日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Genetic Encoding of Pentafluorophosphato-Phenylalanine Provides PF(5)-Proteins as Phosphoprotein Mimetics

五氟磷酸苯丙氨酸的基因编码可提供 PF(5) 蛋白作为磷蛋白模拟物

Ambros, Anna Magdalena; Qianzhu, Haocheng; Tiemann, Markus; Habel, Edan; Denzinger, Katrin; Zupan, Hana; Accorsi, Matteo; Keller, Bettina G; Wolber, Gerhard; Huber, Thomas; Rademann, Jörg

Mechanistic Insights into G Protein-Biased κ-Opioid Receptor Signaling Using Dual-Charged Naltrexamine Amides

利用双电荷纳曲胺酰胺对G蛋白偏向性κ-阿片受体信号传导的机制研究

Doering, Niklas Piet; Puls, Kristina; Diceglie, Marta; Meraner, Anja; Hentsch, Axel; Hongnak, Siriwat; Wurzer, Armin; Schmidhammer, Helmut; Spetea, Mariana; Nazare, Marc; Wolber, Gerhard

CACHE Challenge #3: Targeting the Nsp3 Macrodomain of SARS-CoV-2

CACHE挑战赛#3:靶向SARS-CoV-2的Nsp3宏结构域

Herasymenko, Oleksandra; Silva, Madhushika; Correy, Galen J; Abu-Saleh, Abd Al-Aziz A; Ackloo, Suzanne; Arrowsmith, Cheryl; Ashworth, Alan; Ban, Fuqiang; Beck, Hartmut; Bishop, Kevin P; Bohórquez, Hugo J; Bolotokova, Albina; Breznik, Marko; Chau, Irene; Chen, Yu; Cherkasov, Artem; Dehaen, Wim; Della Corte, Dennis; Denzinger, Katrin; Doering, Niklas P; Edfeldt, Kristina; Edwards, Aled; Fayne, Darren; Gentile, Francesco; Gibson, Elisa; Gokdemir, Ozan; Gunnarsson, Anders; Günther, Judith; Irwin, John J; Jensen, Jan Halborg; Harding, Rachel J; Hillisch, Alexander; Hoffer, Laurent; Hogner, Anders; Hutchinson, Ashley; Kandwal, Shubhangi; Karlova, Andrea; Koirala, Kushal; Kotelnikov, Sergei; Kozakov, Dima; Lee, Juyong; Lee, Soowon; Lessel, Uta; Liu, Sijie; Liu, Xuefeng; Loppnau, Peter; Meiler, Jens; Moretti, Rocco; Moroz, Yurii S; Muvva, Charuvaka; Oprea, Tudor I; Paige, Brooks; Pandit, Amit; Park, Keunwan; Poda, Gennady; Protopopov, Mykola V; Pütter, Vera; Ravichandran, Rahul; Rognan, Didier; Rosta, Edina; Sabnis, Yogesh; Scott, Thomas; Seitova, Almagul; Sharma, Purshotam; Sindt, François; Song, Minghu; Steinmann, Casper; Stevens, Rick; Talagayev, Valerij; Tararina, Valentyna V; Tarkhanova, Olga; Tingey, Damon; Trant, John F; Treleaven, Dakota; Tropsha, Alexander; Walters, Patrick; Wells, Jude; Westermaier, Yvonne; Wolber, Gerhard; Wortmann, Lars; Zheng, Shuangjia; Fraser, James S; Schapira, Matthieu

Hexahydroquinoline Featuring Amide Functionality: A Promising Scaffold With Calcium Channel Blocking Activity

具有酰胺官能团的六氢喹啉:一种具有钙通道阻断活性的潜在骨架

Koçak Aslan, Ebru; Lam, Kevin; Huang, Sun; Coşkun, Göknil Pelin; Karagüzel, Ayşe; Denzinger, Katrin; Birgül, Kaan; Ülgen, Mert; Nafie, Jordan W; Şahin, Onur; Armstrong, Daniel W; Zamponi, Gerald W; Wolber, Gerhard; Gündüz, Miyase Gözde

Deciphering Opioid Peptide Binding Modes at Atypical Chemokine Receptor 3

解析非典型趋化因子受体3的阿片肽结合模式

Wunsch, Friederike; Cassano, Ester; Puls, Kristina; Wolber, Gerhard; Szpakowska, Martyna; Chevigné, Andy; Bermudez, Marcel

Further Insights Into the Metabolism of LGD-4033 in Human Urine. Part 2. A New Minor Metabolite With Antagonistic Activity on the Androgen Receptor Can Indicate Recent Substance Intake

进一步研究LGD-4033在人体尿液中的代谢。第二部分:一种对雄激素受体具有拮抗活性的新型微量代谢物可指示近期物质摄入情况

Angelis, Yiannis S; Sakellariou, Panagiotis; Keiler, Annekathrin M; Thevis, Mario; Thomas, Andreas; Lam, Kevin; Wolber, Gerhard; Vonaparti, Ariadni; Voss, Sven; Petrou, Michael; Pitsinos, Emmanuel N

The Kifc3 Motor Protein Controls Centrosomal Factor Cep192 in Ontogenic Coordination of Megakaryocyte Development

Kifc3马达蛋白在巨核细胞发育的个体发育协调中调控中心体因子Cep192

Elagib, Kamaleldin E; Liu, Sijie; Burguener, Valentin; Sahu, Ranjit; Kotay, Deepika M; Watts, Ciorsdaidh; Wolber, Gerhard; Goldfarb, Adam N

Discovery of Novel Isoxazole-Based Small-Molecule Toll-Like Receptor 8 Antagonists

发现新型异噁唑类小分子 Toll 样受体 8 拮抗剂

Matziol, Troy; Talagayev, Valerij; Slokan, Tjaša; Strašek Benedik, Nika; Holze, Janine; Sova, Matej; Wolber, Gerhard; Weindl, Günther

Structure-based virtual screening identifies potent CD28 inhibitors that suppress T cell co-stimulation in cellular and mucosal models.

基于结构的虚拟筛选鉴定出有效的 CD28 抑制剂,这些抑制剂能够抑制细胞和粘膜模型中的 T 细胞共刺激。

Upadhyay Saurabh, Talagayev Valerij, Cho Sungwoo, Wolber Gerhard, Gabr Moustafa

Fingerprint-Based Machine Learning for SARS-CoV-2 and MERS-CoV M(pro) Inhibition: Highlighting the Potential of Bayesian Neural Networks

基于指纹的机器学习在SARS-CoV-2和MERS-CoV M(pro)抑制中的应用:凸显贝叶斯神经网络的潜力

Doering, Niklas Piet; Talagayev, Valerij; Liu, Sijie; Wolber, Gerhard