日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

From Inhibitors to PET: SAR-Based Development of [(18)F]SK60 for mIDH1 Imaging.

从抑制剂到 PET:基于 SAR 的 [(18)F]SK60 在 mIDH1 成像中的开发

Kaur Sarandeep, Dukic-Stefanovic Sladjana, Deuther-Conrad Winnie, Toussaint Magali, Wenzel Barbara, Lönnecke Peter, Donat Cornelius K, Moldovan Rareş-Petru, Kopka Klaus

Radiosynthesis and biological evaluation of [(18)F]AG-120 for PET imaging of the mutant isocitrate dehydrogenase 1 in glioma

[(18)F]AG-120 的放射合成和生物学评价,用于胶质瘤中突变异柠檬酸脱氢酶 1 的 PET 成像

Lai, Thu Hang; Wenzel, Barbara; Dukić-Stefanović, Sladjana; Teodoro, Rodrigo; Arnaud, Lucie; Maisonial-Besset, Aurélie; Weber, Valérie; Moldovan, Rareş-Petru; Meister, Sebastian; Pietzsch, Jens; Kopka, Klaus; Juratli, Tareq A; Deuther-Conrad, Winnie; Toussaint, Magali

Correction to: Radiosynthesis and biological evaluation of [(18)F]AG-120 for PET imaging of the mutant isocitrate dehydrogenase 1 in glioma

更正:[(18)F]AG-120 的放射合成和生物学评价用于胶质瘤中突变异柠檬酸脱氢酶 1 的 PET 成像

Lai, Thu Hang; Wenzel, Barbara; Dukić-Stefanović, Sladjana; Teodoro, Rodrigo; Arnaud, Lucie; Maisonial-Besset, Aurélie; Weber, Valérie; Moldovan, Rareş-Petru; Meister, Sebastian; Pietzsch, Jens; Kopka, Klaus; Juratli, Tareq A; Deuther-Conrad, Winnie; Toussaint, Magali

Synthesis, Structure-Activity Relationships, Radiofluorination, and Biological Evaluation of [(18)F]RM365, a Novel Radioligand for Imaging the Human Cannabinoid Receptor Type 2 (CB2R) in the Brain with PET

本文研究了新型放射性配体[(18)F]RM365的合成、构效关系、放射性氟化及其在PET成像中对人脑内大麻素受体2型(CB2R)的生物学评价。

Teodoro, Rodrigo; Gündel, Daniel; Deuther-Conrad, Winnie; Kazimir, Aleksandr; Toussaint, Magali; Wenzel, Barbara; Bormans, Guy; Hey-Hawkins, Evamarie; Kopka, Klaus; Brust, Peter; Moldovan, Rareş-Petru

Efficacy and safety of cotadutide, a dual glucagon-like peptide-1 and glucagon receptor agonist, in a randomized phase 2a study of patients with type 2 diabetes and chronic kidney disease

一项针对2型糖尿病合并慢性肾病患者的随机2a期研究评估了双重胰高血糖素样肽-1和胰高血糖素受体激动剂cotadutide的疗效和安全性。

Parker, Victoria E R; Hoang, Thuong; Schlichthaar, Heike; Gibb, Fraser W; Wenzel, Barbara; Posch, Maximillian G; Rose, Ludger; Chang, Yi-Ting; Petrone, Marcella; Hansen, Lars; Ambery, Philip; Jermutus, Lutz; Heerspink, Hiddo J L; McCrimmon, Rory J

Radiosynthesis and Preclinical Evaluation of an (18)F-Labeled Triazolopyridopyrazine-Based Inhibitor for Neuroimaging of the Phosphodiesterase 2A (PDE2A)

(18)F标记的三唑并吡啶并吡嗪类磷酸二酯酶2A(PDE2A)抑制剂的放射合成及临床前评价用于神经影像学

Wenzel, Barbara; Fritzsche, Stefan R; Toussaint, Magali; Briel, Detlef; Kopka, Klaus; Brust, Peter; Scheunemann, Matthias; Deuther-Conrad, Winnie

A Convenient Route to New (Radio)Fluorinated and (Radio)Iodinated Cyclic Tyrosine Analogs

合成新型(放射性)氟化和(放射性)碘化环状酪氨酸类似物的便捷途径

Chao, Maria Noelia; Chezal, Jean-Michel; Debiton, Eric; Canitrot, Damien; Witkowski, Tiffany; Levesque, Sophie; Degoul, Françoise; Tarrit, Sébastien; Wenzel, Barbara; Miot-Noirault, Elisabeth; Serre, Audrey; Maisonial-Besset, Aurélie

Improved in vivo PET imaging of the adenosine A(2A) receptor in the brain using [(18)F]FLUDA, a deuterated radiotracer with high metabolic stability

利用具有高代谢稳定性的氘代放射性示踪剂[(18)F]FLUDA,改进了脑内腺苷A(2A)受体的体内PET成像。

Lai, Thu Hang; Toussaint, Magali; Teodoro, Rodrigo; Dukić-Stefanović, Sladjana; Gündel, Daniel; Ludwig, Friedrich-Alexander; Wenzel, Barbara; Schröder, Susann; Sattler, Bernhard; Moldovan, Rareş-Petru; Falkenburger, Björn H; Sabri, Osama; Deuther-Conrad, Winnie; Brust, Peter

Preclinical Evaluation of [(18)F]FACH in Healthy Mice and Piglets: An (18)F-Labeled Ligand for Imaging of Monocarboxylate Transporters with PET

[(18)F]FACH 在健康小鼠和仔猪中的临床前评估:一种用于 PET 成像单羧酸转运蛋白的 (18)F 标记配体

Gündel, Daniel; Sadeghzadeh, Masoud; Deuther-Conrad, Winnie; Wenzel, Barbara; Cumming, Paul; Toussaint, Magali; Ludwig, Friedrich-Alexander; Moldovan, Rareş-Petru; Kranz, Mathias; Teodoro, Rodrigo; Sattler, Bernhard; Sabri, Osama; Brust, Peter

Challenges on Cyclic Nucleotide Phosphodiesterases Imaging with Positron Emission Tomography: Novel Radioligands and (Pre-)Clinical Insights since 2016

利用正电子发射断层扫描成像环核苷酸磷酸二酯酶面临的挑战:2016年以来的新型放射性配体和(临床前)研究进展

Schröder, Susann; Scheunemann, Matthias; Wenzel, Barbara; Brust, Peter