日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Dynamically chiral phosphonic acid-type metallo-β-lactamase inhibitors

动态手性膦酸型金属β-内酰胺酶抑制剂

Gulyás, Kinga Virág; Zhou, Liping; Salamonsen, Daniel; Prester, Andreas; Bartels, Kim; Bosman, Robert; Haffke, Paul; Li, Jintian; Tamási, Viola; Deufel, Fritz; Thoma, Johannes; Andersson Rasmussen, Anna; Csala, Miklós; Schroder Leiros, Hanna-Kirsti; Xu, Zhijian; Widersten, Mikael; Rohde, Holger; Schulz, Eike C; Zhu, Weiliang; Erdélyi, Máté

Structural enzymology studies with the substrate 3S-hydroxybutanoyl-CoA: bifunctional MFE1 is a less efficient dehydrogenase than monofunctional HAD

以 3S-羟基丁酰辅酶A为底物的结构酶学研究表明:双功能 MFE1 的脱氢酶效率低于单功能 HAD。

Sridhar, Shruthi; Kiema, Tiila-Riikka; Schmitz, Werner; Widersten, Mikael; Wierenga, Rik K

Structures of lactaldehyde reductase, FucO, link enzyme activity to hydrogen bond networks and conformational dynamics

乳醛还原酶 FucO 的结构将酶活性与氢键网络和构象动力学联系起来

Alberto Zavarise, Shruthi Sridhar, Tiila-Riikka Kiema, Rikkert K Wierenga, Mikael Widersten

Crystal structures and kinetic studies of a laboratory evolved aldehyde reductase explain the dramatic shift of its new substrate specificity

实验室进化的醛还原酶的晶体结构和动力学研究解释了其新底物特异性的急剧转变

Shruthi Sridhar, Alberto Zavarise, Tiila Riikka Kiema, Subhadra Dalwani, Tor Eriksson, Yannick Hajee, Thilak Reddy Enugala, Rik K Wierenga, Mikael Widersten

Structure and Mechanism of a Cold-Adapted Bacterial Lipase.

冷适应细菌脂肪酶的结构和机制

van der Ent Florian, Lund Bjarte A, Svalberg Linn, Purg Miha, Chukwu Ghislean, Widersten Mikael, Isaksen Geir V, Brandsdal Bjørn O, à qvist Johan

Facile synthesis of 2-hydroxyacetophenone from racemic styrene oxide catalyzed by engineered enzymes

利用工程酶催化外消旋苯乙烯氧化物简便合成2-羟基苯乙酮

Söderlund, Isac; Tjärnhage, Elias; Hamnevik, Emil; Widersten, Mikael

Epoxide hydrolysis as a model system for understanding flux through a branched reaction scheme

环氧化物水解作为理解支链反应通量的模型体系

Janfalk Carlsson, Åsa; Bauer, Paul; Dobritzsch, Doreen; Kamerlin, Shina C L; Widersten, Mikael

Linking coupled motions and entropic effects to the catalytic activity of 2-deoxyribose-5-phosphate aldolase (DERA)

将耦合运动和熵效应与 2-脱氧核糖-5-磷酸醛缩酶 (DERA) 的催化活性联系起来

Ma, Huan; Szeler, Klaudia; Kamerlin, Shina C L; Widersten, Mikael

Laboratory-Evolved Enzymes Provide Snapshots of the Development of Enantioconvergence in Enzyme-Catalyzed Epoxide Hydrolysis

实验室进化酶提供了酶催化环氧化物水解中对映体趋同发展过程的快照

Janfalk Carlsson, Åsa; Bauer, Paul; Dobritzsch, Doreen; Nilsson, Mikael; Kamerlin, S C Lynn; Widersten, Mikael

Expanding the Catalytic Triad in Epoxide Hydrolases and Related Enzymes

扩展环氧化物水解酶及相关酶的催化三元组

Amrein, Beat A; Bauer, Paul; Duarte, Fernanda; Janfalk Carlsson, Åsa; Naworyta, Agata; Mowbray, Sherry L; Widersten, Mikael; Kamerlin, Shina C L