日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification of spirodioxolane nsP2 helicase inhibitors with antialphaviral activity

鉴定具有抗甲病毒活性的螺二氧戊环nsP2解旋酶抑制剂

Oh, Hans J; Sears, John D; Ramalingam, Bose Muthu; Saleem, Rahman Shah Zaib; Davis-Gilbert, Zachary W; Hossain, Mohammed Anwar; Moorman, Stella R; Ohja, Durbadal; Martinez, Sabian A; Burdick, Jane E; Couñago, Rafael M; Moorman, Nathaniel J; Heise, Mark T; Todd, Matthew H; Willson, Timothy M

Structure-guided optimization of small molecules targeting Yck2 as a strategy to combat Candida albicans

以Yck2为靶点的小分子结构导向优化作为对抗白色念珠菌的策略

Puumala, Emily; Nandakumar, Meganathan; Yiu, Bonnie; Stogios, Peter J; Strickland, Benjamin G; Zarnowski, Robert; Wang, Xiaoyu; Williams, Noelle S; Savchenko, Alexei; Andes, David R; Robbins, Nicole; Whitesell, Luke; Willson, Timothy M; Cowen, Leah E

Identification of Direct-Acting nsP2 Helicase Inhibitors with Antialphaviral Activity

鉴定具有抗甲病毒活性的直接作用nsP2解旋酶抑制剂

Muthu Ramalingam, Bose; Sears, John D; Talbot, Kacey M; Su, Yuan-Wei Norman; Houliston, Scott; Hossain, Mohammed Anwar; Davis-Gilbert, Zachary W; Zhao, Chunqing; Oh, Hans J; Brown, Peter J; Sanders, Marcia K; Moorman, Stella R; Ojha, Durbadal; Burdick, Jane E; Law, Isabella; Morales, Noah L; Martinez, Sabian A; Loppnau, Peter; Garcia Perez, Julia; Drobish, Adam M; Morrison, Thomas E; Streblow, Zachary J; Streblow, Daniel N; Arrowsmith, Cheryl H; Vargason, Ava; Couñago, Rafael M; Halabelian, Levon; Arnold, Jamie J; Cameron, Craig E; Moorman, Nathaniel J; Heise, Mark T; Willson, Timothy M

N-Alkyl Sulfamates as a New Class of nsP2 Cysteine Protease Inhibitors with Broad-Spectrum Antialphaviral Activity

N-烷基氨基磺酸酯作为一类新型nsP2半胱氨酸蛋白酶抑制剂,具有广谱抗甲病毒活性

Ghoshal, Anirban; Sears, John D; Hossain, Mohammad Anwar; Tse, Edwin G; Howell, Stefanie; Burdick, Jane E; Morales, Noah L; Martinez, Sabian A; Law, Isabella; Streblow, Zachary J; Streblow, Daniel N; Couñago, Rafael M; Moorman, Nathaniel J; Heise, Mark T; Willson, Timothy M

Structural Chemistry of Helicase Inhibition

解旋酶抑制的结构化学

Selvaratnam, Lakshi; Willson, Timothy M; Schapira, Matthieu

Chemoproteomic Profiling of C. albicans for Characterization of Antifungal Kinase Inhibitors.

念珠菌化学蛋白质组学分析用于鉴定抗真菌激酶抑制剂

Shirley David J, Nandakumar Meganathan, Cabrera Aurora, Yiu Bonnie, Puumala Emily, Liu Zhongle, Robbins Nicole, Whitesell Luke, Smith Jeffrey L, Lyons Scott, Mordant Angie L, Herring Laura E, Graves Lee M, Couñago Rafael M, Drewry David H, Cowen Leah E, Willson Timothy M

Species-Dependent Metabolism of a Covalent nsP2 Protease Inhibitor with In Vivo Antialphaviral Activity.

具有体内抗甲病毒活性的共价nsP2蛋白酶抑制剂的物种依赖性代谢

Hossain Mohammad Anwar, Mayo Abigail K, Ghoshal Anirban, Taft-Benz Sharon, Anderson Elizabeth, Morales Noah L, Pressey Katia D, Vargason Ava, Brouwer Kim L R, Moorman Nathaniel J, Heise Mark T, Willson Timothy M

Chemical arsenal for helicase Hunters: Striking the toughest targets in antiviral research

用于解旋酶猎杀的化学武器库:打击抗病毒研究中最棘手的目标

Martin, Holli-Joi; Hossain, Mohammad Anwar; Wellnitz, James; Kelestemur, Enes; Hochuli, Joshua E; Perveen, Sumera; Arrowsmith, Cheryl; Willson, Timothy M; Muratov, Eugene N; Tropsha, Alexander

Enantioselective Chemical Probe for Chikungunya nsP2 Helicase with Antialphaviral Activity

具有抗甲病毒活性的基孔肯雅病毒nsP2解旋酶对映选择性化学探针

Muthu Ramalingam, Bose; Oh, Hans J; Sears, John D; Chen, Chun-Hsing; Vala, Anand; Liu, Shubin; Talbot, Kacey M; Hossain, Mohammed Anwar; Brown, Peter J; Houliston, Scott; Garcia Perez, Julia; Li, Fengling; Amare, Meareg G; Halfmann, Peter; Smith, Jessica L; Hirsch, Alec J; Arrowsmith, Cheryl H; Halabelian, Levon; Vargason, Ava; Couñago, Rafael M; Arnold, Jamie J; Cameron, Craig E; Moorman, Nathaniel J; Heise, Mark T; Willson, Timothy M

Toward target 2035: EUbOPEN - a public-private partnership to enable & unlock biology in the open

迈向2035年目标:EUbOPEN——一项旨在促进和开放生物学的公私合作项目

Tredup, Claudia; Ackloo, Suzanne; Beck, Hartmut; Brown, Peter J; Bullock, Alex N; Ciulli, Alessio; Dikic, Ivan; Edfeldt, Kristina; Edwards, Aled M; Elkins, Jonathan M; Farin, Henner F; Fon, Edward A; Gstaiger, Matthias; Günther, Judith; Gustavsson, Anna-Lena; Häberle, Sandra; Isigkeit, Laura; Huber, Kilian V M; Kotschy, Andras; Krämer, Oliver; Leach, Andrew R; Marsden, Brian D; Matsui, Hisanori; Merk, Daniel; Montel, Florian; Mulder, Monique P C; Müller, Susanne; Owen, Dafydd R; Proschak, Ewgenij; Röhm, Sandra; Stolz, Alexandra; Sundström, Michael; von Delft, Frank; Willson, Timothy M; Arrowsmith, Cheryl H; Knapp, Stefan