日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of 2-Amide-3-methylester Thiophenes that Target SARS-CoV-2 Mac1 and Repress Coronavirus Replication, Validating Mac1 as an Antiviral Target.

发现靶向 SARS-CoV-2 Mac1 并抑制冠状病毒复制的 2-酰胺-3-甲基酯噻吩类化合物,验证 Mac1 作为抗病毒靶点

Wazir Sarah, Parviainen Tomi A O, Pfannenstiel Jessica J, Duong Men Thi Hoai, Cluff Daniel, Sowa Sven T, Galera-Prat Albert, Ferraris Dana, Maksimainen Mirko M, Fehr Anthony R, Heiskanen Juha P, Lehtiö Lari

Discovery of compounds that inhibit SARS-CoV-2 Mac1-ADP-ribose binding by high-throughput screening.

利用高通量筛选发现抑制SARS-CoV-2 Mac1-ADP-核糖结合的化合物

Roy Anu, Alhammad Yousef M, McDonald Peter, Johnson David K, Zhuo Junlin, Wazir Sarah, Ferraris Dana, Lehtiö Lari, Leung Anthony K L, Fehr Anthony R

Macrodomain Binding Compound MRS 2578 Inhibits Alphavirus Replication

宏结构域结合化合物MRS 2578抑制甲病毒复制

Mattila, Sari; Merilahti, Pirjo; Wazir, Sarah; Quirin, Tania; Maksimainen, Mirko M; Zhang, Yuezhou; Xhaard, Henri; Lehtiö, Lari; Ahola, Tero

Multiple crystal forms of human MacroD2

人类MacroD2的多种晶体形式

Wazir, Sarah; Maksimainen, Mirko M; Lehtiö, Lari