日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Benzoic Acid Derivatives Improve Plasma Stability of Diester Butyrophilin Ligand Prodrugs

苯甲酸衍生物可提高二酯丁酰辅酶A配体前药的血浆稳定性

Kintigh, Parker A; Singh, Umed; Pawge, Girija; Bashir, Sidra; Hsiao, Chia-Hung Christine; Wiemer, Andrew J; Wiemer, David F

Impact of fixed phosphorus position on activity of triazole bisphosphonates as geranylgeranyl diphosphate synthase inhibitors

固定磷位置对三唑双膦酸盐作为香叶基香叶基二磷酸合酶抑制剂活性的影响

Ayub Ali, Md; Maalouf, Mona A; Feng, Dan; Rashid, Mamunur; Gehrke, Nathaniel R; Chhonker, Yashpal S; Murry, Daryl J; Wiemer, David F; Holstein, Sarah A

Cost‐Effective DNA Storage System with DNA Movable Type (Adv. Sci. 9/2025)

采用可移动DNA的低成本DNA存储系统(Adv. Sci. 9/2025)

Wiemer, Andrew J; Wiemer, David F; Wang, Chenyang; Wei, Di; Wei, Zheng; Yang, Dongxin; Xing, Jing; Wang, Yunze; Wang, Xiaotong; Wang, Pei; Ma, Guannan; Zhang, Xinru; Li, Haolan; Tang, Chuan; Hou, Pengfei; Wang, Jie; Gao, Renjun; Xie, Guiqiu; Li, Cuidan; Ju, Yingjiao; Wang, Peihan; Yue, Liya; Zhao, Yongliang; Sheng, Yongjie; Xiao, Jingfa; Niu, Haitao; Xu, Sihong; Yang, Huaiyi; Liu, Di; Duan, Bo; Bu, Dongbo; Tan, Guangming; Chen, Fei

Enhanced Plasma Stability and Potency of Aryl/Acyloxy Prodrugs of a BTN3A1 Ligand

BTN3A1配体的芳基/酰氧基前药的血浆稳定性和效力增强

Singh, Umed; Pawge, Girija; Rani, Sarita; Hsiao, Chia-Hung Christine; Wiemer, David F; Wiemer, Andrew J

α-Amino bisphosphonate triazoles serve as GGDPS inhibitors

α-氨基双膦酸酯三唑类化合物可作为GGDPS抑制剂。

Gehrke, Nathaniel R; Feng, Dan; Ayub Ali, Md; Maalouf, Mona A; Holstein, Sarah A; Wiemer, David F

Diester Prodrugs of a Phosphonate Butyrophilin Ligand Display Improved Cell Potency, Plasma Stability, and Payload Internalization

膦酸酯丁酰辅酶A配体的二酯前药表现出更高的细胞效力、血浆稳定性和有效载荷内化能力。

Singh, Umed; Pawge, Girija; Rani, Sarita; Hsiao, Chia-Hung Christine; Wiemer, Andrew J; Wiemer, David F

Efficiency of bis-amidate phosphonate prodrugs

双酰胺膦酸酯前药的效率

Lentini, Nicholas A; Huang, Xueting; Schladetsch, Megan A; Hsiao, Chia-Hung Christine; Wiemer, David F; Wiemer, Andrew J

Substitution of a triazole for the central olefin in biologically active stilbenes

生物活性芪类化合物中中心烯烃被三唑取代

Stockdale, David P; Beutler, John A; Wiemer, David F

Conjugate reduction of vinyl bisphosphonates

乙烯基双膦酸酯的共轭还原

Harmon, Nyema M; Gehrke, Nathaniel R; Wiemer, David F

Incorporation of a FRET pair within a phosphonate diester

将FRET对引入膦酸酯二酯中

Harmon, Nyema M; Huang, Xueting; Hsiao, Chia-Hung Christine; Wiemer, Andrew J; Wiemer, David F