日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Oligomerization of transmembrane adenylyl cyclase isoforms

跨膜腺苷酸环化酶同工酶的寡聚化

Aryal, Sadikshya; Tesmer, John J G; Dessauer, Carmen W; Watts, Val J

The ulcerative colitis risk gene adenylyl cyclase 7 restrains the T-helper 2 phenotype and Class II antigen presentation

溃疡性结肠炎风险基因腺苷酸环化酶7抑制T辅助细胞2表型和II类抗原呈递。

Cardinale, Christopher J; Liu, Yichuan; Kevadia, Aayush; Strong, Alanna; Watts, Val J; Hakonarson, Hakon

Discovery of novel and selective GPR17 antagonists as pharmacological tools for developing new therapeutic strategies in diabetes and obesity.

发现新型选择性 GPR17 拮抗剂,作为开发糖尿病和肥胖症新治疗策略的药理学工具。

Zhu Hu, Conley Jason M, Karavadhi Surendra, LaVigne Justin E, Watts Val J, Sun Hongmao, Shen Min, Hall Matthew D, Ren Hongxia, Patnaik Samarjit

Inhibition of adenylyl cyclase 1 (AC1) and exchange protein directly activated by cAMP (EPAC) restores ATP-sensitive potassium (K(ATP)) channel activity after chronic opioid exposure.

抑制腺苷酸环化酶 1 (AC1) 和 cAMP 直接激活的交换蛋白 (EPAC) 可恢复慢性阿片类药物暴露后 ATP 敏感钾 (K(ATP)) 通道的活性

Klein Amanda H, Alam Sabbir, Johnson Kayla, Kriner Christian, Beck Brie, Nelson Bethany, Hill Cassidy, Meyer Belle, Mellang Jonas, Watts Val J

Germline mutations in a G protein identify signaling cross-talk in T cells

G蛋白的种系突变可揭示T细胞中的信号传导串扰

Ham, Hyoungjun; Jing, Huie; Lamborn, Ian T; Kober, Megan M; Koval, Alexey; Berchiche, Yamina A; Anderson, D Eric; Druey, Kirk M; Mandl, Judith N; Isidor, Bertrand; Ferreira, Carlos R; Freeman, Alexandra F; Ganesan, Sundar; Karsak, Meliha; Mustillo, Peter J; Teo, Juliana; Zolkipli-Cunningham, Zarazuela; Chatron, Nicolas; Lecoquierre, François; Oler, Andrew J; Schmid, Jana Pachlopnik; Kuhns, Douglas B; Xu, Xuehua; Hauck, Fabian; Al-Herz, Waleed; Wagner, Matias; Terhal, Paulien A; Muurinen, Mari; Barlogis, Vincent; Cruz, Phillip; Danielson, Jeffrey; Stewart, Helen; Loid, Petra; Rading, Sebastian; Keren, Boris; Pfundt, Rolph; Zarember, Kol A; Vill, Katharina; Potocki, Lorraine; Olivier, Kenneth N; Lesca, Gaetan; Faivre, Laurence; Wong, Melanie; Puel, Anne; Chou, Janet; Tusseau, Maud; Moutsopoulos, Niki M; Matthews, Helen F; Simons, Cas; Taft, Ryan J; Soldatos, Ariane; Masle-Farquhar, Etienne; Pittaluga, Stefania; Brink, Robert; Fink, Danielle L; Kong, Heidi H; Kabat, Juraj; Kim, Woo Sung; Bierhals, Tatjana; Meguro, Kazuyuki; Hsu, Amy P; Gu, Jingwen; Stoddard, Jennifer; Banos-Pinero, Benito; Slack, Maria; Trivellin, Giampaolo; Mazel, Benoît; Soomann, Maarja; Li, Samuel; Watts, Val J; Stratakis, Constantine A; Rodriguez-Quevedo, Maria F; Bruel, Ange-Line; Lipsanen-Nyman, Marita; Saultier, Paul; Jain, Rashmi; Lehalle, Daphne; Torres, Daniel; Sullivan, Kathleen E; Barbarot, Sébastien; Neu, Axel; Duffourd, Yannis; Similuk, Morgan; McWalter, Kirsty; Blanc, Pierre; Bézieau, Stéphane; Jin, Tian; Geha, Raif S; Casanova, Jean-Laurent; Makitie, Outi M; Kubisch, Christian; Edery, Patrick; Christodoulou, John; Germain, Ronald N; Goodnow, Christopher C; Sakmar, Thomas P; Billadeau, Daniel D; Küry, Sébastien; Katanaev, Vladimir L; Zhang, Yu; Lenardo, Michael J; Su, Helen C

Structure of adenylyl cyclase 5 in complex with Gβγ offers insights into ADCY5-related dyskinesia.

腺苷酸环化酶 5 与 Gββ 复合物的结构为 ADCY5 相关运动障碍提供了见解

Yen Yu-Chen, Li Yong, Chen Chun-Liang, Klose Thomas, Watts Val J, Dessauer Carmen W, Tesmer John J G

Biochemical pharmacology of adenylyl cyclases in cancer

癌症中腺苷酸环化酶的生化药理学

Chandra Jena, Bikash; Flaherty, Daniel P; O'Brien, Valerie P; Watts, Val J

Discovery of a potent and selective human AC2 inhibitor based on 7-deazapurine analogues of adefovir.

基于阿德福韦的 7-脱氮嘌呤类似物,发现了一种强效且选择性的人类 AC2 抑制剂

Kraina Pavel, Česnek Michal, Tloušťová Eva, Mertlíková-Kaiserová Helena, Fulton Camryn J, Davidson Emily K, Smith Brenton P, Watts Val J, Janeba Zlatko

Isoform Specific Regulation of Adenylyl Cyclase 5 by Gβγ

Gβγ对腺苷酸环化酶5的同工型特异性调控

Yen, Yu-Chen; Li, Yong; Chen, Chun-Liang; Klose, Thomas; Watts, Val J; Dessauer, Carmen W; Tesmer, John J G

Physiological roles of mammalian transmembrane adenylyl cyclase isoforms

哺乳动物跨膜腺苷酸环化酶同工酶的生理作用

Ostrom, Katrina F; LaVigne, Justin E; Brust, Tarsis F; Seifert, Roland; Dessauer, Carmen W; Watts, Val J; Ostrom, Rennolds S