日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Optimization of Cyclophilin B-Targeted Tri-vector Inhibitors for Novel MASH Treatments

针对环孢素B靶向的三载体抑制剂的优化及其在新型MASH治疗中的应用

Kouridaki, Maria-Eleni; Gillespie, Jonathan; Robinson, John; Mathie, Tanya; Bain, Laura; McArthur, Duncan; Morrison, Angus; Greenslade, Daniel B; Papadourakis, Michail; Maj, Kasia; Cameron, Kate; Turner, Darryl; Webster, Scott P; Wear, Martin A; Doughty-Shenton, Dahlia; Hulme, Alison N; Michel, Julien

Redox regulation of pyruvate kinase M2 by cysteine oxidation and S-nitrosation.

半胱氨酸氧化和S-亚硝化对丙酮酸激酶M2的氧化还原调控

Mitchell Alice Rose, Yuan Meng, Morgan Hugh P, McNae Iain W, Blackburn Elizabeth A, Le Bihan Thierry, Homem Rafael A, Yu Manda, Loake Gary J, Michels Paul A, Wear Martin A, Walkinshaw Malcolm D

Molecular basis for Cdk1-regulated timing of Mis18 complex assembly and CENP-A deposition

Cdk1调控Mis18复合物组装和CENP-A沉积的分子机制

Spiller, Frances; Medina-Pritchard, Bethan; Abad, Maria Alba; Wear, Martin A; Molina, Oscar; Earnshaw, William C; Jeyaprakash, A Arockia

Cyclophilin40 isomerase activity is regulated by a temperature-dependent allosteric interaction with Hsp90

环孢亲和素40异构酶活性受与Hsp90的温度依赖性变构相互作用调控。

Blackburn, Elizabeth A; Wear, Martin A; Landré, Vivian; Narayan, Vikram; Ning, Jia; Erman, Burak; Ball, Kathryn L; Walkinshaw, Malcolm D

A new family of covalent inhibitors block nucleotide binding to the active site of pyruvate kinase.

一类新型共价抑制剂可阻断核苷酸与丙酮酸激酶活性位点的结合

Morgan Hugh P, Walsh Martin J, Blackburn Elizabeth A, Wear Martin A, Boxer Matthew B, Shen Min, Veith Henrike, McNae Iain W, Nowicki Matthew W, Michels Paul A M, Auld Douglas S, Fothergill-Gilmore Linda A, Walkinshaw Malcolm D

The mitosis and neurodevelopment proteins NDE1 and NDEL1 form dimers, tetramers, and polymers with a folded back structure in solution

有丝分裂和神经发育蛋白NDE1和NDEL1在溶液中形成二聚体、四聚体和具有折叠结构的聚合物。

Soares, Dinesh C; Bradshaw, Nicholas J; Zou, Juan; Kennaway, Christopher K; Hamilton, Russell S; Chen, Zhuo A; Wear, Martin A; Blackburn, Elizabeth A; Bramham, Janice; Böttcher, Bettina; Millar, J Kirsty; Barlow, Paul N; Walkinshaw, Malcolm D; Rappsilber, Juri; Porteous, David J

A t(1;11) translocation linked to schizophrenia and affective disorders gives rise to aberrant chimeric DISC1 transcripts that encode structurally altered, deleterious mitochondrial proteins

与精神分裂症和情感障碍相关的t(1;11)易位导致异常嵌合DISC1转录本的产生,这些转录本编码结构改变的有害线粒体蛋白。

Eykelenboom, Jennifer E; Briggs, Gareth J; Bradshaw, Nicholas J; Soares, Dinesh C; Ogawa, Fumiaki; Christie, Sheila; Malavasi, Elise L V; Makedonopoulou, Paraskevi; Mackie, Shaun; Malloy, Mary P; Wear, Martin A; Blackburn, Elizabeth A; Bramham, Janice; McIntosh, Andrew M; Blackwood, Douglas H; Muir, Walter J; Porteous, David J; Millar, J Kirsty

Crystallization and X-ray structure of cold-shock protein E from Salmonella typhimurium

鼠伤寒沙门氏菌冷休克蛋白E的结晶和X射线结构

Morgan, Hugh P; Wear, Martin A; McNae, Iain; Gallagher, Maurice P; Walkinshaw, Malcolm D

Mammalian CARMIL inhibits actin filament capping by capping protein

哺乳动物 CARMIL 通过帽状蛋白抑制肌动蛋白丝帽状化。

Yang, Changsong; Pring, Martin; Wear, Martin A; Huang, Minzhou; Cooper, John A; Svitkina, Tatyana M; Zigmond, Sally H

Biological role and structural mechanism of twinfilin-capping protein interaction

双丝蛋白-帽蛋白相互作用的生物学作用和结构机制

Falck, Sandra; Paavilainen, Ville O; Wear, Martin A; Grossmann, J Günter; Cooper, John A; Lappalainen, Pekka