日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A phase 1 study of the CDK9 inhibitor voruciclib in relapsed/refractory acute myeloid leukemia and B-cell malignancies

CDK9抑制剂voruciclib治疗复发/难治性急性髓系白血病和B细胞恶性肿瘤的I期研究

Davids, Matthew S; Brander, Danielle M; Alvarado-Valero, Yesid; Diefenbach, Catherine S; Egan, Daniel N; Dinner, Shira N; Javidi-Sharifi, Nathalie; Al Malki, Monzr M; Begna, Kebede H; Bhatt, Vijaya Raj; Abedin, Sameem; Cook, Rachel J; Collins, Mary C; Roleder, Carly; Dominguez, Edward C; Rajagopalan, Prabhu; Wiley, Sandra E; Ghalie, Richard G; Danilov, Alexey V

A Phase 1b study of the OxPhos inhibitor ME-344 with bevacizumab in refractory metastatic colorectal cancer

一项针对难治性转移性结直肠癌的氧化磷酸化抑制剂ME-344联合贝伐单抗的1b期研究

Boland, Patrick M; Lenz, Heinz-Josef; Ciombor, Kristen K; Florou, Vaia; Pishvaian, Michael J; Cusnir, Michael; Cohen, Deirdre; Guo, Jessie Y; Tang, Min; Rajagopalan, Prabhu; Wiley, Sandra E; Ghalie, Richard G; Hochster, Howard S

The oral CDK9 inhibitor voruciclib combined with venetoclax for patients with relapsed/refractory acute myeloid leukemia

口服 CDK9 抑制剂 voruciclib 与 venetoclax 联合用于治疗复发/难治性急性髓系白血病患者

Alvarado-Valero, Yesid; Cook, Rachel J; Dinner, Shira N; Keng, Michael; Begna, Kebede H; Javidi-Sharifi, Nathalie; Abedin, Sameem; Al Malki, Monzr M; Bhatt, Vijaya Raj; Rajagopalan, Prabhu; Tang, Min; Wiley, Sandra E; Ghalie, Richard G; Davids, Matthew S

Enhancing anti-AML activity of venetoclax by isoflavone ME-344 through suppression of OXPHOS and/or purine biosynthesis in vitro

异黄酮ME-344通过抑制体外氧化磷酸化和/或嘌呤生物合成增强维奈托克的抗急性髓系白血病活性

Hurrish, Katie H; Su, Yongwei; Patel, Shraddha; Ramage, Cassandra L; Zhao, Jianlei; Temby, Brianna R; Carter, Jenna L; Edwards, Holly; Buck, Steven A; Wiley, Sandra E; Hüttemann, Maik; Polin, Lisa; Kushner, Juiwanna; Dzinic, Sijana H; White, Kathryn; Bao, Xun; Li, Jing; Yang, Jay; Boerner, Julie; Hou, Zhanjun; Al-Atrash, Gheath; Konoplev, Sergej N; Busquets, Jonathan; Tiziani, Stefano; Matherly, Larry H; Taub, Jeffrey W; Konopleva, Marina; Ge, Yubin; Baran, Natalia

Reversible phosphorylation of Rpn1 regulates 26S proteasome assembly and function

Rpn1的可逆磷酸化调控26S蛋白酶体的组装和功能

Liu, Xiaoyan; Xiao, Weidi; Zhang, Yanan; Wiley, Sandra E; Zuo, Tao; Zheng, Yingying; Chen, Natalie; Chen, Lu; Wang, Xiaorong; Zheng, Yawen; Huang, Lan; Lin, Shixian; Murphy, Anne N; Dixon, Jack E; Xu, Ping; Guo, Xing

Inhibition of dual-specificity tyrosine phosphorylation-regulated kinase 2 perturbs 26S proteasome-addicted neoplastic progression

双特异性酪氨酸磷酸化调节激酶2的抑制会扰乱26S蛋白酶体依赖的肿瘤进展。

Banerjee, Sourav; Wei, Tiantian; Wang, Jue; Lee, Jenna J; Gutierrez, Haydee L; Chapman, Owen; Wiley, Sandra E; Mayfield, Joshua E; Tandon, Vasudha; Juarez, Edwin F; Chavez, Lukas; Liang, Ruqi; Sah, Robert L; Costello, Caitlin; Mesirov, Jill P; de la Vega, Laureano; Cooper, Kimberly L; Dixon, Jack E; Xiao, Junyu; Lei, Xiaoguang

Enzymatic Phosphorylation of Ser in a Type I Collagen Peptide

I型胶原蛋白肽中丝氨酸的酶促磷酸化

Qiu, Yimin; Poppleton, Erik; Mekkat, Arya; Yu, Hongtao; Banerjee, Sourav; Wiley, Sandra E; Dixon, Jack E; Kaplan, David L; Lin, Yu-Shan; Brodsky, Barbara

A Single Kinase Generates the Majority of the Secreted Phosphoproteome

单个激酶生成大部分分泌型磷酸化蛋白质组

Tagliabracci, Vincent S; Wiley, Sandra E; Guo, Xiao; Kinch, Lisa N; Durrant, Eric; Wen, Jianzhong; Xiao, Junyu; Cui, Jixin; Nguyen, Kim B; Engel, James L; Coon, Joshua J; Grishin, Nick; Pinna, Lorenzo A; Pagliarini, David J; Dixon, Jack E

Thiazolidinediones are acute, specific inhibitors of the mitochondrial pyruvate carrier

噻唑烷二酮类药物是线粒体丙酮酸载体的急性特异性抑制剂。

Divakaruni, Ajit S; Wiley, Sandra E; Rogers, George W; Andreyev, Alexander Y; Petrosyan, Susanna; Loviscach, Mattias; Wall, Estelle A; Yadava, Nagendra; Heuck, Alejandro P; Ferrick, David A; Henry, Robert R; McDonald, William G; Colca, Jerry R; Simon, Melvin I; Ciaraldi, Theodore P; Murphy, Anne N

Wolfram Syndrome protein, Miner1, regulates sulphydryl redox status, the unfolded protein response, and Ca2+ homeostasis.

Wolfram 综合征蛋白 Miner1 调节巯基氧化还原状态、未折叠蛋白反应和 Ca2+ 稳态

Wiley Sandra E, Andreyev Alexander Y, Divakaruni Ajit S, Karisch Robert, Perkins Guy, Wall Estelle A, van der Geer Peter, Chen Yi-Fan, Tsai Ting-Fen, Simon Melvin I, Neel Benjamin G, Dixon Jack E, Murphy Anne N