Discovery of Pan-TEAD Inhibitors That Disrupt YAP-TEAD Interaction as a Potential Therapy for Gastric Cancers and Mutant KRAS and EGFR Lung Cancers
发现可破坏YAP-TEAD相互作用的泛TEAD抑制剂,有望成为胃癌以及KRAS和EGFR突变型肺癌的潜在疗法
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.5c00590
Kumar, Ramesh; Thian, Joanne; Toh, Joel D W; Farzana, Noorul; Sun, Jialin; Kang, CongBao; Low, Suet Mei Crystal; Wee, Sheena; Lim, Zijie; Gunaratne, Jayantha; Loh, Hui Mun; Kannan, Srinivasaraghavan; Verma, Chandra S; Chakraborty, Sayan; Hong, Wanjin