日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification of KLHL12 Ligands Using Fragment-Based Methods

利用基于片段的方法鉴定KLHL12配体

Waterson, Alex G; Vadukoot, Anish; Jana, Somnath; Cui, Jianwen; Luong, Kelvin; Rietz, Tyson A; Madrigal-Carrillo, Ezequiel Alejandro; Lehmann, Brian D; Sensintaffar, John L; Zhao, Bin; Amporndanai, Kangsa; Petros, Zoe A; Scaggs, William Rush; Chacon Simon, Selena; Vekariya, Rakesh H; Kim, Kwangho; Thangaraj, Manikandan; Christov, Plamen P; South, Taylor M; Sai, Jiqing; Thiruvaipati, Anusha; Schmidt, Charles R; Eells, Rebecca; Moore, William J; Olejniczak, Edward T; Phan, Jason; Fesik, Stephen W

High-throughput screening identifies a trafficking corrector for long QT syndrome-associated KCNQ1 variants

高通量筛选鉴定出一种与长QT综合征相关的KCNQ1变异体的转运校正因子

Moster, Katherine R Clowes; Vanoye, Carlos G; Chang-Gonzalez, Ana C; Romaine, Ian M; Stefanski, Katherine M; Wilkinson, Mason C; Bauer, Joshua A; Hasaka, Thomas P; Days, Emily L; Desai, Reshma R; Butcher, Kathryn R; Sulikowski, Gary A; Waterson, Alex G; Meiler, Jens; Ledwitch, Kaitlyn V; George, Alfred L Jr; Sanders, Charles R

Drugit: crowd-sourcing molecular design of non-peptidic VHL binders

Drugit:众包非肽类VHL结合剂的分子设计

Scott, Thomas; Smethurst, Christian Alan Paul; Westermaier, Yvonne; Mayer, Moriz; Greb, Peter; Kousek, Roland; Biberger, Tobias; Bader, Gerd; Jandova, Zuzana; Schmalhorst, Philipp S; Fuchs, Julian E; Magarkar, Aniket; Hoenke, Christoph; Gerstberger, Thomas; Combs, Steven A; Pape, Richard; Phul, Saksham; Kothiwale, Sandeepkumar; Bergner, Andreas; Waterson, Alex G; Weinstabl, Harald; McConnell, Darryl B; Meiler, Jens; Böttcher, Jark; Moretti, Rocco

Switching It up with New KRAS Inhibitors

用新型KRAS抑制剂改变策略

Waterson, Alex G

Discovery of BI-2493, a Pan-KRAS Inhibitor Showing In Vivo Efficacy.

发现 BI-2493,一种泛 KRAS 抑制剂,显示出体内疗效

Bröker Joachim, Waterson Alex G, Hodges Timothy R, Abbott Jason R, Arnold Allison, Böttcher Jark, Braun Nina, Cui Jianwen, Fuchs Julian E, Gerstberger Thomas, Gogg Sebastian, Hanner Sabine, Herdeis Lorenz, Howell Lucas W, Mantoulidis Andreas, Mayer Moriz, Phan Jason, Rocchetti Francesca, Sankar Kyra, Sarkar Dhruba, Schaaf Otmar, Sensintaffar John L, Sun Qi, Wunberg Tobias, Fesik Stephen W

Nuclear Magnetic Resonance-based fragment screen of the E3 ligase Fem-1 homolog B

基于核磁共振的E3连接酶Fem-1同源物B片段筛选

Katinas, Jade M; Amporndanai, Kangsa; Taylor, Ashley J; Rose, Kristie L; Gareiss, Peter C; Crespo, Roberto A; Phan, Jason; Waterson, Alex G; Fesik, Stephen W

NMR-Based Fragment Screen of the von Hippel-Lindau Elongin C&B Complex

基于核磁共振的von Hippel-Lindau Elongin C&B复合物片段筛选

Amporndanai, Kangsa; Katinas, Jade M; Chopra, Ashima; Kayode, Olumide; Vadukoot, Anish K; Waterson, Alex G; Fesik, Stephen W

Identification of ligands for E3 ligases with restricted expression using fragment-based methods

利用基于片段的方法鉴定表达受限的E3连接酶的配体

Waterson, Alex G; Lehmann, Brian D; Lu, Zhenwei; Sensintaffar, John L; Olejniczak, Edward T; Zhao, Bin; Rietz, Tyson; Payne, William G; Phan, Jason; Fesik, Stephen W

High Throughput Screening Identifies a Small Molecule Trafficking Corrector for Long-QT Syndrome Associated KCNQ1 Variants

高通量筛选鉴定出一种针对长QT综合征相关KCNQ1变异的小分子转运校正剂

Moster, Katherine R Clowes; Vanoye, Carlos G; Chang-Gonzalez, Ana C; Romaine, Ian M; Stefanski, Katherine M; Wilkinson, Mason C; Bauer, Joshua A; Hasaka, Thomas P; Days, Emily L; Desai, Reshma R; Butcher, Kathryn R; Sulikowski, Gary A; Waterson, Alex G; Meiler, Jens; Ledwitch, Kaitlyn V; George, Alfred L Jr; Sanders, Charles R

Simultaneous Exposure to Intracellular and Extracellular Photosensitizers for the Treatment of Staphylococcus aureus Infections

同时使用细胞内和细胞外光敏剂治疗金黄色葡萄球菌感染

Drury, Sydney L; Miller, Anderson R; Laut, Clare L; Walter, Alec B; Bennett, Monique R; Su, Meng; Bai, Mingfeng; Jing, Bingwen; Joseph, Scott B; Metzger, Edward J; Bane, Charles E; Black, Chad C; Macdonald, Mary T; Dutter, Brendan F; Romaine, Ian M; Waterson, Alex G; Sulikowski, Gary A; Jansen, E Duco; Crowe, James E Jr; Sciotti, Richard J; Skaar, Eric P