日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification of DC-174 as a Novel Hydroxamic Precandidate for the Development of an Oral Snakebite Treatment

鉴定出DC-174是一种新型羟肟酸类候选药物,可用于开发口服蛇咬伤治疗药物。

Chong, Daniel J W; Albulescu, Laura-Oana; Westhorpe, Adam; Clare, Rachel H; Marriott, Amy E; Woodley, Christopher M; Gunasekar, Ramachandran; Mosallam, Nada; Crittenden, Edouard; Stars, Emma; Dawson, Charlotte; Kool, Jeroen; Wilkinson, Mark C; Leung, Suet C; Berry, Neil G; Casewell, Nicholas R; O'Neill, Paul M

Biochemical characterisation and substrate-specific proteolytic diversity of venom metalloproteinases in African puff adders

非洲鼓腹蝰蛇毒液金属蛋白酶的生化特性及底物特异性蛋白水解多样性

Wilkinson, Mark C; Modahl, Cassandra M; Waterhouse, David T K; Saviola, Anthony; Albulescu, Laura-Oana; Tianyi, Frank-Leonel; Kazandjian, Taline D; Wüster, Wolfgang; Theart, Francois; Oluoch, George O; Harrison, Robert A; Casewell, Nicholas R

Quantifying venom in African snakes: Insights into protein content, yield and body size associations

量化非洲蛇毒:蛋白质含量、产量和体型关联性研究

French, Stephanie; Da Silva, Rachael; Have, Martijn Ten; Crittenden, Edouard; Rowley, Paul; Cullen, India C; Holland, Zachary; Wilkinson, Mark C; Modahl, Cassandra M

Snake Venom Metalloproteinases from Puff Adder and Saw-Scaled Viper Venoms Cause Cytotoxic Effects in Human Keratinocytes.

来自鼓腹蝰蛇和锯鳞蝰蛇毒液的蛇毒金属蛋白酶对人类角质形成细胞具有细胞毒性作用

Bartlett Keirah E, Westhorpe Adam, Wilkinson Mark C, Casewell Nicholas R

Preclinical evaluation of the neutralising efficacy of three antivenoms against the venoms of the recently taxonomically partitioned E. ocellatus and E. romani.

对三种抗蛇毒血清中和最近分类学上划分的眼斑蝾螈和罗马蝾螈毒液的功效进行临床前评估

Edge Rebecca J, Marriott Amy E, Keen Molly, Xie Tiffany, Crittenden Edouard P, Dawson Charlotte A, Wilkinson Mark C, Wüster Wolfgang, Casewell Nicholas R, Ainsworth Stuart, Menzies Stefanie K

Dermonecrosis caused by a spitting cobra snakebite results from toxin potentiation and is prevented by the repurposed drug varespladib

喷毒眼镜蛇咬伤引起的皮肤坏死是由于毒素增强所致,而重新利用的药物瓦雷斯普拉地(varespladib)可以预防这种坏死。

Bartlett, Keirah E; Hall, Steven R; Rasmussen, Sean A; Crittenden, Edouard; Dawson, Charlotte A; Albulescu, Laura-Oana; Laprade, William; Harrison, Robert A; Saviola, Anthony J; Modahl, Cassandra M; Jenkins, Timothy P; Wilkinson, Mark C; Gutiérrez, José María; Casewell, Nicholas R

African polyvalent antivenom can maintain pharmacological stability and ability to neutralise murine venom lethality for decades post-expiry: evidence for increasing antivenom shelf life to aid in alleviating chronic shortages

非洲多价抗蛇毒血清在过期后数十年仍能保持药理稳定性并中和鼠毒的致死性:证据表明,延长抗蛇毒血清的保质期有助于缓解长期短缺问题。

Solano, Gabriela; Cunningham, Sinead; Edge, Rebecca J; Duran, Gina; Sanchez, Adriana; Villalta, Mauren; Clare, Rachel H; Wilkinson, Mark C; Marriott, Amy E; Abada, Camille; Menzies, Stefanie K; Keen, Molly; Lalloo, David G; Stienstra, Ymkje; Abouyannis, Michael; Casewell, Nicholas R; León, Guillermo; Ainsworth, Stuart

Plug and play virus-like particles for the generation of anti-toxin antibodies

用于生成抗毒素抗体的即插即用型病毒样颗粒

Edge, Rebecca J; Marriott, Amy E; Stars, Emma L; Patel, Rohit N; Wilkinson, Mark C; King, Lloyd D W; Slagboom, Julien; Tan, Choo Hock; Ratanabanangkoon, Kavi; Draper, Simon J; Ainsworth, Stuart

Investigating Viral Inoculation and Recovery from Medical Masks

调查医用口罩上的病毒接种和恢复情况

Wilkinson, Mark C; Carney, Jennifer

Preclinical validation of a repurposed metal chelator as an early-intervention therapeutic for hemotoxic snakebite

对一种重新利用的金属螯合剂作为早期干预治疗血液毒性蛇咬伤的临床前验证

Albulescu, Laura-Oana; Hale, Melissa S; Ainsworth, Stuart; Alsolaiss, Jaffer; Crittenden, Edouard; Calvete, Juan J; Evans, Chloe; Wilkinson, Mark C; Harrison, Robert A; Kool, Jeroen; Casewell, Nicholas R