日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The p53 R181C mutation accumulates through impaired deacetylation by Sirt1 and facilitates tumor development.

p53 R181C 突变通过 Sirt1 的去乙酰化作用受损而积累,并促进肿瘤发展。

Wang Erli, Cao Liangzi, Guo Wendong, Dong Xiang, Zhang Wanying, Zhang Xiaowen, Wang Zhuo, Chen Xia, Li Aicun, Zou Yu, Li Shikun, Chen Kedian, Su Han, Cao Sunrun, Du Ning, Wang Pingyuan, Hwang Paul M, Liu Xiangsheng, Song Xiaoyu, Xu Hongde, Liu Jingwei, Cao Liu

Virtual Screening of Marine Natural Products Targeting the F Protein for Anti-RSV Drug Discovery

利用虚拟筛选方法筛选靶向F蛋白的海洋天然产物用于抗RSV药物发现

Liu, Wenqing; Gu, Xuran; Du, Ruikun; Liu, Zhiqing; Wang, Pingyuan; Wang, Chang-Yun

Sensory neuron-expressed FGF13 controls nociceptive signaling in diabetic neuropathy models

感觉神经元表达的FGF13控制糖尿病神经病变模型中的伤害性信号传导

Singh, Aditya K; Bernabucci, Matteo; Dvorak, Nolan M; Haghighijoo, Zahra; Di Re, Jessica; Goode, Nana A; Kadakia, Feni K; Maile, Laura A; Folorunso, Olumarotimi O; Wadsworth, Paul A; Tapia, Cynthia M; Wang, Pingyuan; Wang, Jigong; Chen, Haiying; Xue, Yu; Singh, Jully; Hankerd, Kali; Gamez, Isaac J; Kager, Makenna; Truong, Vincent; Walsh, Patrick; Shiers, Stephanie I; Kuttanna, Nishka; Liao, Hanyue; Marchi, Margherita; Salvi, Erika; D'Amato, Ilaria; D'Amico, Daniela; Arman, Parsa; Faber, Catharina G; Malik, Rayaz A; de Tommaso, Marina; Ziegler, Dan; Rajarathnam, Krishna; Green, Thomas A; Grace, Peter M; Sapio, Matthew R; Iadarola, Michael J; Cuny, Gregory D; Chow, Diana S; Lauria Pinter, Giuseppe; Davidson, Steve; Green, Dustin P; La, Jun-Ho; Chung, Jin Mo; Zhou, Jia; Price, Theodore J; Salisbury, Elizabeth; Yuan, Subo; Laezza, Fernanda

MR2938 relieves DSS-induced colitis in mice through inhibiting NF-κB signaling and improving epithelial barrier

MR2938 通过抑制 NF-κB 信号通路和改善上皮屏障功能,缓解 DSS 诱导的小鼠结肠炎。

Lv, Ling; Maimaitiming, Mireguli; Xia, Shuli; Yang, Jichen; Zhang, Tiantian; Wang, Yuming; Li, Xin; Pinchuk, Iryna; Wang, Pingyuan; Wang, Chang-Yun; Liu, Zhiqing

Quinazolinone Derivative MR2938 Protects DSS-Induced Barrier Dysfunction in Mice Through Regulating Gut Microbiota

喹唑啉酮衍生物MR2938通过调节肠道菌群保护小鼠免受DSS诱导的屏障功能障碍。

Lv, Ling; Maimaitiming, Mireguli; Yang, Jichen; Xia, Shuli; Li, Xin; Wang, Pingyuan; Liu, Zhiqing; Wang, Chang-Yun

FGF14 Peptide Derivative Differentially Regulates Nav1.2 and Na(v)1.6 Function.

FGF14 肽衍生物差异性地调节 Nav1.2 和 Na(v)1.6 的功能

Arman Parsa, Haghighijoo Zahra, Lupascu Carmen A, Singh Aditya K, Goode Nana A, Baumgartner Timothy J, Singh Jully, Xue Yu, Wang Pingyuan, Chen Haiying, Antunes Dinler A, Lijffijt Marijn, Zhou Jia, Migliore Michele, Laezza Fernanda

Orphan GPR52 as an emerging neurotherapeutic target

孤儿GPR52作为一种新兴的神经治疗靶点

Ali, Saghir; Wang, Pingyuan; Murphy, Ryan E; Allen, John A; Zhou, Jia

Discovery of 3-((4-Benzylpyridin-2-yl)amino)benzamides as Potent GPR52 G Protein-Biased Agonists

发现 3-((4-苄基吡啶-2-基)氨基)苯甲酰胺类化合物作为强效 GPR52 G 蛋白偏向性激动剂

Murphy, Ryan E; Wang, Pingyuan; Ali, Saghir; Smith, Hudson R; Felsing, Daniel E; Chen, Haiying; Zhou, Jia; Allen, John A

Functionally selective dopamine D1 receptor endocytosis and signaling by catechol and non-catechol agonists

儿茶酚和非儿茶酚激动剂对多巴胺D1受体的功能选择性内吞作用和信号传导

Nilson, Ashley N; Felsing, Daniel E; Wang, Pingyuan; Jain, Manish; Zhou, Jia; Allen, John

Thioparib inhibits homologous recombination repair, activates the type I IFN response, and overcomes olaparib resistance

硫代帕尼抑制同源重组修复,激活 I 型干扰素反应,并克服奥拉帕尼耐药性

Li-Min Wang #, Pingyuan Wang #, Xiao-Min Chen #, Hui Yang, Shan-Shan Song, Zilan Song, Li Jia, Hua-Dong Chen, Xu-Bin Bao, Ne Guo, Xia-Juan Huan, Yong Xi, Yan-Yan Shen, Xin-Ying Yang, Yi Su, Yi-Ming Sun, Ying-Lei Gao, Yi Chen, Jian Ding, Jing-Yu Lang, Ze-Hong Miao, Ao Zhang, Jin-Xue He