Targeting the Spliceosomal Protein USP39 Through Allosteric Ligands and PROTAC-Induced Degradation
通过变构配体和PROTAC诱导降解靶向剪接体蛋白USP39
期刊:Angewandte Chemie-International Edition
影响因子:16.9
doi:10.1002/anie.202516809
Schäfer, Daniel; Prieto-Garcia, Cristian; Wang, Jianhui; Heinz, Marcel; Matkovic, Vigor; Kielkowski, Pavel; Hasselbeck, Sebastian; Shah, Varun Jayeshkumar; Knapp, Stefan; Hummer, Gerhard; Dikic, Ivan; Cheng, Xinlai