Examination of Noncanonical Kinase Hinge Binders Leads to Thiadiazoles as Potent IRAK4 Inhibitors
对非经典激酶铰链结合剂的研究发现噻二唑类化合物是强效的IRAK4抑制剂
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.5c00602
Ammann, Stephen E; Brizgys, Gediminas; Ferrao, Ryan D; Wright, Nathan E; Mukherjee, Prasenjit Kumar; Bacon, Elizabeth M; Chin, Elbert; Chou, Chienhung; Cottell, Jeromy J; Hammond, Angela; Ndukwe, Marilyn S; Park, Grace Y; Shatskikh, Marina E; Suekawa-Pirrone, Kimberly; Warr, Matthew R; Yang, Zheng-Yu; Zipfel, Sheila M; Taylor, James G