Brigatinib causes tumor shrinkage in both NF2-deficient meningioma and schwannoma through inhibition of multiple tyrosine kinases but not ALK
布加替尼通过抑制多种酪氨酸激酶(但不抑制 ALK)导致 NF2 缺陷型脑膜瘤和神经鞘瘤的肿瘤缩小
期刊:PLoS One
影响因子:2.9
doi:10.1371/journal.pone.0252048
Long-Sheng Chang, Janet L Oblinger, Abbi E Smith, Marc Ferrer, Steven P Angus, Eric Hawley, Alejandra M Petrilli, Roberta L Beauchamp, Lars Björn Riecken, Serkan Erdin, Ming Poi, Jie Huang, Waylan K Bessler, Xiaohu Zhang, Rajarshi Guha, Craig Thomas, Sarah S Burns, Thomas S K Gilbert, Li Jiang, Xiao