals critical determinants of virulence and stability

日本脑炎病毒的近原子结构揭示了其毒力和稳定性的关键决定因素

Wang, Xiangxi; Li, Shi-Hua; Zhu, Ling; Nian, Qing-Gong; Yuan, Shuai; Gao, Qiang; Hu, Zhongyu; Ye, Qing; Li, Xiao-Feng; Xie, Dong-Yang; Shaw, Neil; Wang, Junzhi; Walter, Thomas S; Huiskonen, Juha T; Fry, Elizabeth E; Qin, Cheng-Feng; Stuart, David I; Rao, Zihe

The crystal structure of human dopamine β-hydroxylase at 2.9 Å resolution

人类多巴胺β-羟化酶的晶体结构,分辨率为2.9 Å

Vendelboe, Trine V; Harris, Pernille; Zhao, Yuguang; Walter, Thomas S; Harlos, Karl; El Omari, Kamel; Christensen, Hans E M