日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

R-loop editing by DNA cytosine deaminase APOBEC3B modulates the activity of oestrogen receptor enhancers.

DNA胞嘧啶脱氨酶APOBEC3B对R环的编辑调节雌激素受体增强子的活性。

Zhang Chi, Lu Yu-Jing, Chen Bingjie, Bai Zhiyan, Zeng Qiaoxi, Hervieu Alexia, Licciardello Marco P, Mitsopoulos Konstantinos, Al-Lazikani Bissan, Tortorici Marcello, Rossanese Olivia W, Workman Paul, Clarke Paul A

Intracameral Cefuroxime Use in Cataract Surgery After Penicillin Allergy Reclassification

青霉素过敏重新分类后,白内障手术中使用前房注射头孢呋辛

Reddy, Karthik; Workman, Paul; Eschenauer, Greg; Bixler, Jill; Mian, Shahzad I

Unhooking the Hook: Optimization of the Aurora A Targeting PROTAC JB170 to CCT400028, an In Vitro Degrader Chemical Probe

解开钩子:优化 Aurora A 靶向 PROTAC JB170 至 CCT400028,一种体外降解化学探针

O'Hanlon, Jack A; Gutsche, Katrin; Müller, Juliane Elisabeth; Ranjan Prusty, Nihar; Mirza, Amin; Roumeliotis, Theodoros I; Yang, Hengzhang; Stubbs, Mark; Hallett, Stephen T; Eing, Lorenz; McAndrew, Peter Craig; Choudhary, Jyoti Sharma; Le Bihan, Yann-Vaï; Caldwell, John; van Montfort, Rob L M; Workman, Paul; Wolf, Elmar; Newton, Gary K; Evans, Lindsay E

Human DEAH-box helicase 8 regulates HSF1-mediated stress response and cancer-associated pre-mRNA splicing in tumour cells.

人类 DEAH 盒解旋酶 8 调节 HSF1 介导的应激反应和肿瘤细胞中与癌症相关的 pre-mRNA 剪接。

Tall Jennifer R, Te Poele Robert, Vasile Alexandra, Ramagiri Pradeep, Campbell James, Davies Caitlin R, Powers Marissa V, Roe Toby, Sankaran Deivendran, Wang Hannah, Mitsopoulos Konstantinos, Al-Lazikani Bissan, van Montfort Rob L M, de Billy Emmanuel, Workman Paul, Clarke Paul A

Structural insights into human brachyury DNA recognition and discovery of progressible binders for cancer therapy

对人类短尾蛋白DNA识别的结构性见解以及用于癌症治疗的新型结合剂的发现

Newman, Joseph A; Gavard, Angeline E; Imprachim, Nergis; Aitkenhead, Hazel; Sheppard, Hadley E; Te Poele, Robert; Clarke, Paul A; Hossain, Mohammad Anwar; Temme, Louisa; Oh, Hans J; Wells, Carrow I; Davis-Gilbert, Zachary W; Workman, Paul; Gileadi, Opher; Drewry, David H

canSAR 2024-an update to the public drug discovery knowledgebase

canSAR 2024——公共药物发现知识库的更新

Gingrich, Phillip W; Chitsazi, Rezvan; Biswas, Ansuman; Jiang, Chunjie; Zhao, Li; Tym, Joseph E; Brammer, Kevin M; Li, Jun; Shu, Zhigang; Maxwell, David S; Tacy, Jeffrey A; Mica, Ioan L; Darkoh, Michael; di Micco, Patrizio; Russell, Kaitlyn P; Workman, Paul; Al-Lazikani, Bissan

The Chemical Probes Portal - 2024: update on this public resource to support best-practice selection and use of small molecules in biomedical research

化学探针门户网站 - 2024:更新此公共资源,以支持生物医学研究中小分子的最佳实践选择和使用

Sanfelice, Domenico; Antolin, Albert A; Crisp, Alisa; Chen, Yi; Bellenie, Benjamin; Brennan, Paul E; Edwards, Aled; Müller, Susanne; Al-Lazikani, Bissan; Workman, Paul

Mediator Kinase Inhibitor Selectivity and Activity in Colorectal Cancer

介导激酶抑制剂在结直肠癌中的选择性和活性

Ortiz-Ruiz, Maria J; Popoola, Olajumoke; Mitsopoulos, Konstantinos; Te-Poele, Robert; Samant, Rahul S; Box, Gary; Court, Will; Brandon, Alexis De Haven; Gowan, Sharon; Mallinger, Aurelie; Roe, Toby; Swabey, Kate; Valenti, Melanie; Al-Lazikani, Bissan; Blagg, Julian; Esdar, Christina; Schiemann, Kai; Wienke, Dirk; Eccles, Suzanne A; Workman, Paul; Clarke, Paul A

canSAR: update to the cancer translational research and drug discovery knowledgebase

canSAR:癌症转化研究和药物发现知识库的更新

di Micco, Patrizio; Antolin, Albert A; Mitsopoulos, Costas; Villasclaras-Fernandez, Eloy; Sanfelice, Domenico; Dolciami, Daniela; Ramagiri, Pradeep; Mica, Ioan L; Tym, Joseph E; Gingrich, Philip W; Hu, Huabin; Workman, Paul; Al-Lazikani, Bissan

The Chemical Probes Portal: an expert review-based public resource to empower chemical probe assessment, selection and use

化学探针门户网站:一个基于专家评审的公共资源,旨在促进化学探针的评估、选择和使用。

Antolin, Albert A; Sanfelice, Domenico; Crisp, Alisa; Villasclaras Fernandez, Eloy; Mica, Ioan L; Chen, Yi; Collins, Ian; Edwards, Aled; Müller, Susanne; Al-Lazikani, Bissan; Workman, Paul