日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification of KLHL12 Ligands Using Fragment-Based Methods

利用基于片段的方法鉴定KLHL12配体

Waterson, Alex G; Vadukoot, Anish; Jana, Somnath; Cui, Jianwen; Luong, Kelvin; Rietz, Tyson A; Madrigal-Carrillo, Ezequiel Alejandro; Lehmann, Brian D; Sensintaffar, John L; Zhao, Bin; Amporndanai, Kangsa; Petros, Zoe A; Scaggs, William Rush; Chacon Simon, Selena; Vekariya, Rakesh H; Kim, Kwangho; Thangaraj, Manikandan; Christov, Plamen P; South, Taylor M; Sai, Jiqing; Thiruvaipati, Anusha; Schmidt, Charles R; Eells, Rebecca; Moore, William J; Olejniczak, Edward T; Phan, Jason; Fesik, Stephen W

High-throughput screening identifies a trafficking corrector for long QT syndrome-associated KCNQ1 variants

高通量筛选鉴定出一种与长QT综合征相关的KCNQ1变异体的转运校正因子

Moster, Katherine R Clowes; Vanoye, Carlos G; Chang-Gonzalez, Ana C; Romaine, Ian M; Stefanski, Katherine M; Wilkinson, Mason C; Bauer, Joshua A; Hasaka, Thomas P; Days, Emily L; Desai, Reshma R; Butcher, Kathryn R; Sulikowski, Gary A; Waterson, Alex G; Meiler, Jens; Ledwitch, Kaitlyn V; George, Alfred L Jr; Sanders, Charles R

Drugit: crowd-sourcing molecular design of non-peptidic VHL binders

Drugit:众包非肽类VHL结合剂的分子设计

Scott, Thomas; Smethurst, Christian Alan Paul; Westermaier, Yvonne; Mayer, Moriz; Greb, Peter; Kousek, Roland; Biberger, Tobias; Bader, Gerd; Jandova, Zuzana; Schmalhorst, Philipp S; Fuchs, Julian E; Magarkar, Aniket; Hoenke, Christoph; Gerstberger, Thomas; Combs, Steven A; Pape, Richard; Phul, Saksham; Kothiwale, Sandeepkumar; Bergner, Andreas; Waterson, Alex G; Weinstabl, Harald; McConnell, Darryl B; Meiler, Jens; Böttcher, Jark; Moretti, Rocco

Discovery of Small Molecules that Bind to Son of Sevenless 2 (SOS2)

发现与SOS2结合的小分子

Krzysztof M Zak, Alex G Waterson, Leonhard Geist, Nina Braun, Katja Hauer, Klaus Rumpel, Juergen Ramharter, Heinz Stadtmueller, Bernhard Wolkerstorfer, David Schoenbauer, Jianwen Cui, Jason Phan, Jason R Abbott, Dhruba Sarkar, Timothy R Hodges, Allison Arnold, John L Sensintaffar, Stephen W Fesik, D

Switching It up with New KRAS Inhibitors

用新型KRAS抑制剂改变策略

Waterson, Alex G

Discovery of BI-2493, a Pan-KRAS Inhibitor Showing In Vivo Efficacy.

发现 BI-2493,一种泛 KRAS 抑制剂,显示出体内疗效

Bröker Joachim, Waterson Alex G, Hodges Timothy R, Abbott Jason R, Arnold Allison, Böttcher Jark, Braun Nina, Cui Jianwen, Fuchs Julian E, Gerstberger Thomas, Gogg Sebastian, Hanner Sabine, Herdeis Lorenz, Howell Lucas W, Mantoulidis Andreas, Mayer Moriz, Phan Jason, Rocchetti Francesca, Sankar Kyra, Sarkar Dhruba, Schaaf Otmar, Sensintaffar John L, Sun Qi, Wunberg Tobias, Fesik Stephen W

Nuclear Magnetic Resonance-based fragment screen of the E3 ligase Fem-1 homolog B

基于核磁共振的E3连接酶Fem-1同源物B片段筛选

Katinas, Jade M; Amporndanai, Kangsa; Taylor, Ashley J; Rose, Kristie L; Gareiss, Peter C; Crespo, Roberto A; Phan, Jason; Waterson, Alex G; Fesik, Stephen W

The adaptive dynamic programming signal control system for person in a connected vehicle environment

联网车辆环境中人员自适应动态规划信号控制系统

Wu, Zongyuan; Li, Shiming; Li, Gen; Waterson, Ben; Zhu, Luyao; Wang, Decai

The effect of the COVID-19 pandemic on the baby-friendly community initiative and maternal infant and young child nutrition in Kenya

新冠疫情对肯尼亚母婴友好社区倡议及孕产妇、婴幼儿营养的影响

Mutoro, Antonina Namaemba; Wanjohi, Milka; Wilunda, Calistus; Koech, Maureen J; Ogunsola, Ajibola; Tako, Antuela; Jun, Thomas Gyuchan; Waterson, Patrick; Griffiths, Paula L; Kimani-Murage, Elizabeth Wambui

Alternative alignment clinical study: study protocol for a prospective, randomised, controlled study of the outcomes and cost effectiveness of triathlon CR knee replacement system: traditional philosophy versus alternative alignment philosophy

替代对线临床研究:一项前瞻性、随机、对照研究方案,旨在评估 Triathlon CR 膝关节置换系统的疗效和成本效益:传统理念与替代对线理念的比较。

Sheen, Jonathon; Abdul, Wahid; Corroon, Ciara; Waterson, Ben; Toms, Andy