日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Combined targeted and epigenetic-based therapy enhances antitumor immunity by stabilizing GATA6-dependent MHCI expression in pancreatic ductal adenocarcinoma.

靶向治疗与表观遗传治疗相结合,通过稳定胰腺导管腺癌中 GATA6 依赖的 MHCI 表达来增强抗肿瘤免疫力。

Peng JuanFei, Yang JiaJin, Antonopoulou Georgia, Fang Rui, Adhikari Bikash, Vogt Markus, Wolf Elmar, Sun Chong, Du Shangce, Godfrey Laura, Gupta Aayush, Trajkovic-Arsic Marija, Teichmann Nicole, Grünwald Barbara T, Krebs Niklas, Steiger Katja, Mogler Carolin, Althoff Kristina, Wang Xin, Giglio Giovanni, Liffers Sven-Thorsten, Savvatakis Konstantinos, Braren Rickmer, Lawlor Rita T, Scarpa Aldo, Behrens Diana, Lang Karl S, Cheung Phyllis F, Siveke Jens T

Unhooking the Hook: Optimization of the Aurora A Targeting PROTAC JB170 to CCT400028, an In Vitro Degrader Chemical Probe

解开钩子:优化 Aurora A 靶向 PROTAC JB170 至 CCT400028,一种体外降解化学探针

O'Hanlon, Jack A; Gutsche, Katrin; Müller, Juliane Elisabeth; Ranjan Prusty, Nihar; Mirza, Amin; Roumeliotis, Theodoros I; Yang, Hengzhang; Stubbs, Mark; Hallett, Stephen T; Eing, Lorenz; McAndrew, Peter Craig; Choudhary, Jyoti Sharma; Le Bihan, Yann-Vaï; Caldwell, John; van Montfort, Rob L M; Workman, Paul; Wolf, Elmar; Newton, Gary K; Evans, Lindsay E

Click. Screen. Degrade. A Miniaturized D2B Workflow for Rapid PROTAC Discovery

点击。屏幕。降级。用于快速 PROTAC 发现的微型化 D2B 工作流程

Mitrović, Marko; Greco, Francesco Aleksy; García, Yiliam Cruz; Lučić, Aleksandar; Hoffmann, Lasse; Chander, Rohit; Schönfeld, Julia; Liebisch, Nick; Sivashanmugam, Saran Aswathaman; Schwalm, Martin Peter; Egner, Markus; Lewandowski, Max; Merk, Daniel; Morasch, Viktoria; Wolf, Elmar; Müller, Susanne; Hanke, Thomas; Proschak, Ewgenij; Hiesinger, Kerstin; Knapp, Stefan

Induced proximity to PML protects TDP-43 from aggregation via SUMO-ubiquitin networks

诱导的与PML的接近通过SUMO-泛素网络保护TDP-43免受聚集。

Wagner, Kristina; Keiten-Schmitz, Jan; Adhikari, Bikash; Patra, Upayan; Husnjak, Koraljka; McNicoll, François; Dormann, Dorothee; Müller-McNicoll, Michaela; Tascher, Georg; Wolf, Elmar; Müller, Stefan

Correction: USP10 drives cancer stemness and enables super-competitor signalling in colorectal cancer

更正:USP10 驱动癌症干细胞特性并促进结直肠癌中的超级竞争者信号传导

Reissland, Michaela; Hartmann, Oliver; Tauch, Saskia; Bugter, Jeroen M; Prieto-Garcia, Cristian; Schulte, Clemens; Loebbert, Sinah; Solvie, Daniel; Bitman-Lotan, Eliya; Narain, Ashwin; Jacomin, Anne-Claire; Schuelein-Voelk, Christina; Fuss, Carmina T; Pahor, Nikolett; Ade, Carsten; Buck, Viktoria; Potente, Michael; Li, Vivian; Beliu, Gerti; Wiegering, Armin; Grossmann, Tom; Eilers, Martin; Wolf, Elmar; Maric, Hans; Rosenfeldt, Mathias; Maurice, Madelon M; Dikic, Ivan; Gallant, Peter; Orian, Amir; Diefenbacher, Markus E

Workflow for E3 Ligase Ligand Validation for PROTAC Development

PROTAC 开发中 E3 连接酶配体验证的工作流程

Miletić, Nebojša; Weckesser, Janik; Mosler, Thorsten; Rathore, Rajeshwari; Hoffmann, Marina E; Gehrtz, Paul; Schlesiger, Sarah; Hartung, Ingo V; Berner, Nicola; Wilhelm, Stephanie; Müller, Juliane; Adhikari, Bikash; Němec, Václav; Sivashanmugam, Saran Aswathaman; Elson, Lewis; Holzmann, Hanna; Schwalm, Martin P; Hoffmann, Lasse; Abdul Azeez, Kamal Rayees; Müller, Susanne; Kuster, Bernhard; Wolf, Elmar; Đikić, Ivan; Knapp, Stefan

Correcting 4sU induced quantification bias in nucleotide conversion RNA-seq data

校正核苷酸转换RNA-seq数据中4sU诱导的定量偏差

Berg, Kevin; Lodha, Manivel; Delazer, Isabel; Bartosik, Karolina; Garcia, Yilliam Cruz; Hennig, Thomas; Wolf, Elmar; Dölken, Lars; Lusser, Alexandra; Prusty, Bhupesh K; Erhard, Florian

USP10 drives cancer stemness and enables super-competitor signalling in colorectal cancer

USP10 驱动癌症干细胞特性并促进结直肠癌中的超级竞争者信号传导

Reissland, Michaela; Hartmann, Oliver; Tauch, Saskia; Bugter, Jeroen M; Prieto-Garcia, Cristian; Schulte, Clemens; Loebbert, Sinah; Solvie, Daniel; Bitman-Lotan, Eliya; Narain, Ashwin; Jacomin, Anne-Claire; Schuelein-Voelk, Christina; Fuss, Carmina T; Pahor, Nikolett; Ade, Carsten; Buck, Viktoria; Potente, Michael; Li, Vivian; Beliu, Gerti; Wiegering, Armin; Grossmann, Tom; Eilers, Martin; Wolf, Elmar; Maric, Hans; Rosenfeldt, Mathias; Maurice, Madelon M; Dikic, Ivan; Gallant, Peter; Orian, Amir; Diefenbacher, Markus E

Spatial transcriptomics reveals molecular cues underlying the site specificity of the adult mouse oral mucosa and its stem cell niches

空间转录组学揭示了成年小鼠口腔黏膜及其干细胞微环境的位点特异性背后的分子线索

Seubert, Anna C; Krafft, Marion; Bopp, Sarah; Helal, Moutaz; Bhandare, Pranjali; Wolf, Elmar; Alemany, Anna; Riedel, Angela; Kretzschmar, Kai

Development of 2-Aminoadenine-Based Proteolysis-Targeting Chimeras (PROTACs) as Novel Potent Degraders of Monopolar Spindle 1 and Aurora Kinases.

开发基于 2-氨基腺嘌呤的蛋白水解靶向嵌合体(PROTACs)作为单极纺锤体 1 和 Aurora 激酶的新型高效降解剂

Sflakidou Eleni, Adhikari Bikash, Siokatas Christos, Wolf Elmar, Sarli Vasiliki