日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Library docking for Cannabinoid-2 Receptor ligands

大麻素-2受体配体的库对接

Rachman, Moira M; Iliopoulos-Tsoutsouvas, Christos; Sacco, Michael D; Xu, Xinyu; Wu, Cheng-Guo; Santos, Emma; Glenn, Isabella S; Paris, Lu; Cahill, Michelle K; Ganapathy, Suthakar; Tummino, Tia A; Moroz, Yurii S; Radchenko, Dmytro S; Okorie, Meri; Tawfik, Vivianne; Irwin, John J; Makriyannis, Alexandros; Skiniotis, Georgios; Shoichet, Brian K

Structural insight into the catalytic mechanism of the bifunctional enzyme l-fucokinase/GDP-fucose pyrophosphorylase

对双功能酶L-岩藻糖激酶/GDP-岩藻糖焦磷酸化酶催化机制的结构解析

Lin, Sheng-Wei; Ko, Tzu-Ping; Chiang, Hung-Yu; Wu, Cheng-Guo; Hsu, Min-Feng; Wang, Andrew H-J; Lin, Chun-Hung

Allosteric modulation and G-protein selectivity of the Ca(2+)-sensing receptor.

Ca(2+)敏感受体的变构调节和G蛋白选择性

He Feng, Wu Cheng-Guo, Gao Yang, Rahman Sabrina N, Zaoralová Magda, Papasergi-Scott Makaía M, Gu Ting-Jia, Robertson Michael J, Seven Alpay B, Li Lingjun, Mathiesen Jesper M, Skiniotis Georgios

Large library docking identifies positive allosteric modulators of the calcium-sensing receptor.

大型化合物库对接鉴定出钙敏感受体的正向变构调节剂

Liu Fangyu, Wu Cheng-Guo, Tu Chia-Ling, Glenn Isabella, Meyerowitz Justin, Kaplan Anat Levit, Lyu Jiankun, Cheng Zhiqiang, Tarkhanova Olga O, Moroz Yurii S, Irwin John J, Chang Wenhan, Shoichet Brian K, Skiniotis Georgios

Small vs. Large Library Docking for Positive Allosteric Modulators of the Calcium Sensing Receptor.

钙敏感受体正向变构调节剂的小分子与大分子库对接

Liu Fangyu, Wu Cheng-Guo, Tu Chia-Ling, Glenn Isabella, Meyerowitz Justin, Levit Kaplan Anat, Lyu Jiankun, Cheng Zhiqiang, Tarkhanova Olga O, Moroz Yurii S, Irwin John J, Chang Wenhan, Shoichet Brian K, Skiniotis Georgios

Disease mutations and phosphorylation alter the allosteric pathways involved in autoinhibition of protein phosphatase 2A.

疾病突变和磷酸化改变了参与蛋白磷酸酶 2A 自身抑制的变构途径

Konovalov Kirill A, Wu Cheng-Guo, Qiu Yunrui, Balakrishnan Vijaya Kumar, Parihar Pankaj Singh, O'Connor Michael S, Xing Yongna, Huang Xuhui

A comprehensive genome-wide analysis of long non-coding RNA and mRNA expression profiles of JAK2V617F-positive classical myeloproliferative neoplasms

JAK2V617F 阳性经典骨髓增生性肿瘤的长链非编码 RNA 和 mRNA 表达谱的全面全基因组分析

Jie Zhou, Hao Wu, Cheng Guo, Bing Li, Li-Li Zhou, Ai-Bin Liang, Jian-Fei Fu

Structure of a Highly Active Cephalopod S-crystallin Mutant: New Molecular Evidence for Evolution from an Active Enzyme into Lens-Refractive Protein

高活性头足类S-晶状体蛋白突变体的结构:从活性酶进化为晶状体折射蛋白的新分子证据

Tan, Wei-Hung; Cheng, Shu-Chun; Liu, Yu-Tung; Wu, Cheng-Guo; Lin, Min-Han; Chen, Chiao-Che; Lin, Chao-Hsiung; Chou, Chi-Yuan

Interleukin-13 suppresses interleukin-10 via inhibiting A20 in peripheral B cells of patients with food allergy

白细胞介素-13通过抑制食物过敏患者外周血B细胞中的A20来抑制白细胞介素-10。

Li, Ming-Yang; Zhu, Min; Linghu, En-Qiang; Feng, Fan; Zhu, Bing; Wu, Cheng; Guo, Ming-Zhou

Cathepsin K-mediated Notch1 activation contributes to neovascularization in response to hypoxia

组织蛋白酶 K 介导的 Notch1 激活促进缺氧引起的新血管形成

Haiying Jiang, Xian Wu Cheng, Guo-Ping Shi, Lina Hu, Aiko Inoue, Yumiko Yamamura, Hongxian Wu, Kyosuke Takeshita, Xiang Li, Zhe Huang, Haizhen Song, Masashi Asai, Chang-Ning Hao, Kazumasa Unno, Teruhiro Koike, Yoshiharu Oshida, Kenji Okumura, Toyoaki Murohara, Masafumi Kuzuya