Discovery of New Binders for DCAF1, an Emerging Ligase Target in the Targeted Protein Degradation Field
在靶向蛋白降解领域,发现了一种新兴的连接酶靶点——DCAF1 的新型结合剂。
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.3c00104
Vulpetti, Anna; Holzer, Philipp; Schmiedeberg, Niko; Imbach-Weese, Patricia; Pissot-Soldermann, Carole; Hollingworth, Gregory J; Radimerski, Thomas; Thoma, Claudio R; Stachyra, Therese-Marie; Wojtynek, Matthias; Maschlej, Magdalena; Chau, Suzanne; Schuffenhauer, Ansgar; Fernández, César; Schröder, Martin; Renatus, Martin