日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Hypothesis-Driven, Structure-Based Design in Photopharmacology: The Case of eDHFR Inhibitors

光药理学中的假设驱动、基于结构的设计:以 eDHFR 抑制剂为例

Piermichele Kobauri, Nicole S Galenkamp, Albert M Schulte, Jisk de Vries, Nadja A Simeth, Giovanni Maglia, Sebastian Thallmair, Dušan Kolarski, Wiktor Szymanski, Ben L Feringa

Patient-derived parathyroid organoids as a tracer and drug-screening application model

患者来源的甲状旁腺类器官作为示踪剂和药物筛选应用模型

Milou E Noltes, Luc H J Sondorp, Laura Kracht, Inês F Antunes, René Wardenaar, Wendy Kelder, Annelies Kemper, Wiktor Szymanski, Wouter T Zandee, Liesbeth Jansen, Adrienne H Brouwers, Robert P Coppes, Schelto Kruijff

Light-Control over Casein Kinase 1δ Activity with Photopharmacology: A Clear Case for Arylazopyrazole-Based Inhibitors

利用光药理学对酪蛋白激酶 1δ 活性进行光控制:芳基偶氮吡唑类抑制剂的明确案例

Albert M Schulte, Dušan Kolarski, Vidya Sundaram, Ashutosh Srivastava, Florence Tama, Ben L Feringa, Wiktor Szymanski

Reversible modulation of circadian time with chronophotopharmacology

利用时间光药理学对昼夜节律进行可逆调节

Dušan Kolarski, Carla Miró-Vinyals #, Akiko Sugiyama #, Ashutosh Srivastava, Daisuke Ono, Yoshiko Nagai, Mui Iida, Kenichiro Itami, Florence Tama, Wiktor Szymanski, Tsuyoshi Hirota, Ben L Feringa

Mechanism of Resistance Development in E. coli against TCAT, a Trimethoprim-Based Photoswitchable Antibiotic

大肠杆菌对基于甲氧苄啶的光开关抗生素 TCAT 产生耐药性的机制

Anna I Lauxen, Piermichele Kobauri, Michael Wegener, Mickel J Hansen, Nicole S Galenkamp, Giovanni Maglia, Wiktor Szymanski, Ben L Feringa, Oscar P Kuipers

HDAC1 and HDAC3 underlie dynamic H3K9 acetylation during embryonic neurogenesis and in schizophrenia-like animals

HDAC1 和 HDAC3 是胚胎神经发生过程中和精神分裂症样动物中动态 H3K9 乙酰化的基础

Josef Večeřa, Eva Bártová, Jana Krejčí, Soňa Legartová, Denisa Komůrková, Jana Rudá-Kučerová, Tibor Štark, Eva Dražanová, Tomáš Kašpárek, Alexandra Šulcová, Frank J Dekker, Wiktor Szymanski, Christian Seiser, Georg Weitzer, Raphael Mechoulam, Vincenzo Micale, Stanislav Kozubek

Characterization of a thermostable methylaspartate ammonia lyase from Carboxydothermus hydrogenoformans

氢化碳嗜热菌热稳定性甲基天冬氨酸氨裂解酶的表征

Hans Raj, Vinod Puthan Veetil, Wiktor Szymanski, Frank J Dekker, Wim J Quax, Ben L Feringa, Dick B Janssen, Gerrit J Poelarends