日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structural basis for selective inhibition of human GABA transporter GAT3

选择性抑制人GABA转运蛋白GAT3的结构基础

Mortensen, Jonas Sigurd; Bavo, Francesco; Jensen, Malene Hall; Pedersen, Alexander Peder Smiszek; Storm, Julian Philipp; Pape, Tillmann; Frølund, Bente; Wellendorph, Petrine; Shahsavar, Azadeh

Allosteric factors in the calcium/calmodulin-responsive kinase II hub domain determine selectivity of GHB ligands for CaMKIIα

钙/钙调蛋白反应性激酶II枢纽结构域中的变构因子决定了GHB配体对CaMKIIα的选择性

Gauger, Stine J; Palmelund, Line B; Tian, Yongsong; Marek, Aleš; Namini, Mathias R; Griem-Krey, Nane; Petersen, Madeline Y; Kickinger, Stefanie; Mortensen, Jonas S; Frølund, Bente; Wellendorph, Petrine

Radiofluorinated Analogs of NCS-382 as Potential PET Tracers for Imaging the CaMKIIα Hub Domain

NCS-382 的放射性氟化类似物作为潜在的 PET 示踪剂用于 CaMKIIα 中心结构域的成像

Sirocchi, Ludovica S; Stotz, Sophie; Müller, Marius; Pedersen, Nadia Billesborg; Thiesen, Louise; Mattiussi, Simona; Avgerinos, Christos; Shalgunov, Vladimir; Wellendorph, Petrine; Fro̷lund, Bente; Herth, Matthias M

Systemic antibiotics for Pseudomonas aeruginosa infection in outpatients with non-hospitalised exacerbations of pre-existing lung diseases: a randomised clinical trial

门诊患者非住院急性加重合并铜绿假单胞菌感染的全身性抗生素治疗:一项随机临床试验

Eklöf, Josefin; Alispahic, Imane Achir; Armbruster, Karin; Lapperre, Therese Sophie; Browatzki, Andrea; Overgaard, Rikke Holmen; Harboe, Zitta Barrella; Janner, Julie; Moberg, Mia; Ulrik, Charlotte Suppli; Andreassen, Helle Frost; Weinreich, Ulla Møller; Kjærgaard, Jakob Lyngby; Villadsen, Jenny; Fenlev, Camilla Sund; Jensen, Torben Tranborg; Christensen, Christina Wellendorph; Bangsborg, Jette; Ostergaard, Christian; Ghathian, Khaled Saoud Ali; Jordan, Alexander; Klausen, Tobias Wirenfeldt; Nielsen, Thyge Lynghøj; Wilcke, Torgny; Seersholm, Niels; Sivapalan, Pradeesh; Jensen, Jens-Ulrik Stæhr

Ligand-induced CaMKIIα hub Trp403 flip, hub domain stacking, and modulation of kinase activity

配体诱导的 CaMKIIα 枢纽 Trp403 翻转、枢纽域堆积和激酶活性调节

Dilip Narayanan, Anne Sofie G Larsen, Stine Juul Gauger, Ruth Adafia, Rikke Bartschick Hammershøi, Louise Hamborg, Jesper Bruus-Jensen, Nane Griem-Krey, Christine L Gee, Bente Frølund, Margaret M Stratton, John Kuriyan, Jette Sandholm Kastrup, Annette E Langkilde, Petrine Wellendorph, Sara M Ø Solba

Rodent ischemic stroke models and their relevance in preclinical research

啮齿动物缺血性中风模型及其在临床前研究中的意义

Thaysen, Maria; Westi, Emil; Clarkson, Andrew N; Wellendorph, Petrine; Kristensen, Mie

The GHB analogue HOCPCA improves deficits in cognition and sensorimotor function after MCAO via CaMKIIα

GHB 类似物 HOCPCA 通过 CaMKIIα 改善 MCAO 后的认知和感觉运动功能障碍

Nane Griem-Krey, Anders B Klein, Bettina H Clausen, Mathias Rj Namini, Pernille V Nielsen, Mozammel Bhuiyan, Raghavendra Y Nagaraja, T Michael De Silva, Christopher G Sobey, Heung-Chin Cheng, Cyrille Orset, Denis Vivien, Kate L Lambertsen, Andrew N Clarkson, Petrine Wellendorph

Elucidating Pathway and Anesthetic Mechanism of Action of Clove Oil Nanoformulations in Fish

阐明丁香油纳米制剂在鱼类中的作用途径和麻醉机制

Kheawfu, Kantaporn; Pikulkaew, Surachai; Wellendorph, Petrine; Jørgensen, Louise von Gersdorff; Rades, Thomas; Müllertz, Anette; Okonogi, Siriporn

The Binding of Alpinia galanga Oil and Its Nanoemulsion to Mammal GABA(A) Receptors Using Rat Cortical Membranes and an In Silico Modeling Platform

利用大鼠皮质膜和计算机模拟平台研究高良姜油及其纳米乳液与哺乳动物GABA(A)受体的结合

Khumpirapang, Nattakanwadee; Suknuntha, Krit; Wongrattanakamon, Pathomwat; Jiranusornkul, Supat; Anuchapreeda, Songyot; Wellendorph, Petrine; Müllertz, Anette; Rades, Thomas; Okonogi, Siriporn

GHB analogs confer neuroprotection through specific interaction with the CaMKIIα hub domain

GHB类似物通过与CaMKIIα枢纽结构域的特异性相互作用发挥神经保护作用。

Leurs, Ulrike; Klein, Anders B; McSpadden, Ethan D; Griem-Krey, Nane; Solbak, Sara M Ø; Houlton, Josh; Villumsen, Inge S; Vogensen, Stine B; Hamborg, Louise; Gauger, Stine J; Palmelund, Line B; Larsen, Anne Sofie G; Shehata, Mohamed A; Kelstrup, Christian D; Olsen, Jesper V; Bach, Anders; Burnie, Robert O; Kerr, D Steven; Gowing, Emma K; Teurlings, Selina M W; Chi, Chris C; Gee, Christine L; Frølund, Bente; Kornum, Birgitte R; van Woerden, Geeske M; Clausen, Rasmus P; Kuriyan, John; Clarkson, Andrew N; Wellendorph, Petrine