日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Pharmacologic Targeting of TFIIH Suppresses KRAS-Mutant Pancreatic Ductal Adenocarcinoma and Synergizes with TRAIL

TFIIH 的药物靶向作用可抑制 KRAS 突变型胰腺导管腺癌并与 TRAIL 产生协同作用

Russell Moser, James Annis, Olga Nikolova, Cliff Whatcott, Kay Gurley, Eduardo Mendez, Kim Moran-Jones, Craig Dorrell, Rosalie C Sears, Calvin Kuo, Haiyong Han, Andrew Biankin, Carla Grandori, Daniel D Von Hoff, Christopher J Kemp

TNK1 is a ubiquitin-binding and 14-3-3-regulated kinase that can be targeted to block tumor growth

TNK1是一种泛素结合且受14-3-3蛋白调控的激酶,可作为靶点阻断肿瘤生长。

Tsz-Yin Chan #,Christina M Egbert #,Julia E Maxson,Adam Siddiqui,Logan J Larsen,Kristina Kohler,Eranga Roshan Balasooriya,Katie L Pennington,Tsz-Ming Tsang,Madison Frey,Erik J Soderblom,Huimin Geng,Markus Müschen,Tetyana V Forostyan,Savannah Free,Gaelle Mercenne,Courtney J Banks,Jonard Valdoz,Clifford J Whatcott,Jason M Foulks,David J Bearss,Thomas O'Hare,David C S Huang,Kenneth A Christensen,James Moody,Steven L Warner,Jeffrey W Tyner,Joshua L Andersen

Drug Repurposing to Identify Nilotinib as a Potential SARS-CoV-2 Main Protease Inhibitor: Insights from a Computational and In Vitro Study

药物再利用:尼洛替尼作为潜在的SARS-CoV-2主蛋白酶抑制剂的发现:一项计算和体外研究的启示

Banerjee, Souvik; Yadav, Shalini; Banerjee, Sourav; Fakayode, Sayo O; Parvathareddy, Jyothi; Reichard, Walter; Surendranathan, Surekha; Mahmud, Foyez; Whatcott, Ryan; Thammathong, Joshua; Meibohm, Bernd; Miller, Duane D; Jonsson, Colleen B; Dubey, Kshatresh Dutta

TP-0903 is active in models of drug-resistant acute myeloid leukemia

TP-0903 在耐药性急性髓系白血病模型中有效

Jae Yoon Jeon, Daelynn R Buelow, Dominique A Garrison, Mingshan Niu, Eric D Eisenmann, Kevin M Huang, Megan E Zavorka Thomas, Robert H Weber, Clifford J Whatcott, Steve L Warner, Shelley J Orwick, Bridget Carmichael, Emily Stahl, Lindsey T Brinton, Rosa Lapalombella, James S Blachly, Erin Hertlein, 

Parallel Accumulation of Tumor Hyaluronan, Collagen, and Other Drivers of Tumor Progression

肿瘤透明质酸、胶原蛋白和其他肿瘤进展驱动因素的平行积累

Xiaoming Li, H Michael Shepard, Jessica A Cowell, Chunmei Zhao, Ryan J Osgood, Sanna Rosengren, Barbara Blouw, Sheryl A Garrovillo, Mark D Pagel, Clifford J Whatcott, Haiyong Han, Daniel D Von Hoff, Darin M Taverna, Michael J LaBarre, Daniel C Maneval, Curtis B Thompson

Inhibition of ROCK1 kinase modulates both tumor cells and stromal fibroblasts in pancreatic cancer

抑制 ROCK1 激酶可调节胰腺癌中的肿瘤细胞和基质成纤维细胞

Clifford J Whatcott, Serina Ng, Michael T Barrett, Galen Hostetter, Daniel D Von Hoff, Haiyong Han

Combined venetoclax and alvocidib in acute myeloid leukemia

维奈克拉与阿沃昔布联合治疗急性髓系白血病

James Bogenberger, Clifford Whatcott, Nanna Hansen, Devora Delman, Chang-Xin Shi, Wontak Kim, Hillary Haws, Katherine Soh, Ye Sol Lee, Peter Peterson, Adam Siddiqui-Jain, Steven Weitman, Keith Stewart, David Bearss, Ruben Mesa, Steven Warner, Raoul Tibes

Phenotypic chemical screening using a zebrafish neural crest EMT reporter identifies retinoic acid as an inhibitor of epithelial morphogenesis

使用斑马鱼神经嵴 EMT 报告基因进行表型化学筛选,鉴定出视黄酸是上皮形态发生的抑制剂

Laura Jimenez, Jindong Wang, Monique A Morrison, Clifford Whatcott, Katherine K Soh, Steven Warner, David Bearss, Cicely A Jette, Rodney A Stewart

Adenosquamous carcinoma of the pancreas: Molecular characterization of 23 patients along with a literature review

胰腺腺鳞癌:23例患者的分子特征分析及文献综述

Borazanci, Erkut; Millis, Sherri Z; Korn, Ron; Han, Haiyong; Whatcott, Clifford J; Gatalica, Zoran; Barrett, Michael T; Cridebring, Derek; Von Hoff, Daniel D

Orchestrating the Tumor Microenvironment to Improve Survival for Patients With Pancreatic Cancer: Normalization, Not Destruction

通过调控肿瘤微环境来提高胰腺癌患者的生存率:正常化而非破坏

Whatcott, Clifford J; Han, Haiyong; Von Hoff, Daniel D