日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Correction to "From Discovery to Clinical Trial: YCT-529, an Oral NonHormonal Male Contraceptive Targeting the Retinoic Acid Receptor Alpha"

更正“从发现到临床试验:YCT-529,一种靶向视黄酸受体α的口服非激素男性避孕药”

Shi, Rui; Al Noman, Md Abdullah; Mannowetz, Nadja; Cheryala, Narsihmulu; Haque, Ehfazul; Taher, Noha; Maitra, Soma; Naqvi, Tahmina; Chung, Sanny S W; Bakshi, Akash; Hawkinson, Jon E; Wong, Henry L; Wolgemuth, Debra J; Georg, Gunda I

From Discovery to Clinical Trial: YCT-529, an Oral NonHormonal Male Contraceptive Targeting the Retinoic Acid Receptor Alpha

从发现到临床试验:YCT-529,一种靶向视黄酸受体α的口服非激素男性避孕药

Shi, Rui; Al Noman, Md Abdullah; Mannowetz, Nadja; Cheryala, Narsihmulu; Haque, Ehfazul; Maitra, Soma; Naqvi, Tahmina; Chung, Sanny S W; Bakshi, Akash; Hawkinson, Jon E; Wong, Henry L; Wolgemuth, Debra J; Georg, Gunda I

Development of the retinoic acid receptor alpha-specific antagonist YCT-529 for male contraception: A brief review

用于男性避孕的视黄酸受体α特异性拮抗剂YCT-529的研发:简要回顾

Shi, Rui; Wolgemuth, Debra J; Georg, Gunda I

Targeting the retinoid signaling pathway with YCT-529 for effective and reversible oral contraception in mice and primates

利用YCT-529靶向类视黄醇信号通路,在小鼠和灵长类动物中实现有效且可逆的口服避孕

Mannowetz, Nadja; Chung, Sanny S W; Maitra, Soma; Noman, Md Abdullah Al; Wong, Henry L; Cheryala, Narsihmulu; Bakshi, Akash; Wolgemuth, Debra J; Georg, Gunda I

Strategies for developing retinoic acid receptor alpha-selective antagonists as novel agents for male contraception

开发视黄酸受体α选择性拮抗剂作为新型男性避孕药的策略

Al Noman, Md Abdullah; Cuellar, Rebecca A D; Kyzer, Jillian L; Chung, Sanny S W; Cheryala, Narsihmulu; Holth, Trinh A D; Maitra, Soma; Naqvi, Tahmina; Wong, Henry L; Schönbrunn, Ernst; Hawkinson, Jon E; Wolgemuth, Debra J; Georg, Gunda I

Genome-wide chromatin occupancy of BRDT and gene expression analysis suggest transcriptional partners and specific epigenetic landscapes that regulate gene expression during spermatogenesis.

BRDT 的全基因组染色质占据情况和基因表达分析表明,转录伙伴和特定的表观遗传景观在精子发生过程中调控基因表达

Her Yoon Ra, Wang Li, Chepelev Iouri, Manterola Marcia, Berkovits Binyamin, Cui Kairong, Zhao Keji, Wolgemuth Debra J

Retinoic acid receptor antagonists for male contraception: current status†

维甲酸受体拮抗剂在男性避孕中的应用:现状†

Noman, Md Abdullah Al; Kyzer, Jillian L; Chung, Sanny S W; Wolgemuth, Debra J; Georg, Gunda I

Pleiotrophin antagonizes Brd2 during neuronal differentiation

多效蛋白在神经元分化过程中拮抗Brd2。

Garcia-Gutierrez, Pablo; Juarez-Vicente, Francisco; Wolgemuth, Debra J; Garcia-Dominguez, Mario

The role of the double bromodomain-containing BET genes during mammalian spermatogenesis

双溴结构域BET基因在哺乳动物精子发生过程中的作用

Berkovits, Binyamin D; Wolgemuth, Debra J

Bromodomain-dependent stage-specific male genome programming by Brdt

Brdt 介导的依赖于溴结构域的阶段特异性雄性基因组编程

Gaucher, Jonathan; Boussouar, Fayçal; Montellier, Emilie; Curtet, Sandrine; Buchou, Thierry; Bertrand, Sarah; Hery, Patrick; Jounier, Sylvie; Depaux, Arnaud; Vitte, Anne-Laure; Guardiola, Philippe; Pernet, Karin; Debernardi, Alexandra; Lopez, Fabrice; Holota, Hélène; Imbert, Jean; Wolgemuth, Debra J; Gérard, Matthieu; Rousseaux, Sophie; Khochbin, Saadi