日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Correction: Identification of acrylamide-based covalent inhibitors of SARS-CoV-2 (SCoV-2) Nsp15 using high-throughput screening and machine learning

更正:利用高通量筛选和机器学习鉴定基于丙烯酰胺的SARS-CoV-2 (SCoV-2) Nsp15共价抑制剂

Bajaj, Teena; Mosavati, Babak; Zhang, Lydia H; Parsa, Mohammad S; Wang, Huanchen; Kerek, Evan M; Liang, Xueying; Tabatabaei Dakhili, Seyed Amir; Wehri, Eddie; Guo, Silin; Desai, Rushil N; Orr, Lauren M; Mofrad, Mohammad R K; Schaletzky, Julia; Ussher, John R; Deng, Xufang; Stanley, Robin; Hubbard, Basil P; Nomura, Daniel K; Murthy, Niren

Identification of acrylamide-based covalent inhibitors of SARS-CoV-2 (SCoV-2) Nsp15 using high-throughput screening and machine learning.

利用高通量筛选和机器学习鉴定 SARS-CoV-2 (SCoV-2) Nsp15 的丙烯酰胺基共价抑制剂

Bajaj Teena, Mosavati Babak, Zhang Lydia H, Parsa Mohammad S, Wang Huanchen, Kerek Evan M, Liang Xueying, Tabatabaei Dakhili Seyed Amir, Wehri Eddie, Guo Silin, Desai Rushil N, Orr Lauren M, Mofrad Mohammad R K, Schaletzky Julia, Ussher John R, Deng Xufang, Stanley Robin, Hubbard Basil P, Nomura Daniel K, Murthy Niren

Aficamten is a small-molecule cardiac myosin inhibitor designed to treat hypertrophic cardiomyopathy

Aficamten是一种小分子心肌肌球蛋白抑制剂,旨在治疗肥厚型心肌病。

Hartman, James J; Hwee, Darren T; Robert-Paganin, Julien; Chuang, Chihyuan; Chin, Eva R; Edell, Samantha; Lee, Ken H; Madhvani, Roshni; Paliwal, Preeti; Pernier, Julien; Sarkar, Saswata Sankar; Schaletzky, Julia; Schauer, Kristine; Taheri, Khanha D; Wang, Jingying; Wehri, Eddie; Wu, Yangsong; Houdusse, Anne; Morgan, Bradley P; Malik, Fady I

MyosinA is a druggable target in the widespread protozoan parasite Toxoplasma gondii

肌球蛋白A是广泛分布的原生动物寄生虫弓形虫的一个可药物靶点。

Kelsen, Anne; Kent, Robyn S; Snyder, Anne K; Wehri, Eddie; Bishop, Stephen J; Stadler, Rachel V; Powell, Cameron; Martorelli di Genova, Bruno; Rompikuntal, Pramod K; Boulanger, Martin J; Warshaw, David M; Westwood, Nicholas J; Schaletzky, Julia; Ward, Gary E

SARS-CoV-2 nucleocapsid protein forms condensates with viral genomic RNA

SARS-CoV-2 核衣壳蛋白与病毒基因组 RNA 形成凝聚体

Jack, Amanda; Ferro, Luke S; Trnka, Michael J; Wehri, Eddie; Nadgir, Amrut; Nguyenla, Xammy; Costa, Katelyn; Stanley, Sarah; Schaletzky, Julia; Yildiz, Ahmet