日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Harnessing oligonucleotide architecture for potent multivalent inhibition of human carbonic anhydrases

利用寡核苷酸结构实现对人类碳酸酐酶的强效多价抑制

Abbass, Eslam M; Ladu, Federico; Mansot, Justine; Noël, Mathieu; Nocentini, Alessio; Sechi, Mario; Supuran, Claudiu T; Smietana, Michael; Winum, Jean-Yves

Benzoxaboroles Are Inhibitors of the η-Class Carbonic Anhydrase From Plasmodium falciparum

苯并硼氧杂环己烷是恶性疟原虫η类碳酸酐酶的抑制剂

Bonardi, Alessandro; Wein, Sharon; Mustafa, Muhamad; Cerdan, Rachel; de Luca, Viviana; Capasso, Clemente; Gratteri, Paola; Supuran, Claudiu T; Nocentini, Alessio; Winum, Jean-Yves

RETRACTED: Sarnella et al. A Novel Inhibitor of Carbonic Anhydrases Prevents Hypoxia-Induced TNBC Cell Plasticity. Int. J. Mol. Sci. 2020, 21, 8405

撤稿:Sarnella 等人,《一种新型碳酸酐酶抑制剂可阻止缺氧诱导的三阴性乳腺癌细胞可塑性》,《国际分子科学杂志》,2020 年,21 卷,8405 页。

Sarnella, Annachiara; D'Avino, Giuliana; Hill, Billy Samuel; Alterio, Vincenzo; Winum, Jean-Yves; Supuran, Claudiu T; De Simone, Giuseppina; Zannetti, Antonella

Targeting Tumor-Associated Carbonic Anhydrases in Photothermal Therapy

靶向肿瘤相关碳酸酐酶的光热疗法

Clément, Sébastien; Richeter, Sébastien; Winum, Jean-Yves

Impact of Neuroeffector Adrenergic Receptor Polymorphisms on Incident Ventricular Fibrillation During Acute Myocardial Ischemia

神经效应肾上腺素能受体多态性对急性心肌缺血期间发生室颤的影响

Chevalier, Philippe; Roy, Pascal; Bessière, Francis; Morel, Elodie; Ankou, Bénédicte; Morgan, Gina; Halder, Indrani; London, Barry; Minobe, Wayne A; Slavov, Dobromir; Delinière, Antoine; Bochaton, Thomas; Paganelli, Franck; Lesavre, Nathalie; Boiteux, Clément; Mansourati, Jacques; Maury, Philippe; Clerici, Gaël; Winum, Pierre François; Huebler, Sophia P; Carroll, Ian A; Bristow, Michael R

GABAA receptor-mediated seizure liabilities: a mixed-methods screening approach

GABAA 受体介导的癫痫发作倾向:一种混合方法筛查方法

Konstantina Bampali, Filip Koniuszewski, Florian D Vogel, Jure Fabjan, Christos Andronis, Eftychia Lekka, Vassilis Virvillis, Thomas Seidel, Annie Delaunois, Leandro Royer, Michael G Rolf, Chiara Giuliano, Martin Traebert, Gautier Roussignol, Magali Fric-Bordat, Ludmilla Mazelin-Winum, Sharon D Brya

Reconsidering anion inhibitors in the general context of drug design studies of modulators of activity of the classical enzyme carbonic anhydrase

在经典碳酸酐酶活性调节剂的药物设计研究的总体背景下,重新审视阴离子抑制剂

Nocentini, Alessio; Angeli, Andrea; Carta, Fabrizio; Winum, Jean-Yves; Zalubovskis, Raivis; Carradori, Simone; Capasso, Clemente; Donald, William A; Supuran, Claudiu T

Response to Perspectives on the Classical Enzyme Carbonic Anhydrase and the Search for Inhibitors

对经典酶碳酸酐酶及其抑制剂研究的回应

Angeli, Andrea; Carta, Fabrizio; Nocentini, Alessio; Winum, Jean-Yves; Zalubovskis, Raivis; Onnis, Valentina; Eldehna, Wagdy M; Capasso, Clemente; Carradori, Simone; Donald, William A; Dedhar, Shoukat; Supuran, Claudiu T

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-7

药物化学的突破:新靶点和机制、新药物、新希望-7

Gütschow, Michael; Eynde, Jean Jacques Vanden; Jampilek, Josef; Kang, CongBao; Mangoni, Arduino A; Fossa, Paola; Karaman, Rafik; Trabocchi, Andrea; Scott, Peter J H; Reynisson, Jóhannes; Rapposelli, Simona; Galdiero, Stefania; Winum, Jean-Yves; Brullo, Chiara; Prokai-Tatrai, Katalin; Sharma, Arun K; Schapira, Matthieu; Azuma, Yasu-Taka; Cerchia, Laura; Spetea, Mariana; Torri, Giangiacomo; Collina, Simona; Geronikaki, Athina; García-Sosa, Alfonso T; Vasconcelos, M Helena; Sousa, Maria Emília; Kosalec, Ivan; Tuccinardi, Tiziano; Duarte, Iola F; Salvador, Jorge A R; Bertinaria, Massimo; Pellecchia, Maurizio; Amato, Jussara; Rastelli, Giulio; Gomes, Paula A C; Guedes, Rita C; Sabatier, Jean-Marc; Estévez-Braun, Ana; Pagano, Bruno; Mangani, Stefano; Ragno, Rino; Kokotos, George; Brindisi, Margherita; González, Florenci V; Borges, Fernanda; Miloso, Mariarosaria; Rautio, Jarkko; Muñoz-Torrero, Diego

A Novel Inhibitor of Carbonic Anhydrases Prevents Hypoxia-Induced TNBC Cell Plasticity

新型碳酸酐酶抑制剂可防止缺氧诱导的 TNBC 细胞可塑性

Annachiara Sarnella, Giuliana D'Avino, Billy Samuel Hill, Vincenzo Alterio, Jean-Yves Winum, Claudiu T Supuran, Giuseppina De Simone, Antonella Zannetti