日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Tetrahydropyrazolopyridinones as a Novel Class of Potent and Highly Selective LIMK Inhibitors

四氢吡唑并吡啶酮类化合物作为一类新型高效高选择性LIMK抑制剂

Baldwin, Alex G; Foley, David W; Jones, D Heulyn; Lee, Hyunah; Collins, Ross; Wahab, Ben; Pedder, Josephine H; Waters, Loren; Paine, Marie; Schino, Lauramariú; Feng, Gui Jie; Kariuki, Benson M; Elkins, Jonathan M; Atack, John R; Ward, Simon E

Discovery of MDI-114215: A Potent and Selective LIMK Inhibitor To Treat Fragile X Syndrome.

MDI-114215 的发现:一种强效且选择性的 LIMK 抑制剂,可用于治疗脆性 X 综合征

Baldwin Alex G, Foley David W, Collins Ross, Lee Hyunah, Jones D Heulyn, Wahab Ben, Waters Loren, Pedder Josephine, Paine Marie, Feng Gui Jie, Privitera Lucia, Ashall-Kelly Alexander, Thomas Carys, Gillespie Jason A, Schino Lauramariú, Belelli Delia, Rocha Cecilia, Maussion Gilles, Krahn Andrea I, Durcan Thomas M, Elkins Jonathan M, Lambert Jeremy J, Atack John R, Ward Simon E