日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

An accessible 3D HepG2/C3A liver spheroid model supporting the complete intrahepatocytic lifecycle of Plasmodium falciparum.

一种易于操作的 3D HepG2/C3A 肝球体模型,支持恶性疟原虫完整的肝细胞内生命周期。

Caygill Claire H, Alqurashi Salwa Omar, Adolfi Adriana, Carson Jessica, Sturm Angelika, Evans Daniel S, Jinks Jess B, Dechering Koen J, Reimer Lisa, Pennington Shaun H, Sharma Parveen, Ward Stephen A, Biagini Giancarlo A

Design, synthesis and modelling of photoreactive chemical probes for investigating target engagement of plasmepsin IX and X in Plasmodium falciparum

设计、合成和建模光反应化学探针,用于研究恶性疟原虫中疟原虫蛋白酶IX和X的靶标结合

Lisauskaitė, Monika; Nixon, Gemma L; Woodley, Christopher M; Berry, Neil G; Coninckx, Andy; Qie, L Charlie; Leung, Suet C; Taramelli, Donatella; Basilico, Nicoletta; Parapini, Silvia; Ward, Stephen A; Vadas, Oscar; Soldati-Favre, Dominique; Hong, W David; O'Neill, Paul M

Targeting the Ubiquinol-Reduction (Q(i)) Site of the Mitochondrial Cytochrome bc(1) Complex for the Development of Next Generation Quinolone Antimalarials

靶向线粒体细胞色素bc(1)复合物的泛醌还原(Q(i))位点以开发下一代喹诺酮类抗疟药

Amporndanai, Kangsa; Pinthong, Nattapon; O'Neill, Paul M; Hong, W David; Amewu, Richard K; Pidathala, Chandrakala; Berry, Neil G; Leung, Suet C; Ward, Stephen A; Biagini, Giancarlo A; Hasnain, S Samar; Antonyuk, Svetlana V

Co-transmission of Related Malaria Parasite Lineages Shapes Within-Host Parasite Diversity.

相关疟原虫谱系的共同传播塑造了宿主内寄生虫的多样性

Nkhoma Standwell C, Trevino Simon G, Gorena Karla M, Nair Shalini, Khoswe Stanley, Jett Catherine, Garcia Roy, Daniel Benjamin, Dia Aliou, Terlouw Dianne J, Ward Stephen A, Anderson Timothy J C, Cheeseman Ian H

In vivo efficacy of the boron-pleuromutilin AN11251 against Wolbachia of the rodent filarial nematode Litomosoides sigmodontis

硼-截短侧耳素AN11251对啮齿类丝状线虫Litomosoides sigmodontis沃尔巴克氏体的体内疗效

Ehrens, Alexandra; Lunde, Christopher S; Jacobs, Robert T; Struever, Dominique; Koschel, Marianne; Frohberger, Stefan J; Lenz, Franziska; Fendler, Martina; Turner, Joseph D; Ward, Stephen A; Taylor, Mark J; Freund, Yvonne R; Stefanakis, Rianna; Easom, Eric; Li, Xianfeng; Plattner, Jacob J; Hoerauf, Achim; Hübner, Marc P

M1 macrophage features in severe Plasmodium falciparum malaria patients with pulmonary oedema

M1型巨噬细胞在伴有肺水肿的重症恶性疟疾患者中具有特征性表现。

Klinkhamhom, Aekkarin; Glaharn, Supattra; Srisook, Charit; Ampawong, Sumate; Krudsood, Srivicha; Ward, Stephen A; Viriyavejakul, Parnpen

Human Direct Skin Feeding Versus Membrane Feeding to Assess the Mosquitocidal Efficacy of High-Dose Ivermectin (IVERMAL Trial)

人体直接皮肤喂食与膜喂食评估高剂量伊维菌素杀蚊效果(IVERMAL试验)

Smit, Menno R; Ochomo, Eric O; Aljayyoussi, Ghaith; Kwambai, Titus K; Abong'o, Bernard O; Bousema, Teun; Waterhouse, David; Bayoh, Nabie M; Gimnig, John E; Samuels, Aaron M; Desai, Meghna R; Phillips-Howard, Penelope A; Kariuki, Simon K; Wang, Duolao; Ward, Stephen A; Ter Kuile, Feiko O

Pharmacokinetics-Pharmacodynamics of High-Dose Ivermectin with Dihydroartemisinin-Piperaquine on Mosquitocidal Activity and QT-Prolongation (IVERMAL)

高剂量伊维菌素联合双氢青蒿素-哌喹对蚊虫杀灭活性和QT间期延长的药代动力学-药效学研究(IVERMAL)

Smit, Menno R; Ochomo, Eric O; Waterhouse, David; Kwambai, Titus K; Abong'o, Bernard O; Bousema, Teun; Bayoh, Nabie M; Gimnig, John E; Samuels, Aaron M; Desai, Meghna R; Phillips-Howard, Penelope A; Kariuki, Simon K; Wang, Duolao; Ter Kuile, Feiko O; Ward, Stephen A; Aljayyoussi, Ghaith

Intracellular PD Modelling (PD(i)) for the Prediction of Clinical Activity of Increased Rifampicin Dosing

细胞内药效学模型(PD(i))用于预测利福平剂量增加的临床活性

Aljayyoussi, Ghaith; Donnellan, Samantha; Ward, Stephen A; Biagini, Giancarlo A

Intracellular Pharmacodynamic Modeling Is Predictive of the Clinical Activity of Fluoroquinolones against Tuberculosis

细胞内药效学模型可预测氟喹诺酮类药物抗结核病的临床活性

Donnellan, Samantha; Aljayyoussi, Ghaith; Moyo, Emmanuel; Ardrey, Alison; Martinez-Rodriguez, Carmen; Ward, Stephen A; Biagini, Giancarlo A