日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Thymol carbamates bearing cyclic amines as potent and selective BuChE inhibitors alleviate memory impairments for Alzheimer's disease therapy

含有环状胺的百里酚氨基甲酸酯作为强效且选择性的丁酰胆碱酯酶抑制剂,可缓解阿尔茨海默病治疗中的记忆障碍。

Wu, Chengyao; Ding, Yulu; Liu, Xiaodan; Gao, Shan; Wang, Xiaoqing; Tang, Wenjian

Structure of the priming arabinosyltransferase AftA required for AG biosynthesis of Mycobacterium tuberculosis

结核分枝杆菌AG生物合成所需的启动阿拉伯糖基转移酶AftA的结构

Gong, Yicheng; Wei, Chuancun; Wang, Jun; Mu, Nengjiang; Lu, Qinhong; Wu, Chengyao; Yan, Ning; Yang, Huifang; Zhao, Yao; Yang, Xiuna; Gurcha, Sudagar S; Veerapen, Natacha; Batt, Sarah M; Hao, Zhiqiang; Da, Lintai; Besra, Gurdyal S; Rao, Zihe; Zhang, Lu

Microtiter plate-based chemistry and in situ screening: SuFEx-enabled lead discovery of selective AChE inhibitors

基于微孔板的化学方法和原位筛选:SuFEx技术助力选择性AChE抑制剂的先导化合物发现

Tang, Kun; Li, Huan-Huan; Wu, Chengyao; Zhang, Shi-Long; Yang, Jian-Guo; Tang, Wenjian; Qin, Hua-Li

Fluorosulfate-containing pyrazole heterocycles as selective BuChE inhibitors: structure-activity relationship and biological evaluation for the treatment of Alzheimer's disease.

含氟硫酸盐的吡唑杂环化合物作为选择性丁酰胆碱酯酶抑制剂:结构活性关系及治疗阿尔茨海默病的生物学评价

Li Huan-Huan, Wu Chengyao, Zhang Shi-Long, Yang Jian-Guo, Qin Hua-Li, Tang Wenjian

Structure-activity relationship, in vitro and in vivo evaluation of novel dienyl sulphonyl fluorides as selective BuChE inhibitors for the treatment of Alzheimer's disease.

新型二烯基磺酰氟化物作为选择性丁酰胆碱酯酶抑制剂治疗阿尔茨海默病的结构活性关系、体外和体内评价

Wu Chengyao, Zhang Guijuan, Zhang Zai-Wei, Jiang Xia, Zhang Ziwen, Li Huanhuan, Qin Hua-Li, Tang Wenjian