日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-activity relationships of cyanoquinolines with corrector-potentiator activity in ΔF508 cystic fibrosis transmembrane conductance regulator protein

氰基喹啉类化合物与ΔF508囊性纤维化跨膜传导调节蛋白的校正-增强活性之间的构效关系

Knapp, John M; Wood, Alex B; Phuan, Puay-Wah; Lodewyk, Michael W; Tantillo, Dean J; Verkman, A S; Kurth, Mark J

Cyanoquinolines with independent corrector and potentiator activities restore ΔPhe508-cystic fibrosis transmembrane conductance regulator chloride channel function in cystic fibrosis.

具有独立校正和增强活性的氰基喹啉可恢复囊性纤维化中 ΔPhe508-囊性纤维化跨膜电导调节剂氯离子通道的功能

Phuan Puay-Wah, Yang Baoxue, Knapp John M, Wood Alex B, Lukacs Gergely L, Kurth Mark J, Verkman A S