日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Equipotent enantiomers of cyclic opioid peptides at μ opioid receptor

环状阿片肽对 μ 阿片受体的等效对映体

Grazyna Weltrowska, Thi M-D Nguyen, Nga N Chung, Brian C Wilkes, Peter W Schiller

N-terminal guanidinylation of TIPP (Tyr-Tic-Phe-Phe) peptides results in major changes of the opioid activity profile

TIPP(Tyr-Tic-Phe-Phe)肽的N端胍基化会导致阿片类活性谱发生显著变化。

Weltrowska, Grazyna; Nguyen, Thi M-D; Chung, Nga N; Wilkes, Brian C; Schiller, Peter W

"Carba"-analogues of fentanyl are opioid receptor agonists

芬太尼的“卡巴”类似物是阿片受体激动剂。

Weltrowska, Grazyna; Chung, Nga N; Lemieux, Carole; Guo, Jianxin; Lu, Yixin; Wilkes, Brian C; Schiller, Peter W

N-methylated cyclic enkephalin analogues retain high opioid receptor binding affinity

N-甲基化环状脑啡肽类似物保留了较高的阿片受体结合亲和力

Grazyna Weltrowska, Irena Berezowska, Carole Lemieux, Nga N Chung, Brian C Wilkes, Peter W Schiller

Stereoselective synthesis of (3S)- and (3R)-3-hydroxy-3-(2,6-dimethyl-4-hydroxyphenyl)propanoic acid and its incorporation into a cyclic enkephalin analogue

(3S)-和(3R)-3-羟基-3-(2,6-二甲基-4-羟基苯基)丙酸的立体选择性合成及其在环状脑啡肽类似物中的应用

Weltrowska, Grazyna; Lemieux, Carole; Chung, Nga N; Wilkes, Brian C; Schiller, Peter W