日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structural insights into the development of inhibitors for inositol phosphate kinases

肌醇磷酸激酶抑制剂研发的结构解析

Wang, Huanchen

KIDINS220 and InsP8 safeguard the stepwise regulation of phosphate exporter XPR1.

KIDINS220 和 InsP8 保障磷酸盐输出因子 XPR1 的逐步调控

Wang Xiaojie, Bai Zhongjian, Wallis Ciara, Wang Huanchen, Han Yaoyao, Jin Ruitao, Lei Mingguang, Yang Tian, Gu Chunfang, Jessen Henning, Shears Stephen, Sun Yadong, Corry Ben, Zhang Yixiao

Structural Rationalization of IPMK Inhibitor Potency

IPMK抑制剂效力的结构合理化

Wang, Huanchen; Shears, Stephen B; Blind, Raymond D

Correction: Identification of acrylamide-based covalent inhibitors of SARS-CoV-2 (SCoV-2) Nsp15 using high-throughput screening and machine learning

更正:利用高通量筛选和机器学习鉴定基于丙烯酰胺的SARS-CoV-2 (SCoV-2) Nsp15共价抑制剂

Bajaj, Teena; Mosavati, Babak; Zhang, Lydia H; Parsa, Mohammad S; Wang, Huanchen; Kerek, Evan M; Liang, Xueying; Tabatabaei Dakhili, Seyed Amir; Wehri, Eddie; Guo, Silin; Desai, Rushil N; Orr, Lauren M; Mofrad, Mohammad R K; Schaletzky, Julia; Ussher, John R; Deng, Xufang; Stanley, Robin; Hubbard, Basil P; Nomura, Daniel K; Murthy, Niren

Identification of acrylamide-based covalent inhibitors of SARS-CoV-2 (SCoV-2) Nsp15 using high-throughput screening and machine learning.

利用高通量筛选和机器学习鉴定 SARS-CoV-2 (SCoV-2) Nsp15 的丙烯酰胺基共价抑制剂

Bajaj Teena, Mosavati Babak, Zhang Lydia H, Parsa Mohammad S, Wang Huanchen, Kerek Evan M, Liang Xueying, Tabatabaei Dakhili Seyed Amir, Wehri Eddie, Guo Silin, Desai Rushil N, Orr Lauren M, Mofrad Mohammad R K, Schaletzky Julia, Ussher John R, Deng Xufang, Stanley Robin, Hubbard Basil P, Nomura Daniel K, Murthy Niren

Biochemical and biophysical characterization of inositol-tetrakisphosphate 1-kinase inhibitors.

肌醇四磷酸1-激酶抑制剂的生化和生物物理特性

Ng Martin Y, Wang Huanchen, Zhang Haibo, Prucker Isabel, Perera Lalith, Goncharova Ekaterina, Wamiru Antony, Jessen Henning J, Stanley Robin E, Shears Stephen B, Luo Ji, O'Keefe Barry R, Wilson Brice A P

New structural insights reveal an expanded reaction cycle for inositol pyrophosphate hydrolysis by human DIPP1

新的结构分析揭示了人 DIPP1 介导的肌醇焦磷酸水解的扩展反应循环

Zong, Guangning; Jork, Nikolaus; Hostachy, Sarah; Fiedler, Dorothea; Jessen, Henning J; Shears, Stephen B; Wang, Huanchen

Rapid stimulation of cellular Pi uptake by the inositol pyrophosphate InsP(8) induced by its photothermal release from lipid nanocarriers using a near infra-red light-emitting diode

利用近红外发光二极管,通过光热法从脂质纳米载体中释放肌醇焦磷酸酯 InsP(8),可快速刺激细胞对磷酸盐的摄取。

Wang, Zhenzhen; Jork, Nikolaus; Bittner, Tamara; Wang, Huanchen; Jessen, Henning J; Shears, Stephen B

MicroRNA-21 mediates high phosphate-induced endothelial cell apoptosis

MicroRNA-21介导高磷酸盐诱导的内皮细胞凋亡

Li, Zhaoyu; Wiernek, Szymon; Patterson, Cam; Wang, Huanchen; Qi, Guoxian; Dai, Xuming

Use of Protein Kinase-Focused Compound Libraries for the Discovery of New Inositol Phosphate Kinase Inhibitors

利用蛋白激酶靶向化合物库发现新型肌醇磷酸激酶抑制剂

Puhl-Rubio, Ana C; Stashko, Michael A; Wang, Huanchen; Hardy, P Brian; Tyagi, Vikas; Li, Bing; Wang, Xiaodong; Kireev, Dmitri; Jessen, Henning J; Frye, Stephen V; Shears, Stephen B; Pearce, Kenneth H