日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

New Dual Pan-PI3K/mTOR Inhibitor: Design, Synthesis, Cytotoxic Action, Permeation, Metabolic Stability, and In Silico Protein-Ligand Interaction

新型双重泛PI3K/mTOR抑制剂:设计、合成、细胞毒性作用、渗透性、代谢稳定性及计算机模拟蛋白-配体相互作用

Aparecida E Silva, Cristiane; Pillpe-Meza, Raysa Magali; Gouveia, Wesley Leandro; da Silva Trindade, Joana D'Arc; Barbosa, Gisele; Vieira, Amanda Marques Seixas; Tolomeu, Heber Victor; Pereira, Rayane França; Santos, Carlos Antônio do Nascimento; Freire-de-Lima, Leonardo; Lima, Lidia Moreira

Discovery of N‑Acylhydrazone Derivatives as ROCK Inhibitors: A Journey from Virtual Screening and Structure-Based De Novo Design to the Identification of ROCK2 Selective Inhibitors and Beyond

N-酰基腙衍生物作为ROCK抑制剂的发现:从虚拟筛选和基于结构的从头设计到ROCK2选择性抑制剂的鉴定及其他

Pinheiro, Pedro de Sena Murteira; Silva Franco, Lucas; Pillpe-Meza, Raysa Magali; de Jesus, Bárbara da Silva Mascarenhas; Martins, Gabrielli Ayumi Ito; Gouveia, Wesley Leandro; Rodrigues, Daniel Alencar; Alves, Marina Amaral; Lima, Lídia Moreira

Mechanistic Advances in the Therapeutic Application of Bixin for Lung Inflammation In Vitro and In Vivo.

体外和体内研究Bixin治疗肺部炎症的机制进展

Figueiredo-Junior Alexsandro Tavares, Marques Bruno Clemente Brandão, Santos Douglas Galdino Dos, Gouveia Wesley Leandro, Meza Raysa Magali Pillpe, Tinoco Luzineide Wanderley, Lima Lídia Moreira, Valenca Samuel Santos, Lanzetti Manuella

Investigation on LASSBio-1971 and LASSBio-1974 Cellular Cytotoxic Mechanism and Their Comparative DMPK Profile

LASSBio-1971 和 LASSBio-1974 细胞毒性机制及其 DMPK 特征比较研究

de Moraes Junior, Manoel Oliveira; Barbosa, Gisele; da Costa, Caroline Marques Xavier; Pillpe-Meza, Raysa Magali; de Gouveia, Wesley Leandro; do Amaral, Daniel Nascimento; Gelves, Luis Gabriel Valdivieso; Laufer, Stefan; Lima, Lídia Moreira

Cytotoxic and Antiproliferative Activity of LASSBio-2208 and the Attempts to Determine Its Drug Metabolism and Pharmacokinetics In Vitro Profile

LASSBio-2208 的细胞毒性和抗增殖活性以及确定其药物代谢和药代动力学体外概况的尝试

Raysa Magali Pillpe-Meza, Wesley Leandro Gouveia, Gisele Barbosa, Carlos A M Fraga, Eliezer J Barreiro, Lidia Moreira Lima