日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structural Studies of βTrCP Reveal Plasticity in Binding Modes of Consensus and Nonconsensus Degrons

βTrCP的结构研究揭示了其与共有序列和非共有序列降解子结合模式的可塑性。

Collie, Gavin W; Mak, Hazel; Acebrón-García-de-Eulate, Marta; Argyrou, Argyrides; Couturier, Maxime; Cuomo, Maria Emanuela; O Donovan, Daniel H; Russell, Isabella C; Wells, Geoffrey; Winter-Holt, Jon

CACHE Challenge #2: Targeting the RNA Site of the SARS-CoV-2 Helicase Nsp13

CACHE挑战#2:靶向SARS-CoV-2解旋酶Nsp13的RNA位点

Herasymenko, Oleksandra; Silva, Madhushika; Abu-Saleh, Abd Al-Aziz A; Ahmad, Ayaz; Alvarado-Huayhuaz, Jesus; Arce, Oscar E A; Armstrong, Roly J; Arrowsmith, Cheryl; Bachta, Kelly E; Beck, Hartmut; Berta, Denes; Bieniek, Mateusz K; Blay, Vincent; Bolotokova, Albina; Bourne, Philip E; Breznik, Marko; Brown, Peter J; Campbell, Aaron D G; Carosati, Emanuele; Chau, Irene; Cole, Daniel J; Cree, Ben; Dehaen, Wim; Denzinger, Katrin; Dos Santos Machado, Karina; Dunn, Ian; Durai, Prasannavenkatesh; Edfeldt, Kristina; Edwards, Aled; Fayne, Darren; Felfoldi, Daniel; Friston, Kallie; Ghiabi, Pegah; Gibson, Elisa; Günther, Judith; Gunnarsson, Anders; Hillisch, Alexander; Houston, Douglas R; Jensen, Jan Halborg; Harding, Rachel J; Harris, Kate S; Hoffer, Laurent; Hogner, Anders; Horton, Joshua T; Houliston, Scott; Hultquist, Judd F; Hutchinson, Ashley; Irwin, John J; Jukič, Marko; Kandwal, Shubhangi; Karlova, Andrea; Katis, Vittorio L; Kich, Ryan P; Kireev, Dmitri; Koes, David; Inniss, Nicole L; Lessel, Uta; Liu, Sijie; Loppnau, Peter; Lu, Wei; Martino, Sam; McGibbon, Miles; Meiler, Jens; Mettu, Akhila; Money-Kyrle, Sam; Moretti, Rocco; Moroz, Yurii S; Muvva, Charuvaka; Newman, Joseph A; Obendorf, Leon; Paige, Brooks; Pandit, Amit; Park, Keunwan; Perveen, Sumera; Pirie, Rachael; Poda, Gennady; Protopopov, Mykola; Pütter, Vera; Ricci, Federico; Roper, Natalie J; Rosta, Edina; Rzhetskaya, Margarita; Sabnis, Yogesh; Satchell, Karla J F; Schmitt Kremer, Frederico; Scott, Thomas; Seitova, Almagul; Steinmann, Casper; Talagayev, Valerij; Tarkhanova, Olga O; Tatum, Natalie J; Treleaven, Dakota; Velasque Werhli, Adriano; Walters, W Patrick; Wang, Xiaowen; Wells, Jude; Wells, Geoffrey; Westermaier, Yvonne; Wolber, Gerhard; Wortmann, Lars; Zhang, Jixian; Zhao, Zheng; Zheng, Shuangjia; Schapira, Matthieu

Fragment-based drug discovery: A graphical review

基于片段的药物发现:图解综述

AlKharboush, Dana F; Kozielski, Frank; Wells, Geoffrey; Porta, Exequiel O J

Basal activation of astrocytic Nrf2 in neuronal culture media: Challenges and implications for neuron-astrocyte modelling.

神经元培养基中星形胶质细胞 Nrf2 的基础激活:神经元-星形胶质细胞建模的挑战和意义

Elsharkasi Mohamed Moftah Omer, Villani Beatrice, Wells Geoffrey, Kerr Fiona

C2-linked alkynyl poly-ethylene glycol(PEG) adenosine conjugates as water-soluble adenosine receptor agonists

C2连接的炔基聚乙二醇(PEG)腺苷缀合物作为水溶性腺苷受体激动剂

Ferguson, Lindsay; Madieh, Nasrin Shokrzadeh; Vaideanu, Alexandra; Schatzlein, Andreas; Festa, Joseph; Singh, Harprit; Wells, Geoffrey; Bhakta, Sanjib; Brucoli, Federico

The C-terminal head domain of Burkholderia pseudomallei BpaC has a striking hydrophilic core with an extensive solvent network

类鼻疽伯克霍尔德菌BpaC的C端头部结构域具有显著的亲水核心和广泛的溶剂网络。

Kiessling, Andreas R; Harris, Sarah A; Weimer, Kathleen M; Wells, Geoffrey; Goldman, Adrian

Intelligent resolution: Integrating Cryo-EM with AI-driven multi-resolution simulations to observe the severe acute respiratory syndrome coronavirus-2 replication-transcription machinery in action

智能分辨率:将冷冻电镜与人工智能驱动的多分辨率模拟相结合,观察严重急性呼吸综合征冠状病毒2复制转录机制的运作过程。

Trifan, Anda; Gorgun, Defne; Salim, Michael; Li, Zongyi; Brace, Alexander; Zvyagin, Maxim; Ma, Heng; Clyde, Austin; Clark, David; Hardy, David J; Burnley, Tom; Huang, Lei; McCalpin, John; Emani, Murali; Yoo, Hyenseung; Yin, Junqi; Tsaris, Aristeidis; Subbiah, Vishal; Raza, Tanveer; Liu, Jessica; Trebesch, Noah; Wells, Geoffrey; Mysore, Venkatesh; Gibbs, Thomas; Phillips, James; Chennubhotla, S Chakra; Foster, Ian; Stevens, Rick; Anandkumar, Anima; Vishwanath, Venkatram; Stone, John E; Tajkhorshid, Emad; A Harris, Sarah; Ramanathan, Arvind

Atomic force microscopy-A tool for structural and translational DNA research

原子力显微镜——用于DNA结构和转化研究的工具

Main, Kavit H S; Provan, James I; Haynes, Philip J; Wells, Geoffrey; Hartley, John A; Pyne, Alice L B

Protein Encapsulation of Experimental Anticancer Agents 5F 203 and Phortress: Towards Precision Drug Delivery

实验性抗癌药物 5F 203 和 Phortress 的蛋白质封装:迈向精准药物递送

Breen, Alastair F; Scurr, David; Cassioli, Maria Letizia; Wells, Geoffrey; Thomas, Neil R; Zhang, Jihong; Turyanska, Lyudmila; Bradshaw, Tracey D

Development of novel apoferritin formulations for antitumour benzothiazoles

开发用于抗肿瘤苯并噻唑类药物的新型脱铁蛋白制剂

Breen, Alastair F; Wells, Geoffrey; Turyanska, Lyudmila; Bradshaw, Tracey D