日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Ribosomal frameshifting selectively modulates the assembly, function, and pharmacological rescue of a misfolded CFTR variant.

核糖体移码选择性地调节错误折叠的 CFTR 变体的组装、功能和药理学拯救

Carmody Patrick J, Roushar Francis J, Tedman Austin, Wang Wei, Herwig Madeline, Kim Minsoo, McDonald Eli F, Noguera Karen, Wong-Roushar Jennifer, Poirier Jon-Luc, Zelt Nathan B, Pockrass Ben T, McKee Andrew G, Kuntz Charles P, Raju S Vamsee, Plate Lars, Penn Wesley D, Schlebach Jonathan P

Mitochondrial and Cytosolic One-Carbon Metabolism Is a Targetable Metabolic Vulnerability in Cisplatin-Resistant Ovarian Cancer

线粒体和细胞浆一碳代谢是顺铂耐药卵巢癌中可靶向的代谢弱点

Adrianne Wallace-Povirk, Carrie O'Connor, Aamod S Dekhne, Xun Bao, Md Junayed Nayeen, Mathew Schneider, Jade M Katinas, Jennifer Wong-Roushar, Seongho Kim, Lisa Polin, Jing Li, Jessica B Back, Charles E Dann 3rd, Aleem Gangjee, Zhanjun Hou, Larry H Matherly

Ribosomal Frameshifting Selectively Modulates the Assembly, Function, and Pharmacological Rescue of a Misfolded CFTR Variant

核糖体移码选择性地调节错误折叠的 CFTR 变体的组装、功能和药理学拯救

Patrick Carmody, Francis J Roushar, Austin Tedman, Wei Wang, Madeline Herwig, Minsoo Kim, Eli F McDonald, Karen Noguera, Jennifer Wong-Roushar, Jon-Luc Poirier, Nathan B Zelt, Ben T Pockrass, Andrew G McKee, Charles P Kuntz, S Vamsee Raju, Lars Plate, Wesley D Penn, Jonathan P Schlebach

Multitargeted 6-Substituted Thieno[2,3-d]pyrimidines as Folate Receptor-Selective Anticancer Agents that Inhibit Cytosolic and Mitochondrial One-Carbon Metabolism

多靶点6-取代噻吩并[2,3-d]嘧啶类化合物作为叶酸受体选择性抗癌剂,可抑制胞质和线粒体一碳代谢

Tong, Nian; Wong-Roushar, Jennifer; Wallace-Povirk, Adrianne; Shah, Yesha; Nyman, Morgan C; Katinas, Jade M; Schneider, Mathew; O'Connor, Carrie; Bao, Xun; Kim, Seongho; Li, Jing; Hou, Zhanjun; Matherly, Larry H; Dann, Charles E 3rd; Gangjee, Aleem

Novel Pyrrolo[3,2- d]pyrimidine Compounds Target Mitochondrial and Cytosolic One-carbon Metabolism with Broad-spectrum Antitumor Efficacy

新型吡咯并[3,2-d]嘧啶化合物靶向线粒体和细胞浆一碳代谢,具有广谱抗肿瘤功效

Aamod S Dekhne, Khushbu Shah, Gregory S Ducker, Jade M Katinas, Jennifer Wong-Roushar, Md Junayed Nayeen, Arpit Doshi, Changwen Ning, Xun Bao, Josephine Frühauf, Jenney Liu, Adrianne Wallace-Povirk, Carrie O'Connor, Sijana H Dzinic, Kathryn White, Juiwanna Kushner, Seongho Kim, Maik Hüttemann, Lisa