日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Optimization of diastereomeric dihydropyridines as antimalarials

优化非对映异构二氢吡啶类化合物作为抗疟药

Van Horn, Kurt S; Zhao, Yingzhao; Parvatkar, Prakash T; Maier, Julie; Mutka, Tina; Lacrue, Alexis; Brockmeier, Fabian; Ebert, Daniel; Wu, Wesley; Casandra, Debora R; Namelikonda, Niranjan; Yacoub, Jeanine; Sigal, Martina; Knapp, Spencer; Floyd, David; Waterson, David; Burrows, Jeremy N; Duffy, James; DeRisi, Joseph L; Kyle, Dennis E; Guy, R Kiplin; Manetsch, Roman

Exploring a Tetrahydroquinoline Antimalarial Hit from the Medicines for Malaria Pathogen Box and Identification of its Mode of Resistance as PfeEF2

从疟疾病原体药物库中筛选出一种四氢喹啉类抗疟药,并鉴定其耐药机制为 PfeEF2。

Laleu, Benoît; Rubiano, Kelly; Yeo, Tomas; Hallyburton, Irene; Anderson, Mark; Crespo-Fernandez, Benigno; Gamo, Francisco-Javier; Antonova-Koch, Yevgeniya; Orjuela-Sanchez, Pamela; Wittlin, Sergio; Jana, Gouranga P; Maity, Bikash C; Chenu, Elodie; Duffy, James; Sjö, Peter; Waterson, David; Winzeler, Elizabeth; Guantai, Eric; Fidock, David A; Hansson, Thomas G

Lead Optimization of a Pyrrole-Based Dihydroorotate Dehydrogenase Inhibitor Series for the Treatment of Malaria.

吡咯基二氢乳清酸脱氢酶抑制剂系列先导化合物的优化及其在疟疾治疗中的应用

Kokkonda Sreekanth, Deng Xiaoyi, White Karen L, El Mazouni Farah, White John, Shackleford David M, Katneni Kasiram, Chiu Francis C K, Barker Helena, McLaren Jenna, Crighton Elly, Chen Gong, Angulo-Barturen Inigo, Jimenez-Diaz Maria Belen, Ferrer Santiago, Huertas-Valentin Leticia, Martinez-Martinez Maria Santos, Lafuente-Monasterio Maria Jose, Chittimalla Rajesh, Shahi Shatrughan P, Wittlin Sergio, Waterson David, Burrows Jeremy N, Matthews Dave, Tomchick Diana, Rathod Pradipsinh K, Palmer Michael J, Charman Susan A, Phillips Margaret A

Substituted Aminoacetamides as Novel Leads for Malaria Treatment

取代氨基乙酰胺作为疟疾治疗的新型先导化合物

Norcross, Neil R; Wilson, Caroline; Baragaña, Beatriz; Hallyburton, Irene; Osuna-Cabello, Maria; Norval, Suzanne; Riley, Jennifer; Fletcher, Daniel; Sinden, Robert; Delves, Michael; Ruecker, Andrea; Duffy, Sandra; Meister, Stephan; Antonova-Koch, Yevgeniya; Crespo, Benigno; de Cózar, Cristina; Sanz, Laura M; Gamo, Francisco Javier; Avery, Vicky M; Frearson, Julie A; Gray, David W; Fairlamb, Alan H; Winzeler, Elizabeth A; Waterson, David; Campbell, Simon F; Willis, Paul A; Read, Kevin D; Gilbert, Ian H

Erratum for Brunschwig et al., "UCT943, a Next-Generation Plasmodium falciparum PI4K Inhibitor Preclinical Candidate for the Treatment of Malaria"

Brunschwig 等人的论文“UCT943,一种用于治疗疟疾的下一代恶性疟原虫 PI4K 抑制剂临床前候选药物”的勘误

Brunschwig, Christel; Lawrence, Nina; Taylor, Dale; Abay, Efrem; Njoroge, Mathew; Basarab, Gregory S; Le Manach, Claire; Paquet, Tanya; Gonzàlez Cabrera, Diego; Nchinda, Aloysius T; de Kock, Carmen; Wiesner, Lubbe; Denti, Paolo; Waterson, David; Blasco, Benjamin; Leroy, Didier; Witty, Michael J; Donini, Cristina; Duffy, James; Wittlin, Sergio; White, Karen L; Charman, Susan A; Jiménez-Díaz, Maria Belén; Angulo-Barturen, Iñigo; Herreros, Esperanza; Gamo, Francisco Javier; Rochford, Rosemary; Mancama, Dalu; Coetzer, Theresa L; van der Watt, Mariëtte E; Reader, Janette; Birkholtz, Lyn-Marie; Marsh, Kennan C; Solapure, Suresh M; Burke, John E; McPhail, Jacob A; Vanaerschot, Manu; Fidock, David A; Fish, Paul V; Siegl, Peter; Smith, Dennis A; Wirjanata, Grennady; Noviyanti, Rintis; Price, Ric N; Marfurt, Jutta; Silue, Kigbafori D; Street, Leslie J; Chibale, Kelly

UCT943, a Next-Generation Plasmodium falciparum PI4K Inhibitor Preclinical Candidate for the Treatment of Malaria

UCT943,一种用于治疗疟疾的下一代恶性疟原虫PI4K抑制剂临床前候选药物

Brunschwig, Christel; Lawrence, Nina; Taylor, Dale; Abay, Efrem; Njoroge, Mathew; Basarab, Gregory S; Le Manach, Claire; Paquet, Tanya; Cabrera, Diego Gonzàlez; Nchinda, Aloysius T; de Kock, Carmen; Wiesner, Lubbe; Denti, Paolo; Waterson, David; Blasco, Benjamin; Leroy, Didier; Witty, Michael J; Donini, Cristina; Duffy, James; Wittlin, Sergio; White, Karen L; Charman, Susan A; Jiménez-Díaz, Maria Belén; Angulo-Barturen, Iñigo; Herreros, Esperanza; Gamo, Francisco Javier; Rochford, Rosemary; Mancama, Dalu; Coetzer, Theresa L; van der Watt, Mariëtte E; Reader, Janette; Birkholtz, Lyn-Marie; Marsh, Kennan C; Solapure, Suresh M; Burke, John E; McPhail, Jacob A; Vanaerschot, Manu; Fidock, David A; Fish, Paul V; Siegl, Peter; Smith, Dennis A; Wirjanata, Grennady; Noviyanti, Rintis; Price, Ric N; Marfurt, Jutta; Silue, Kigbafori D; Street, Leslie J; Chibale, Kelly

Screening a protein kinase inhibitor library against Plasmodium falciparum

筛选针对恶性疟原虫的蛋白激酶抑制剂库

Hallyburton, Irene; Grimaldi, Raffaella; Woodland, Andrew; Baragaña, Beatriz; Luksch, Torsten; Spinks, Daniel; James, Daniel; Leroy, Didier; Waterson, David; Fairlamb, Alan H; Wyatt, Paul G; Gilbert, Ian H; Frearson, Julie A

Triaminopyrimidine is a fast-killing and long-acting antimalarial clinical candidate

三氨基嘧啶是一种速效且长效的抗疟疾候选药物。

Hameed P, Shahul; Solapure, Suresh; Patil, Vikas; Henrich, Philipp P; Magistrado, Pamela A; Bharath, Sowmya; Murugan, Kannan; Viswanath, Pavithra; Puttur, Jayashree; Srivastava, Abhishek; Bellale, Eknath; Panduga, Vijender; Shanbag, Gajanan; Awasthy, Disha; Landge, Sudhir; Morayya, Sapna; Koushik, Krishna; Saralaya, Ramanatha; Raichurkar, Anandkumar; Rautela, Nikhil; Roy Choudhury, Nilanjana; Ambady, Anisha; Nandishaiah, Radha; Reddy, Jitendar; Prabhakar, K R; Menasinakai, Sreenivasaiah; Rudrapatna, Suresh; Chatterji, Monalisa; Jiménez-Díaz, María Belén; Martínez, María Santos; Sanz, Laura María; Coburn-Flynn, Olivia; Fidock, David A; Lukens, Amanda K; Wirth, Dyann F; Bandodkar, Balachandra; Mukherjee, Kakoli; McLaughlin, Robert E; Waterson, David; Rosenbrier-Ribeiro, Lyn; Hickling, Kevin; Balasubramanian, V; Warner, Peter; Hosagrahara, Vinayak; Dudley, Adam; Iyer, Pravin S; Narayanan, Shridhar; Kavanagh, Stefan; Sambandamurthy, Vasan K

MK-5172, a Selective Inhibitor of Hepatitis C Virus NS3/4a Protease with Broad Activity across Genotypes and Resistant Variants

MK-5172,一种选择性抑制丙型肝炎病毒NS3/4a蛋白酶的药物,对多种基因型和耐药变异株均具有广泛活性。

Draper, Michael P; Weir, S; Macone, A; Donatelli, J; Trieber, C A; Tanaka, S K; Levy, Stuart B; P, Shahul Hameed; Solapure, Suresh; Mukherjee, Kakoli; Nandi, Vrinda; Waterson, David; Shandil, Radha; Balganesh, Meenakshi; Sambandamurthy, Vasan K; Raichurkar, Anand Kumar; Deshpande, Abhijeet; Ghosh, Anirban; Awasthy, Disha; Shanbhag, Gajanan; Sheikh, Gulebahar; McMiken, Helen; Puttur, Jayashree; Reddy, Jitendar; Werngren, Jim; Read, Jon; Kumar, Mahesh; R, Manjunatha; Chinnapattu, Murugan; Madhavapeddi, Prashanti; Manjrekar, Praveena; Basu, Reetobrata; Gaonkar, Sheshagiri; Sharma, Sreevalli; Hoffner, Sven; Humnabadkar, Vaishali; Subbulakshmi, Venkita; Panduga, Vijender; Summa, Vincenzo; Ludmerer, Steven W; McCauley, John A; Fandozzi, Christine; Burlein, Christine; Claudio, Giuliano; Coleman, Paul J; DiMuzio, Jillian M; Ferrara, Marco; Filippo, Marcello Di; Gates, Adam T; Graham, Donald J; Harper, Steven; Hazuda, Daria J; Huang, Qian; McHale, Carolyn; Monteagudo, Edith; Pucci, Vincenzo; Rowley, Michael; Rudd, Michael T; Soriano, Aileen; Stahlhut, Mark W; Vacca, Joseph P; Olsen, David B; Liverton, Nigel J; Carroll, Steven S

Screening and hit evaluation of a chemical library against blood-stage Plasmodium falciparum

针对血液期恶性疟原虫的化学库筛选和先导化合物评价

Avery, Vicky M; Bashyam, Sridevi; Burrows, Jeremy N; Duffy, Sandra; Papadatos, George; Puthukkuti, Shyni; Sambandan, Yuvaraj; Singh, Shivendra; Spangenberg, Thomas; Waterson, David; Willis, Paul