Discovery of 2-Amide-3-methylester Thiophenes that Target SARS-CoV-2 Mac1 and Repress Coronavirus Replication, Validating Mac1 as an Antiviral Target.
发现靶向 SARS-CoV-2 Mac1 并抑制冠状病毒复制的 2-酰胺-3-甲基酯噻吩类化合物,验证 Mac1 作为抗病毒靶点
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.3c02451
Wazir Sarah, Parviainen Tomi A O, Pfannenstiel Jessica J, Duong Men Thi Hoai, Cluff Daniel, Sowa Sven T, Galera-Prat Albert, Ferraris Dana, Maksimainen Mirko M, Fehr Anthony R, Heiskanen Juha P, Lehtiö Lari