N-Arylsulfonyl-α-amino carboxamides are potent and selective inhibitors of the chemokine receptor CCR10 that show efficacy in the murine DNFB model of contact hypersensitivity
N-芳基磺酰基-α-氨基甲酰胺是趋化因子受体 CCR10 的强效选择性抑制剂,在小鼠 DNFB 接触性超敏反应模型中表现出疗效
期刊:Bioorganic & Medicinal Chemistry Letters
影响因子:2.5
doi:10.1016/j.bmcl.2016.09.047
Asitha Abeywardane, Gary Caviness, Younggi Choi, Derek Cogan, Amy Gao, Daniel Goldberg, Alexander Heim-Riether, Debra Jeanfavre, Elliott Klein, Jennifer A Kowalski, Wang Mao, Craig Miller, Neil Moss, Philip Ramsden, Ernest Raymond, Donna Skow, Lana Smith-Keenan, Roger J Snow, Frank Wu, Jiang-Ping Wu