日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Efficacy of ATR Kinase Inhibitor Elimusertib Monotherapy or Combination in Tumors with DNA Damage Response Pathway and Other Genomic Alterations.

ATR激酶抑制剂Elimusertib单药或联合治疗对具有DNA损伤反应通路和其他基因组改变的肿瘤的疗效

Varadarajan Kaushik, Cruz Pico Christian X, Evans Kurt W, Raso Maria Gabriela, Rizvi Yasmeen Qamar, Zheng Xiaofeng, Chachad Dhruv, DiPeri Timothy P, Wang Bailiang, Scott Stephen M, Zhao Ming, Akcakanat Argun, Wengner Antje M, Yap Timothy A, Meric-Bernstam Funda

Dryinones: Structure Elucidation of Red Colorants from Submerged Cultures of Pleurotus dryinus

干侧耳酮:干侧耳深层培养红色色素的结构解析

Broel, Niklas; Stein, Johanna V; Wengner, Franziska V; Domanski, Marvin H J; Zhuk, Tatyana; Gand, Martin

Discovery of IRAK4 Inhibitors BAY1834845 (Zabedosertib) and BAY1830839

发现 IRAK4 抑制剂 BAY1834845 (Zabedosertib) 和 BAY1830839

Bothe, Ulrich; Günther, Judith; Nubbemeyer, Reinhard; Siebeneicher, Holger; Ring, Sven; Bömer, Ulf; Peters, Michaele; Rausch, Alexandra; Denner, Karsten; Himmel, Herbert; Sutter, Andreas; Terebesi, Ildiko; Lange, Martin; Wengner, Antje M; Guimond, Nicolas; Thaler, Tobias; Platzek, Johannes; Eberspächer, Uwe; Schäfer, Martina; Steuber, Holger; Zollner, Thomas M; Steinmeyer, Andreas; Schmidt, Nicole

Elimusertib has Antitumor Activity in Preclinical Patient-Derived Pediatric Solid Tumor Models

Elimusertib在临床前患者来源的儿科实体瘤模型中具有抗肿瘤活性

Pusch, Fabian F; Dorado García, Heathcliff; Xu, Robin; Gürgen, Dennis; Bei, Yi; Brückner, Lotte; Röefzaad, Claudia; von Stebut, Jennifer; Bardinet, Victor; Chamorro Gonzalez, Rocío; Eggert, Angelika; Schulte, Johannes H; Hundsdörfer, Patrick; Seifert, Georg; Haase, Kerstin; Schäfer, Beat W; Wachtel, Marco; Kühl, Anja A; Ortiz, Michael V; Wengner, Antje M; Scheer, Monika; Henssen, Anton G

The ATR inhibitor elimusertib exhibits anti-lymphoma activity and synergizes with the PI3K inhibitor copanlisib

ATR 抑制剂 elimusertib 具有抗淋巴瘤活性,并与 PI3K 抑制剂 copanlisib 产生协同作用

Giulio Sartori, Chiara Tarantelli, Filippo Spriano, Eugenio Gaudio, Luciano Cascione, Michele Mascia, Marilia Barreca, Alberto J Arribas, Luca Licenziato, Gaetanina Golino, Adele Ferragamo, Stefano Pileri, Giovanna Damia, Emanuele Zucca, Anastasios Stathis, Oliver Politz, Antje M Wengner, Francesco

Nuclear pCHK1 as a potential biomarker of increased sensitivity to ATR inhibition

核 pCHK1 是 ATR 抑制敏感性增加的潜在生物标志物

Vignesh Sundararajan, Tuan Zea Tan, Diana Lim, Yanfen Peng, Antje Margret Wengner, Natalie Yan Li Ngoi, Anand D Jeyasekharan, David Shao Peng Tan

A Novel NAMPT Inhibitor-Based Antibody-Drug Conjugate Payload Class for Cancer Therapy

一种新型的基于NAMPT抑制剂的抗体-药物偶联物有效载荷用于癌症治疗

Böhnke, Niels; Berger, Markus; Griebenow, Nils; Rottmann, Antje; Erkelenz, Michael; Hammer, Stefanie; Berndt, Sandra; Günther, Judith; Wengner, Antje M; Stelte-Ludwig, Beatrix; Mahlert, Christoph; Greven, Simone; Dietz, Lisa; Jörißen, Hannah; Barak, Naomi; Bömer, Ulf; Hillig, Roman C; Eberspaecher, Uwe; Weiske, Jörg; Giese, Anja; Mumberg, Dominik; Nising, Carl Friedrich; Weinmann, Hilmar; Sommer, Anette

Targeted thorium-227 conjugates as treatment options in oncology

靶向钍-227偶联物作为肿瘤治疗选择

Karlsson, Jenny; Schatz, Christoph A; Wengner, Antje M; Hammer, Stefanie; Scholz, Arne; Cuthbertson, Alan; Wagner, Volker; Hennekes, Hartwig; Jardine, Vicki; Hagemann, Urs B

First-in-Human Trial of the Oral Ataxia Telangiectasia and RAD3-Related (ATR) Inhibitor BAY 1895344 in Patients with Advanced Solid Tumors

首次人体试验:口服共济失调毛细血管扩张症和RAD3相关(ATR)抑制剂BAY 1895344治疗晚期实体瘤患者

Yap, Timothy A; Tan, David S P; Terbuch, Angelika; Caldwell, Reece; Guo, Christina; Goh, Boon Cher; Heong, Valerie; Haris, Noor R Md; Bashir, Saira; Drew, Yvette; Hong, David S; Meric-Bernstam, Funda; Wilkinson, Gary; Hreiki, Joseph; Wengner, Antje M; Bladt, Friedhelm; Schlicker, Andreas; Ludwig, Matthias; Zhou, Yinghui; Liu, Li; Bordia, Sonal; Plummer, Ruth; Lagkadinou, Eleni; de Bono, Johann S

BAY-8400: A Novel Potent and Selective DNA-PK Inhibitor which Shows Synergistic Efficacy in Combination with Targeted Alpha Therapies

BAY-8400:一种新型强效选择性 DNA-PK 抑制剂,与靶向 Alpha 疗法联合使用可发挥协同作用

Markus Berger, Lars Wortmann, Philipp Buchgraber, Ulrich Lücking, Sabine Zitzmann-Kolbe, Antje M Wengner, Benjamin Bader, Ulf Bömer, Hans Briem, Knut Eis, Hartmut Rehwinkel, Florian Bartels, Dieter Moosmayer, Uwe Eberspächer, Philip Lienau, Stefanie Hammer, Christoph A Schatz, Qiuwen Wang, Qi Wang,