日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A long-lasting PI3Kδ inhibitor zandelisib forms a water-shielded hydrogen bond with p110δ and demonstrates sustained inhibitory effects.

长效 PI3Kδ 抑制剂 zandelisib 与 p110δ 形成水屏蔽氢键,并表现出持续的抑制作用

Kunieda Kana, Nagiri Chisae, Watanabe Miwa, Yoshida Tadashi, Zou Jian, Kaneda Ayumi, Takahashi Yuichi, Aburai Kenichi, Saito Jun-Ichi, Umehara Hiroshi, Otsu Yoshiaki, Ishii Toshihiko

Screening for DAX1/EWS-FLI1 functional inhibitors identified dihydroorotate dehydrogenase as a therapeutic target for Ewing's sarcoma

对 DAX1/EWS-FLI1 功能抑制剂的筛选发现,二氢乳清酸脱氢酶是尤文氏肉瘤的治疗靶点。

Watanabe, Miwa; Kosaka, Hiromichi; Sugawara, Masamori; Maemoto, Michihiro; Ono, Yoko; Uemori, Takeshi; Shizu, Ryota; Yoshinari, Kouichi

Periostin-An inducer of pro-fibrotic phenotype in monocytes and monocyte-derived macrophages in systemic sclerosis

骨膜素——系统性硬化症中单核细胞和单核细胞衍生的巨噬细胞中促纤维化表型的诱导剂

Mao Suzuki, Yasushi Ototake, Asami Akita, Miho Asami, Noriko Ikeda, Tomoya Watanabe, Miwa Kanaoka, Yukie Yamaguchi

Navigational choice between reversal and curve during acidic pH avoidance behavior in Caenorhabditis elegans

秀丽隐杆线虫在酸性pH回避行为中,导航选择是反转还是弯曲

Wakabayashi, Tokumitsu; Sakata, Kazumi; Togashi, Takuya; Itoi, Hiroaki; Shinohe, Sayaka; Watanabe, Miwa; Shingai, Ryuzo