日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Inhibiting peptidylarginine deiminases (PAD1-4) by targeting a Ca(2+) dependent allosteric binding site.

通过靶向 Ca(2+) 依赖性变构结合位点来抑制肽基精氨酸脱亚胺酶 (PAD1-4)

Dakin Leslie A, Xing Li, Hall Justin, Ding Weidong, Vajdos Felix F, Pelker Jeffrey W, Ramsey Simeon, Balbo Paul, Sahasrabudhe Parag V, Banker Mary Ellen, Choi Won Young, Wright Stephen W, Chang Jeanne S, Curto John M, Davoren Jennifer E, Drozda Susan E, Fennell Kimberly F, Futatsugi Kentaro, Kortum Steve, Lee Katherine L, Liu Shenping, Lovering Frank, Nicki Jennifer A, Trujillo John I, Vincent Fabien, Schnute Mark E

Peptidylarginine Deiminase (PAD) Inhibitor Optimization through Displacement of a Trapped Water Molecule

通过置换被捕获的水分子来优化肽基精氨酸脱亚胺酶(PAD)抑制剂

Schnute, Mark E; Chinigo, Gary M; Futatsugi, Kentaro; Yamaguchi, Masaya; Bagley, Scott W; Banker, Mary Ellen; Chang, Jeanne S; Chen, Ming Z; Choi, Won Young; Corbett, Matthew S; Drozda, Susan E; Ebner, David C; Garcia-Irizarry, Carmen; Hicklin, Robert; Hoy, Susan; Jiao, Wenhua; Kortum, Steven; Lee, Katherine L; Limburg, David C; Lovering, Frank; Moreno, Antonio; Mousseau, James J; Pan, Senliang; Parikh, Mihir D; Pelker, Jeffrey W; Ramsey, Simeon; Reilly, Usa; Rescourio, Gwenaella; Schmitt, Daniel C; Simpson, Brittany; Skrzypek, Grzegorz J; Smaltz, Daniel J; Taylor, Alexandria P; Torella, Rubben; Trujillo, John I; Vajdos, Felix F; Wepy, James A; Wright, Stephen W; Blakemore, David C; Vincent, Fabien; Clerin, Valerie M

In Retrospect: Root-Cause Analysis of Structure-Activity Relationships in IRAK4 Inhibitor Zimlovisertib (PF-06650833)

回顾:IRAK4抑制剂Zimlovisertib(PF-06650833)结构-活性关系的根本原因分析

Wright, Stephen W; Farley, Kathleen A; Han, Seungil; Knafels, John D; Lee, Katherine L

Synthesis of Deuterated Enaminones with High Isotopic Fidelity

高同位素保真度氘代烯胺酮的合成

Wright, Stephen W

Synthesis of Deuterated Heterocycles with Me(2)NCD(OMe)(2) and Evaluation of the Products for Metabolism by Aldehyde Oxidase

利用Me(2)NCD(OMe)2合成氘代杂环化合物并评价其醛氧化酶代谢活性

Choi, Chulho; Carlo, Anthony A; Cronin, Ciarán N; Jing, Konghua; Kung, Daniel W; Liu, Jianhua; Lombardo, Vincent M; Turco, Abigail R; Yin, Juxing; Yu, Aijia; Wright, Stephen W

Lithium Enolates Derived from Pyroglutaminol: Aggregation, Solvation, and Atropisomerism

源自焦谷氨酰胺醇的锂烯醇化物:聚集、溶剂化和阻转异构现象

Houghton, Michael J; Biok, Naomi A; Huck, Christopher J; Algera, Russell F; Keresztes, Ivan; Wright, Stephen W; Collum, David B